ES454502A1 - A PROCEDURE FOR THE PREPARATION OF 1,2-BENZOTHIAZIN-3-CARBOXAMIDES. - Google Patents
A PROCEDURE FOR THE PREPARATION OF 1,2-BENZOTHIAZIN-3-CARBOXAMIDES.Info
- Publication number
- ES454502A1 ES454502A1 ES454502A ES454502A ES454502A1 ES 454502 A1 ES454502 A1 ES 454502A1 ES 454502 A ES454502 A ES 454502A ES 454502 A ES454502 A ES 454502A ES 454502 A1 ES454502 A1 ES 454502A1
- Authority
- ES
- Spain
- Prior art keywords
- formula
- preparation
- carboxamides
- benzothiazin
- procedure
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Abstract
A process for the preparation of 1,2-benzothiazine-3-carboxamides according to the formula ** (see formula) ** And its alkali metal and alkaline earth metal salts in which r is 2-thiazolyl or 2-pyridyl, characterized by contacting an alkali metal or alkaline earth metal salt of a compound according to the formula: ** (see formula) ** With at least one mole of a methylating agent in a solvent inert to the reaction at a temperature of 0 to 100ºC (273 to 373º k) and when it is required to prepare the pharmaceutically acceptable salt. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US64850776A | 1976-01-12 | 1976-01-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES454502A1 true ES454502A1 (en) | 1977-12-01 |
Family
ID=24601065
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES454502A Expired ES454502A1 (en) | 1976-01-12 | 1976-12-22 | A PROCEDURE FOR THE PREPARATION OF 1,2-BENZOTHIAZIN-3-CARBOXAMIDES. |
Country Status (15)
| Country | Link |
|---|---|
| JP (1) | JPS5293777A (en) |
| AR (1) | AR210628A1 (en) |
| AT (1) | AT349483B (en) |
| CA (1) | CA1069894A (en) |
| CH (1) | CH594650A5 (en) |
| DD (1) | DD130145A5 (en) |
| DK (1) | DK579876A (en) |
| ES (1) | ES454502A1 (en) |
| FI (1) | FI63231B (en) |
| HU (1) | HU173509B (en) |
| LU (1) | LU76466A1 (en) |
| NL (1) | NL7614135A (en) |
| PL (1) | PL102554B1 (en) |
| SE (1) | SE421792B (en) |
| SU (1) | SU634672A3 (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IN160683B (en) * | 1981-06-01 | 1987-07-25 | Pfizer | |
| US4474955A (en) * | 1981-06-17 | 1984-10-02 | Vincenzo Iannella | Process for preparing 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-[N-(2-pyridinyl)carboxamide]-1,1-dioxide, and its phosphoric ester |
| IN159273B (en) * | 1981-10-05 | 1987-04-25 | Pfizer | |
| DE3217315C2 (en) * | 1982-05-08 | 1986-05-22 | Gödecke AG, 1000 Berlin | Medicinal preparations containing oxicam derivatives |
| IT1216686B (en) * | 1988-04-01 | 1990-03-08 | Chiesi Farma Spa | AQUEOUS PHARMACEUTICAL FORMULATIONS OF PIROXICAM AND PROCEDURE FOR THEIR PREPARATION. |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3591584A (en) * | 1968-08-27 | 1971-07-06 | Pfizer | Benzothiazine dioxides |
-
1976
- 1976-12-06 SE SE7613691A patent/SE421792B/en not_active IP Right Cessation
- 1976-12-07 CA CA267,358A patent/CA1069894A/en not_active Expired
- 1976-12-10 AT AT915876A patent/AT349483B/en active
- 1976-12-20 NL NL7614135A patent/NL7614135A/en not_active Application Discontinuation
- 1976-12-21 JP JP15411376A patent/JPS5293777A/en active Pending
- 1976-12-22 DK DK579876A patent/DK579876A/en not_active Application Discontinuation
- 1976-12-22 ES ES454502A patent/ES454502A1/en not_active Expired
- 1976-12-22 FI FI763680A patent/FI63231B/en not_active Application Discontinuation
- 1976-12-22 CH CH1620476A patent/CH594650A5/en not_active IP Right Cessation
- 1976-12-23 AR AR265984A patent/AR210628A1/en active
- 1976-12-23 LU LU76466A patent/LU76466A1/xx unknown
- 1976-12-29 HU HU76PI556A patent/HU173509B/en not_active IP Right Cessation
- 1976-12-29 SU SU762435654A patent/SU634672A3/en active
- 1976-12-30 DD DD7600196765A patent/DD130145A5/en unknown
- 1976-12-30 PL PL1976194854A patent/PL102554B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA1069894A (en) | 1980-01-15 |
| CH594650A5 (en) | 1978-01-13 |
| JPS5293777A (en) | 1977-08-06 |
| NL7614135A (en) | 1977-07-14 |
| LU76466A1 (en) | 1977-07-05 |
| FI63231B (en) | 1983-01-31 |
| DK579876A (en) | 1977-07-13 |
| PL102554B1 (en) | 1979-04-30 |
| AR210628A1 (en) | 1977-08-31 |
| HU173509B (en) | 1979-05-28 |
| AT349483B (en) | 1979-04-10 |
| SE7613691L (en) | 1977-07-13 |
| FI763680A7 (en) | 1977-07-13 |
| SE421792B (en) | 1982-02-01 |
| DD130145A5 (en) | 1978-03-08 |
| SU634672A3 (en) | 1978-11-25 |
| ATA915876A (en) | 1978-09-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19981103 |