ES471207A1 - Pyrimidino (1,2a)heterocyclic amide derivatives - Google Patents

Pyrimidino (1,2a)heterocyclic amide derivatives

Info

Publication number
ES471207A1
ES471207A1 ES471207A ES471207A ES471207A1 ES 471207 A1 ES471207 A1 ES 471207A1 ES 471207 A ES471207 A ES 471207A ES 471207 A ES471207 A ES 471207A ES 471207 A1 ES471207 A1 ES 471207A1
Authority
ES
Spain
Prior art keywords
pyrimidino
amide derivatives
heterocyclic amide
represent
optically active
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES471207A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Vegyeszeti Termekek Gyara R T
Chinoin Private Co Ltd
Original Assignee
Vegyeszeti Termekek Gyara R T
Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vegyeszeti Termekek Gyara R T, Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt filed Critical Vegyeszeti Termekek Gyara R T
Publication of ES471207A1 publication Critical patent/ES471207A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Procedimiento para la preparación de nuevos derivados condensados de pirimidina, de la fórmula general (I) **(Fórmula)** en donde R y R1 significan un grupo alquilo de C1-6 R2 y R3 significan un átomo de hidrógeno, y m es 0 y n es 0, así como los isómeros ópticamente activos y de las sales fisiológicamente tolerables de estos compuestos, caracterizado porque los derivados condensados de pirimidina existentes, en su caso, como racemato u ópticamente activos.Process for the preparation of new condensed pyrimidine derivatives of the general formula (I) **(Formula)** wherein R and R1 represent a C1-6 alkyl group, R2 and R3 represent a hydrogen atom, and m is 0 and n is 0, as well as the optically active isomers and physiologically tolerable salts of these compounds, characterized in that the condensed pyrimidine derivatives exist, where appropriate, as a racemate or optically active.

ES471207A 1976-06-25 1978-06-16 Pyrimidino (1,2a)heterocyclic amide derivatives Expired ES471207A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU76CI1673A HU174901B (en) 1976-06-25 1976-06-25 SPOSOB POLUCHENIA NOVYKH PROIZVODNYKH PIRIDO / 1,2-A / PIRIMIDINA

Publications (1)

Publication Number Publication Date
ES471207A1 true ES471207A1 (en) 1979-01-16

Family

ID=10994621

Family Applications (3)

Application Number Title Priority Date Filing Date
ES460109A Expired ES460109A1 (en) 1976-06-25 1977-06-25 PROCEDURE FOR THE PREPARATION OF NEW PYRIMIDINE CONDENSED DERIVATIVES.
ES471208A Expired ES471208A1 (en) 1976-06-25 1978-06-16 Pyrimidino (1,2a)heterocyclic amide derivatives
ES471207A Expired ES471207A1 (en) 1976-06-25 1978-06-16 Pyrimidino (1,2a)heterocyclic amide derivatives

Family Applications Before (2)

Application Number Title Priority Date Filing Date
ES460109A Expired ES460109A1 (en) 1976-06-25 1977-06-25 PROCEDURE FOR THE PREPARATION OF NEW PYRIMIDINE CONDENSED DERIVATIVES.
ES471208A Expired ES471208A1 (en) 1976-06-25 1978-06-16 Pyrimidino (1,2a)heterocyclic amide derivatives

Country Status (18)

Country Link
JP (1) JPS5318719A (en)
AT (1) AT362377B (en)
BE (1) BE856085A (en)
CH (3) CH636101A5 (en)
CS (1) CS204004B2 (en)
DD (1) DD131750A5 (en)
DE (1) DE2728198A1 (en)
DK (1) DK151885C (en)
ES (3) ES460109A1 (en)
FI (1) FI771940A7 (en)
FR (1) FR2355844A1 (en)
GB (1) GB1583896A (en)
HU (1) HU174901B (en)
NL (1) NL187575C (en)
PL (3) PL110223B1 (en)
SE (1) SE432594B (en)
SU (1) SU665805A3 (en)
YU (3) YU41576B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3171775A (en) * 1962-05-18 1965-03-02 West Virginia Pulp & Paper Co Distributor system for a paper machine headbox
US4666912A (en) * 1984-11-12 1987-05-19 Chinoin Gyogyszer Es Vegyeszeti Termeker Gyara Rt Treating process
JPH0558850U (en) * 1992-01-13 1993-08-03 株式会社ゼクセル Centrifugal force governor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT296996B (en) * 1966-11-02 1972-03-10 Chinoin Gyogyszer Es Vegyeszet Process for the preparation of homopyrimidazole derivatives and their acid addition salts and quaternary ammonium salts
HU168014B (en) * 1973-03-30 1976-02-28

Also Published As

Publication number Publication date
DK151885B (en) 1988-01-11
PL112745B1 (en) 1980-10-31
YU41576B (en) 1987-10-31
SE432594B (en) 1984-04-09
BE856085A (en) 1977-10-17
DE2728198C2 (en) 1987-12-23
FI771940A7 (en) 1977-12-26
ES460109A1 (en) 1978-11-16
DD131750A5 (en) 1978-07-19
NL187575B (en) 1991-06-17
DK151885C (en) 1988-08-08
FR2355844A1 (en) 1978-01-20
FR2355844B1 (en) 1982-11-05
PL199145A1 (en) 1978-12-04
YU40623B (en) 1986-02-28
YU197782A (en) 1983-01-21
GB1583896A (en) 1981-02-04
YU42048B (en) 1988-04-30
DE2728198A1 (en) 1978-01-05
NL187575C (en) 1991-11-18
PL122962B1 (en) 1982-09-30
YU155477A (en) 1983-01-21
ATA446777A (en) 1980-10-15
DK282777A (en) 1977-12-26
JPS5318719A (en) 1978-02-21
AT362377B (en) 1981-05-11
CH635101A5 (en) 1983-03-15
CH636101A5 (en) 1983-05-13
CH635100A5 (en) 1983-03-15
YU197682A (en) 1983-01-21
CS204004B2 (en) 1981-03-31
PL110223B1 (en) 1980-07-31
HU174901B (en) 1980-04-28
NL7707018A (en) 1977-12-28
JPS62150B2 (en) 1987-01-06
ES471208A1 (en) 1979-01-16
SU665805A3 (en) 1979-05-30
SE7707200L (en) 1977-12-26

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