ES447063A1 - Procedimiento para la produccion de pirazolas-(5) 1-susti- tuidas. - Google Patents

Procedimiento para la produccion de pirazolas-(5) 1-susti- tuidas.

Info

Publication number: ES447063A1
Authority: ES; Spain
Prior art keywords: alkyl; radical; alkenyl; substituted; trifluoromethyl
Prior art date: 1973-04-17
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

ES447063A

Other languages

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer AG

Original Assignee

Bayer AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-04-17

Filing date

1976-04-15

Publication date

1977-06-16

1973-04-17 Priority claimed from DE2319280A external-priority patent/DE2319280A1/de

1973-12-19 Priority claimed from DE2363139A external-priority patent/DE2363139A1/de

1976-04-15 Application filed by Bayer AG filed Critical Bayer AG

1977-06-16 Publication of ES447063A1 publication Critical patent/ES447063A1/es

Status Expired legal-status Critical Current

Links

JEXVQSWXXUJEMA-UHFFFAOYSA-N pyrazol-3-one Chemical class O=C1C=CN=N1 JEXVQSWXXUJEMA-UHFFFAOYSA-N 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 5
125000003342 alkenyl group Chemical group 0.000 abstract 4
-1 carbonamido Chemical group 0.000 abstract 4
125000003545 alkoxy group Chemical group 0.000 abstract 3
229910052736 halogen Inorganic materials 0.000 abstract 3
150000002367 halogens Chemical class 0.000 abstract 3
125000001424 substituent group Chemical group 0.000 abstract 3
125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 3
QGZKDVFQNNGYKY-UHFFFAOYSA-N Ammonia Chemical compound N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
125000003282 alkyl amino group Chemical group 0.000 abstract 1
125000004414 alkyl thio group Chemical group 0.000 abstract 1
229910021529 ammonia Inorganic materials 0.000 abstract 1
125000003710 aryl alkyl group Chemical class 0.000 abstract 1
125000003118 aryl group Chemical class 0.000 abstract 1
150000005840 aryl radicals Chemical class 0.000 abstract 1
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
125000004093 cyano group Chemical group *C#N 0.000 abstract 1
125000000623 heterocyclic group Chemical group 0.000 abstract 1
239000012442 inert solvent Substances 0.000 abstract 1
238000004519 manufacturing process Methods 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
229910052760 oxygen Inorganic materials 0.000 abstract 1
239000001301 oxygen Substances 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
150000003254 radicals Chemical class 0.000 abstract 1
229920006395 saturated elastomer Polymers 0.000 abstract 1
125000003107 substituted aryl group Chemical group 0.000 abstract 1
125000005420 sulfonamido group Chemical group S(=O)(=O)(N*)* 0.000 abstract 1
125000004434 sulfur atom Chemical group 0.000 abstract 1
125000000876 trifluoromethoxy group Chemical group FC(F)(F)O* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
- C07D231/24—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms having sulfone or sulfonic acid radicals in the molecule
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
- C07D231/52—Oxygen atom in position 3 and nitrogen atom in position 5, or vice versa

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Hematology (AREA)
Diabetes (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Catalysts (AREA)

ES447063A 1973-04-17 1976-04-15 Procedimiento para la produccion de pirazolas-(5) 1-susti- tuidas. Expired ES447063A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE2319280A DE2319280A1 (de)	1973-04-17	1973-04-17	1-substituierte pyrazolone-(5), verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
DE2363139A DE2363139A1 (de)	1973-12-19	1973-12-19	1-substituierte pyrazolone-(5), verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Publications (1)

Publication Number	Publication Date
ES447063A1 true ES447063A1 (es)	1977-06-16

Family

ID=25764996

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
ES425373A Expired ES425373A1 (es)	1973-04-17	1974-04-16	Procedimiento para la produccion de pirazolonas-(5) 1-sus- tituidas.
ES447064A Expired ES447064A1 (es)	1973-04-17	1976-04-15	Procedimiento para la produccion de pirazolonas-(5) 1-susti-tuidas.
ES447063A Expired ES447063A1 (es)	1973-04-17	1976-04-15	Procedimiento para la produccion de pirazolas-(5) 1-susti- tuidas.

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
ES425373A Expired ES425373A1 (es)	1973-04-17	1974-04-16	Procedimiento para la produccion de pirazolonas-(5) 1-sus- tituidas.
ES447064A Expired ES447064A1 (es)	1973-04-17	1976-04-15	Procedimiento para la produccion de pirazolonas-(5) 1-susti-tuidas.

Country Status (27)

Country	Link
US (1)	US3957814A (es)
JP (1)	JPS5314071B2 (es)
AR (5)	AR207444A1 (es)
AT (1)	AT337176B (es)
BG (5)	BG21405A3 (es)
CA (1)	CA1034953A (es)
CH (5)	CH603592A5 (es)
DD (1)	DD113757A5 (es)
DK (1)	DK136066C (es)
EG (1)	EG11157A (es)
ES (3)	ES425373A1 (es)
FI (1)	FI57587C (es)
FR (1)	FR2226172B1 (es)
GB (1)	GB1429141A (es)
HK (1)	HK70276A (es)
HU (1)	HU168590B (es)
IE (1)	IE39212B1 (es)
IL (1)	IL44626A (es)
LU (1)	LU69872A1 (es)
NL (1)	NL177917C (es)
NO (1)	NO138530C (es)
PH (1)	PH14829A (es)
PL (1)	PL96883B1 (es)
RO (2)	RO69740A (es)
SE (1)	SE408301B (es)
SU (2)	SU541430A3 (es)
YU (1)	YU104874A (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4056533A (en) *	1973-04-17	1977-11-01	Bayer Aktiengesellschaft	Pyrazol-5-ones
DE2526467A1 (de) *	1975-06-13	1976-12-30	Bayer Ag	4-substituierte pyrazolderivate, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
DE3306366A1 (de) *	1983-02-24	1984-08-30	Bayer Ag, 5090 Leverkusen	Muzolimin enthaltende arzneimittel, deren verwendung und verfahren zu deren herstellung
US4663327A (en) *	1984-05-23	1987-05-05	Bayer Aktiengesellschaft	1-heteroaryl-4-aryl-pyrazolin-5-ones
JPH0730031B2 (ja) *	1986-04-02	1995-04-05	日産化学工業株式会社	２―ピラゾリン―５―オン類の製造法
DE3738963A1 (de) *	1987-11-17	1989-05-24	Bayer Ag	3-aminopyrazolin-5-one
US5711929A (en) *	1989-05-06	1998-01-27	698638 Alberta Ltd.	Purification of elemental sulphur
GB8912861D0 (en) *	1989-06-05	1989-07-26	Sherritt Gordon Ltd	Purification of elemental sulphur
US5300514A (en) *	1990-07-17	1994-04-05	Eli Lilly And Company	Pyrazolidinone CCK and gastrin antagonists and pharmaceutical formulations thereof
US5399565A (en) *	1990-07-17	1995-03-21	Eli Lilly And Company	Pyrazolidinone CCK and gastrin antagonists and pharmaceutical formulations therof
DE69131268T2 (de) *	1990-09-21	1999-12-30	Rohm And Haas Co., Philadelphia	Dihydropyridazinone und Pyridazinone als Fungizide
CN1038249C (zh) *	1991-08-28	1998-05-06	罗姆和哈斯公司	含有二氢哒嗪酮及其相关化合物的杀菌组合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2376380A (en) *		1945-05-22		Preparation of amino pyrazolones
GB636988A (en) *	1947-12-24	1950-05-10	Gevaert Photo Producten Naamlo	Improvements in and relating to the production of colour photographic images
US2511231A (en) *	1949-03-26	1950-06-13	Eastman Kodak Co	1-cyanophenyl-3-acylamino-5-pyrazolone couplers for color photography
US2600788A (en) *	1949-06-07	1952-06-17	Eastman Kodak Co	Halogen-substituted pyrazolone couplers for color photography
US2672417A (en) *	1949-12-31	1954-03-16	Gevaert Photo Prod Nv	Production of color photographic images
NL279140A (es) *	1961-05-31

1974
- 1974-01-01 AR AR253331A patent/AR207444A1/es active
- 1974-03-29 FR FR7411495A patent/FR2226172B1/fr not_active Expired
- 1974-04-09 HU HUBA3058A patent/HU168590B/hu unknown
- 1974-04-11 FI FI1105/74A patent/FI57587C/fi active
- 1974-04-12 BG BG027980A patent/BG21405A3/xx unknown
- 1974-04-12 BG BG026395A patent/BG21217A3/xx unknown
- 1974-04-12 BG BG027979A patent/BG22821A3/xx unknown
- 1974-04-12 BG BG027977A patent/BG21857A3/xx unknown
- 1974-04-12 IL IL44626A patent/IL44626A/xx unknown
- 1974-04-12 BG BG027978A patent/BG21218A3/xx unknown
- 1974-04-15 YU YU01048/74A patent/YU104874A/xx unknown
- 1974-04-15 RO RO7485201A patent/RO69740A/ro unknown
- 1974-04-15 US US05/461,282 patent/US3957814A/en not_active Expired - Lifetime
- 1974-04-15 JP JP4111274A patent/JPS5314071B2/ja not_active Expired
- 1974-04-15 RO RO7400078420A patent/RO63749A/ro unknown
- 1974-04-15 PH PH15730A patent/PH14829A/en unknown
- 1974-04-15 DD DD177913A patent/DD113757A5/xx unknown
- 1974-04-16 NO NO741365A patent/NO138530C/no unknown
- 1974-04-16 ES ES425373A patent/ES425373A1/es not_active Expired
- 1974-04-16 PL PL1974170378A patent/PL96883B1/pl unknown
- 1974-04-16 NL NLAANVRAGE7405115,A patent/NL177917C/xx not_active IP Right Cessation
- 1974-04-16 CH CH524274A patent/CH603592A5/xx not_active IP Right Cessation
- 1974-04-16 DK DK208074A patent/DK136066C/da not_active IP Right Cessation
- 1974-04-16 LU LU69872A patent/LU69872A1/xx unknown
- 1974-04-16 CH CH156477A patent/CH605801A5/xx not_active IP Right Cessation
- 1974-04-16 EG EG119/74A patent/EG11157A/xx active
- 1974-04-16 SE SE7405078A patent/SE408301B/sv not_active IP Right Cessation
- 1974-04-16 CH CH156577A patent/CH605800A5/xx not_active IP Right Cessation
- 1974-04-16 CH CH156377A patent/CH596172A5/xx not_active IP Right Cessation
- 1974-04-16 AT AT313274A patent/AT337176B/de not_active IP Right Cessation
- 1974-04-16 CH CH156677A patent/CH605797A5/xx not_active IP Right Cessation
- 1974-04-16 GB GB1650774A patent/GB1429141A/en not_active Expired
- 1974-04-17 CA CA197,660A patent/CA1034953A/en not_active Expired
- 1974-04-17 IE IE798/74A patent/IE39212B1/xx unknown
1975
- 1975-01-01 AR AR258508A patent/AR205272A1/es active
- 1975-01-01 AR AR258506A patent/AR208192A1/es active
- 1975-01-01 AR AR258507A patent/AR205271A1/es active
- 1975-03-19 SU SU2114308A patent/SU541430A3/ru active
- 1975-03-19 SU SU2115103A patent/SU539525A3/ru active
- 1975-04-25 AR AR258505A patent/AR204951A1/es active
1976
- 1976-04-15 ES ES447064A patent/ES447064A1/es not_active Expired
- 1976-04-15 ES ES447063A patent/ES447063A1/es not_active Expired
- 1976-11-11 HK HK702/76*UA patent/HK70276A/xx unknown

Also Published As

Publication number	Publication date
DD113757A5 (es)	1975-06-20
AR204951A1 (es)	1976-03-19
NO741365L (no)	1974-10-18
RO63749A (fr)	1979-01-15
CH605801A5 (es)	1978-10-13
DK136066B (da)	1977-08-08
AR207444A1 (es)	1976-10-08
IL44626A (en)	1980-01-31
SE408301B (sv)	1979-06-05
RO69740A (ro)	1982-09-09
NL177917C (nl)	1985-12-16
CH605797A5 (es)	1978-10-13
AT337176B (de)	1977-06-10
PH14829A (en)	1981-12-16
ATA313274A (de)	1976-10-15
JPS5018466A (es)	1975-02-26
AR205272A1 (es)	1976-04-21
DK136066C (da)	1978-01-16
FI57587B (fi)	1980-05-30
IL44626A0 (en)	1974-06-30
ES425373A1 (es)	1976-09-01
PL96883B1 (pl)	1978-01-31
JPS5314071B2 (es)	1978-05-15
BG21405A3 (bg)	1976-05-20
CH596172A5 (es)	1978-02-28
SU541430A3 (ru)	1976-12-30
CH605800A5 (es)	1978-10-13
NO138530C (no)	1978-09-20
US3957814A (en)	1976-05-18
FI57587C (fi)	1980-09-10
BG21857A3 (bg)	1976-09-20
CA1034953A (en)	1978-07-18
NO138530B (no)	1978-05-12
LU69872A1 (es)	1974-11-28
GB1429141A (en)	1976-03-24
AU6817474A (en)	1975-10-23
BG21218A3 (bg)	1976-03-20
ES447064A1 (es)	1977-09-16
IE39212B1 (en)	1978-08-30
BG21217A3 (bg)	1976-03-20
BG22821A3 (bg)	1977-04-20
HK70276A (en)	1976-11-19
CH603592A5 (es)	1978-08-31
FR2226172A1 (es)	1974-11-15
EG11157A (en)	1978-03-29
AR208192A1 (es)	1976-12-09
SU539525A3 (ru)	1976-12-15
YU104874A (en)	1982-02-28
HU168590B (es)	1976-06-28
IE39212L (en)	1974-10-17
AR205271A1 (es)	1976-04-21
NL7405115A (es)	1974-10-21
NL177917B (nl)	1985-07-16
FR2226172B1 (es)	1978-07-28

Legal Events

Date	Code	Title	Description
2007-11-16	FD1A	Patent lapsed	Effective date: 19890227

Publication	Publication Date	Title
ES440599A1 (es)	1977-05-16	Procedimiento para la produccion de derivados de 2,1,3-ben- zotiadiazol.
ES447064A1 (es)	1977-09-16	Procedimiento para la produccion de pirazolonas-(5) 1-susti-tuidas.
SE7712630L (sv)	1978-05-10	Forfarande for framstellning av o-alkylerade hydroxylaminer
ES438283A1 (es)	1977-01-16	Procedimiento para la preparacion de aductos cristalinos es-tables.
ES347319A1 (es)	1969-05-16	Un procedimiento para la preparacion de nuevos compuestos aromaticos heterociclicos.
ES420179A1 (es)	1976-05-01	Un procedimiento para la preparacion de iminas triciclicas con actividad farmacodinamica.
ES423058A1 (es)	1976-04-16	Procedimiento de preparacion de nuevos deivados de la i- soindolina.
ES428446A1 (es)	1976-12-16	Procedimiento para la preparacion de isotiazolilureas sus- tituidas.
ES419019A1 (es)	1976-06-16	Procedimiento para la preparacion de compuestos polici- clicos.
ES328052A1 (es)	1967-09-01	Procedimiento para la preparacion de tiofosfatos de efecto antiparasitario.
ES431552A1 (es)	1977-02-01	Procedimiento para preparar triazinadionas herbicidas.
GB1382974A (en)	1975-02-05	Process for the production of thiosemicarbazides
GB1393750A (en)	1975-05-14	Bis-1,2,4-triazolyl 5- compounds and their use as optical brightening agents
ES392665A1 (es)	1973-08-01	Un procedimiento para preparar derivados de benzodiazepina-1-sustituidos y sales de los mismos.
ES388696A1 (es)	1974-03-01	Procedimiento para preparar derivados de 6-nitroanilina sustituidos de efecto herbicida.
ES446592A1 (es)	1977-11-16	Procedimiento para la preparacion de derivados de urea.
ES405984A1 (es)	1976-02-01	Procedimiento para la preparacion de fenilisoindolinas ba- sicamente sustituidas.
ES448275A1 (es)	1977-11-16	Un procedimiento para la produccion de nuevas benzo 2,4-ta- cepinas.
ES429319A1 (es)	1976-08-16	Un metodo para preparar un nuevo derivado de 2-fenilamino- piridina.
ES417403A1 (es)	1976-05-16	Un procedimiento para la preparacion de carboxanilidas.
ES449570A1 (es)	1977-12-01	Un procedimiento para la produccion de tetrazolo (a) quina- zol-5-onas.
GB1326853A (en)	1973-08-15	4,5-bis-trifluoromethylamino derivatives of thiazolidines and to a process for their preparation
ES411828A1 (es)	1976-05-16	Un metodo de preparacion de formadores de color incoloros.
ES388250A1 (es)	1973-05-16	Un procedimiento para preparar compuestos de acido pirazo- lo-piridincarboxilico.
ES251042A1 (es)	1959-12-01	Procedimiento para la obtencion de nuevas hidracidas