ES341324A1 - Un procedimiento para la preparacion de pirazinoilguanidi- nas y pirazinamidoguanidinas. - Google Patents

Un procedimiento para la preparacion de pirazinoilguanidi- nas y pirazinamidoguanidinas.

Info

Publication number
ES341324A1
ES341324A1 ES341324A ES341324A ES341324A1 ES 341324 A1 ES341324 A1 ES 341324A1 ES 341324 A ES341324 A ES 341324A ES 341324 A ES341324 A ES 341324A ES 341324 A1 ES341324 A1 ES 341324A1
Authority
ES
Spain
Prior art keywords
alkyl
phenyl
hydrogen
general formula
pyrazinamido
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES341324A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of ES341324A1 publication Critical patent/ES341324A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D241/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ES341324A 1966-08-25 1967-06-02 Un procedimiento para la preparacion de pirazinoilguanidi- nas y pirazinamidoguanidinas. Expired ES341324A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57492266A 1966-08-25 1966-08-25

Publications (1)

Publication Number Publication Date
ES341324A1 true ES341324A1 (es) 1968-10-01

Family

ID=24298194

Family Applications (1)

Application Number Title Priority Date Filing Date
ES341324A Expired ES341324A1 (es) 1966-08-25 1967-06-02 Un procedimiento para la preparacion de pirazinoilguanidi- nas y pirazinamidoguanidinas.

Country Status (8)

Country Link
BE (1) BE699438A (de)
CH (1) CH487169A (de)
DE (1) DE1695421A1 (de)
ES (1) ES341324A1 (de)
GB (1) GB1145934A (de)
IL (1) IL27897A (de)
NL (1) NL6707570A (de)
SE (1) SE333146B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6858615B2 (en) 2002-02-19 2005-02-22 Parion Sciences, Inc. Phenyl guanidine sodium channel blockers
EA017919B1 (ru) 2007-12-10 2013-04-30 Новартис Аг Производные пиразин-2-карбоксамида для лечения заболеваний, которые поддаются лечению путем блокирования эпителиальных натриевых каналов
AR086745A1 (es) 2011-06-27 2014-01-22 Parion Sciences Inc 3,5-diamino-6-cloro-n-(n-(4-(4-(2-(hexil(2,3,4,5,6-pentahidroxihexil)amino)etoxi)fenil)butil)carbamimidoil)pirazina-2-carboxamida
PE20151054A1 (es) 2012-12-17 2015-08-07 Parion Sciences Inc Derivados de cloro-pirazin carboxamida con actividad bloqueadora sobre los canales de sodio epiteliales
MX2015007797A (es) 2012-12-17 2015-10-05 Parion Sciences Inc Compuestos de 3,5-diamino-6-cloro-n-(n-(4-fenilbutil) carbamimidoil) pirazin-2-carboxamida.
US9102633B2 (en) 2013-12-13 2015-08-11 Parion Sciences, Inc. Arylalkyl- and aryloxyalkyl-substituted epithelial sodium channel blocking compounds

Also Published As

Publication number Publication date
SE333146B (sv) 1971-03-08
GB1145934A (en) 1969-03-19
BE699438A (de) 1967-12-04
NL6707570A (de) 1968-02-26
IL27897A (en) 1972-02-29
DE1695421A1 (de) 1971-04-15
CH487169A (de) 1970-03-15

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