ES417233A2 - Procedure for preparation of new heterocidal organofosforated derivatives. (Machine-translation by Google Translate, not legally binding) - Google Patents
Procedure for preparation of new heterocidal organofosforated derivatives. (Machine-translation by Google Translate, not legally binding)Info
- Publication number
- ES417233A2 ES417233A2 ES417233A ES417233A ES417233A2 ES 417233 A2 ES417233 A2 ES 417233A2 ES 417233 A ES417233 A ES 417233A ES 417233 A ES417233 A ES 417233A ES 417233 A2 ES417233 A2 ES 417233A2
- Authority
- ES
- Spain
- Prior art keywords
- pyrimidine
- carbon atoms
- dihydro
- dimethoxythiophosphoryloxy
- dihydropyrrolo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 238000000034 method Methods 0.000 title abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 9
- -1 diethoxythiophosphoryloxy Chemical group 0.000 abstract 8
- 150000001875 compounds Chemical class 0.000 abstract 4
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- 239000011593 sulfur Substances 0.000 abstract 2
- VTCKWMWUPMBCLU-UHFFFAOYSA-N C(C)OP(=S)(OCC)OC1=NC=CCCC1 Chemical compound C(C)OP(=S)(OCC)OC1=NC=CCCC1 VTCKWMWUPMBCLU-UHFFFAOYSA-N 0.000 abstract 1
- DRUCUKPOWLETMB-UHFFFAOYSA-N COP(=S)(OC)OC1=NC=2N(C(C1)=O)C=CC=CC=2 Chemical compound COP(=S)(OC)OC1=NC=2N(C(C1)=O)C=CC=CC=2 DRUCUKPOWLETMB-UHFFFAOYSA-N 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 125000003158 alcohol group Chemical group 0.000 abstract 1
- 125000003277 amino group Chemical group 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 125000004434 sulfur atom Chemical group 0.000 abstract 1
Abstract
Improvements introduced in the object of the main patent no. 406,728 requested on september 15, 1972 by: "a procedure for preparing new heterocyclic organophosphorus derivatives", to: a) obtain new compounds corresponding to formula i of the products obtained in the main patent, characterized in that 2- (dimethoxythiophosphoryloxy) -4,5-dihydro-azepino- [1,2-a] -pyrimidine-4-one, 2- (diethoxythiophosphoryloxy) -4,5-dihydro-azepine are obtained - [1,2-a] -pyrimidine-4-one, 2- (diethoxythiophosphoryloxy) -3-isopropyl-4,5-dihydro-azepino [1,2-a] -pyrimidine-4-one, 2- (dimethoxythiophosphoryloxy) - [6 h] -7,8-dihydropyrrolo- [1,2-a] -pyrimidine-4-one, 2,5-dibydro-7- (dimethoxythiophosphoryloxy) -thiazolo- [3,2-a] ] -pyrimidine-5-one, 2- (diethoxyphosphoryloxy) -4,5-dihydro-azepino- [1,2-a] -pyrimidine-4-one, 2- (diethoxythiophosphoryloxy) -6,7,8, 9-tetrahydropyrido- [1,2-a] -pyrimidine-4-one, 2- (dimethoxythiophosphoryloxy) -6,7,8,9-tetrahydropyrido-] 1,2-a] -pyrimidine-4-one, 2- (o-methyl-o- ethylthiophosphoryloxy) - [6 h] -7,8-dihydropyrrolo- [1,2-a] -pyrimidine-4-one, 2- (o-ethyl-N-isopropylaminothiophosphoramido-oxy) - [6 h] -7, 8-dihydro [1,2-a] -pyrrolopyrimidin-4-one, 2- (dipropyloxythiophosphoryloxy) - [6 h] -7,8-dihydropyrrolo- [1,2-a] -pyrimidine-4-one, and 2- (diisopropyloxythiophosphoryloxy) - [6 h] -7,8-dihydropyrrolo- [1,2-a] -pyrimidin-4-one; b) obtain compounds related to those of the main patent, of general formula i ': (see formula) Where a represents an alcohol chain comprising from 3 to 5 carbon atoms, optionally interrupted by a heteroatom chosen from sulfur and nitrogen, x represents a sulfur or oxygen atom, y 'represents a hydrogen atom or an alcohol radical comprising from 1 to 6 carbon atoms, linear or branched, a cyano group, a halogen, or an alcoholyl group whose alkyl radical comprises from 1 to 6 carbon atoms, r''1 represents an alkyl radical, linear or branched, comprising 1 to 4 carbon atoms, r "2 represents an alkyl radical, linear or branched, comprising from 1 to 4 carbon atoms and optionally substituted by an alkoxy radical comprising from 1 to 4 carbon atoms, or r "2 represents an alkoxy radical comprising from 1 to 4 carbon atoms and optionally substituted by an alkoxy radical comprising from 1 to 4 carbon atoms, or r" 2 represents an amino group (see formula) in the that r'1 and r'2, analogous or different, represent a hydrogen atom or a linear or branched alkyl radical, comprising from 1 to 3 carbon atoms, with the exception of the compounds corresponding to the general formula of the spanish principal patent no. 406,728, other than the compounds listed above. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7230885A FR2199694A5 (en) | 1971-09-02 | 1972-08-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES417233A2 true ES417233A2 (en) | 1977-06-01 |
Family
ID=9103727
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES417233A Expired ES417233A2 (en) | 1972-08-31 | 1973-07-24 | Procedure for preparation of new heterocidal organofosforated derivatives. (Machine-translation by Google Translate, not legally binding) |
Country Status (1)
| Country | Link |
|---|---|
| ES (1) | ES417233A2 (en) |
-
1973
- 1973-07-24 ES ES417233A patent/ES417233A2/en not_active Expired
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES456575A1 (en) | 2,3-dihydro-imidazo(2,1-b)-thiazole derivatives and applications thereof | |
| ES457993A1 (en) | Isothiazolo-pyridines | |
| ES369479A1 (en) | (1)benzothieno(2 3-d)pyrimidine derivatives | |
| ES454823A1 (en) | Derivatives of imidazo 1,2-a pyridine | |
| ES417233A2 (en) | Procedure for preparation of new heterocidal organofosforated derivatives. (Machine-translation by Google Translate, not legally binding) | |
| ES462685A1 (en) | Rifamycin compounds | |
| ES451466A1 (en) | 5-thiazole-methane-amines, and their use as antilipolytics | |
| ES383467A1 (en) | Procedure for the preparation of pirrol derivatives. (Machine-translation by Google Translate, not legally binding) | |
| ES392364A1 (en) | 7-phenylpyrimido-benzodiazepine derivatives | |
| ES480561A1 (en) | Bridged catharanthus alkaloid dimers, their preparation and formulations containing them. | |
| ES460853A1 (en) | Procedure for the preparation of pirrolo (2,3-d) pyrimidine-2,4-diona derivatives. (Machine-translation by Google Translate, not legally binding) | |
| ES393953A1 (en) | Benzodiazepines and process for their manufacture | |
| ES462845A1 (en) | A procedure for the preparation of compounds imidazo (1,5-a) (1,4) diacepidinicos (Machine-translation by Google Translate, not legally binding) | |
| ES461191A1 (en) | New nn**11piperidinyl*alkyl* aryl carboxysamide derivative | |
| IL90172A (en) | 2,3-dihydro-5-(substituted phenyl)-imidazo(1,2-a)furo and thieno pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
| ES431477A1 (en) | Procedure for preparing glycerol derivatives. (Machine-translation by Google Translate, not legally binding) | |
| ES460855A1 (en) | Procedure for the preparation of pirrolo (2,3-d) pyrimidine-2,4-diona derivatives. (Machine-translation by Google Translate, not legally binding) | |
| JPS51118784A (en) | Method for preparing thienodiazepine derivatives | |
| ES459331A1 (en) | Procedure for preparation of derivatives of tetrahidro-1,5,10,10a-tiazol (3,4-b) isoquinoleina. (Machine-translation by Google Translate, not legally binding) | |
| ES462656A1 (en) | A procedure for the preparation of cefalosporine derivatives. (Machine-translation by Google Translate, not legally binding) | |
| ES405913A3 (en) | Procedure for the preparation of derivatives of alcohilxantina basically substituted. (Machine-translation by Google Translate, not legally binding) | |
| ES438557A1 (en) | A procedure for the preparation of new tiazol derivatives. (Machine-translation by Google Translate, not legally binding) | |
| ES403885A1 (en) | A procedure for preparing derivatives substituted in n 'of N- (trimetoxy-3,4,5) cinamoil-piperazine. (Machine-translation by Google Translate, not legally binding) | |
| ES470709A3 (en) | Procedure for the manufacture of heterociclic derivatives (Machine-translation by Google Translate, not legally binding) | |
| ES459332A1 (en) | Procedure for preparation of derivatives of tetrahidro-1,5,10,10a-tiazol (3,4-b) isoquinoleina. (Machine-translation by Google Translate, not legally binding) |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD2A | Announcement of lapse in spain |
Effective date: 20170704 |