ES441002A1 - A PROCEDURE FOR PREPARING OXAPROSTAGLANDINS. - Google Patents

A PROCEDURE FOR PREPARING OXAPROSTAGLANDINS.

Info

Publication number
ES441002A1
ES441002A1 ES441002A ES441002A ES441002A1 ES 441002 A1 ES441002 A1 ES 441002A1 ES 441002 A ES441002 A ES 441002A ES 441002 A ES441002 A ES 441002A ES 441002 A1 ES441002 A1 ES 441002A1
Authority
ES
Spain
Prior art keywords
formula
oxaprostaglandins
procedure
compound
ligation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES441002A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/355,644 external-priority patent/US4094899A/en
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES441002A1 publication Critical patent/ES441002A1/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/93Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
    • C07D307/935Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10Oxygen atoms
    • C07D309/12Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

A procedure to prepare oxaprostaglandins of the following structure: ** (See formula) ** in which R is hydrogen or an alkyl of 1 to 3 carbon atoms; W is a single tie or a double cis tie; Z is a single ligation or a double trans ligation; n is an integer from 0 to 2 and m is an integer ranging from 1 to 5, provided that the sum of n and m does not exceed 6, and THP is 2-tetrahydropyranil; characterized by the fact that: a compound of the formula is reacted: ** (See formula) ** with an iluro of the formula (C6H5) 3P = CH-CH2CH2CH2-COOH and, when required, subsequently reduce the product thus formed to yield a compound in which: n, m R and Z represent what is indicated above and W is a single bond. (Machine-translation by Google Translate, not legally binding)
ES441002A 1972-06-02 1975-09-16 A PROCEDURE FOR PREPARING OXAPROSTAGLANDINS. Expired ES441002A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25921572A 1972-06-02 1972-06-02
US05/355,644 US4094899A (en) 1972-06-02 1973-04-30 Oxaprostaglandins

Publications (1)

Publication Number Publication Date
ES441002A1 true ES441002A1 (en) 1977-03-01

Family

ID=26947161

Family Applications (2)

Application Number Title Priority Date Filing Date
ES441002A Expired ES441002A1 (en) 1972-06-02 1975-09-16 A PROCEDURE FOR PREPARING OXAPROSTAGLANDINS.
ES441003A Expired ES441003A1 (en) 1972-06-02 1975-09-16 Oxaprostaglandins

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES441003A Expired ES441003A1 (en) 1972-06-02 1975-09-16 Oxaprostaglandins

Country Status (19)

Country Link
JP (3) JPS5314062B2 (en)
AR (2) AR199300A1 (en)
CA (1) CA1095034A (en)
CH (3) CH586716A5 (en)
DD (2) DD109859A5 (en)
DE (2) DE2327813A1 (en)
DK (1) DK143498C (en)
ES (2) ES441002A1 (en)
FI (1) FI55995C (en)
GB (3) GB1440603A (en)
IE (1) IE38568B1 (en)
IL (2) IL42373A (en)
IN (1) IN138739B (en)
LU (1) LU67738A1 (en)
NL (1) NL162902C (en)
NO (1) NO145438C (en)
PH (3) PH11300A (en)
SE (4) SE415756B (en)
YU (1) YU36497B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES416865A1 (en) * 1972-07-13 1976-03-01 Pfizer 15-substituted-omega-pentanorprostaglandins
US11756356B2 (en) 2019-08-28 2023-09-12 Igloocompany Pte. Ltd. System and method for controlling multiple locks

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3538120A (en) * 1967-05-22 1970-11-03 Ciba Geigy Corp Cyclopentyl-alkanoic acids
ZA721159B (en) * 1971-03-22 1972-12-27 Ici Ltd Process for the separation of the c-15 epimers of 20-ethyl-9a,11alpha,15-trihydroxy-5-cis-13-trans-prostadienoic acid

Also Published As

Publication number Publication date
AU5639373A (en) 1974-12-05
JPS5231054A (en) 1977-03-09
JPS5728706B2 (en) 1982-06-18
DE2344839B2 (en) 1976-06-24
PH11931A (en) 1978-09-13
FI55995C (en) 1979-11-12
YU146973A (en) 1982-02-25
DE2344838C3 (en) 1982-03-18
SE418857B (en) 1981-06-29
NL7307740A (en) 1973-12-04
JPS4954349A (en) 1974-05-27
DD124594A5 (en) 1977-03-02
PH12035A (en) 1978-10-16
DK143498C (en) 1982-01-11
IE38568L (en) 1973-12-02
GB1440603A (en) 1976-06-23
LU67738A1 (en) 1973-12-10
JPS5314062B2 (en) 1978-05-15
DE2344839A1 (en) 1974-02-28
DE2344838B2 (en) 1981-04-09
DD109859A5 (en) 1974-11-20
JPS5239629A (en) 1977-03-28
CH589074A5 (en) 1977-06-30
SE7608222L (en) 1976-07-19
AR199300A1 (en) 1974-08-23
DK143498B (en) 1981-08-31
DE2327813A1 (en) 1973-12-20
GB1440601A (en) 1976-06-23
IL42373A0 (en) 1973-07-30
NO740849L (en) 1973-12-04
ES441003A1 (en) 1977-03-16
SE415756B (en) 1980-10-27
CA1095034A (en) 1981-02-03
FI55995B (en) 1979-07-31
PH11300A (en) 1977-11-02
NO145438B (en) 1981-12-14
GB1440602A (en) 1976-06-23
IL42373A (en) 1977-08-31
IE38568B1 (en) 1978-04-12
CH590224A5 (en) 1977-07-29
IL50311A (en) 1977-08-31
NO145438C (en) 1982-03-24
CH586716A5 (en) 1977-04-15
NL162902C (en) 1980-07-15
YU36497B (en) 1984-02-29
SE7608221L (en) 1976-07-19
NL162902B (en) 1980-02-15
IN138739B (en) 1976-03-27
SE7608223L (en) 1976-07-19
DE2344838A1 (en) 1973-12-20
AR203386A1 (en) 1975-09-08

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