ES472813A1 - Procedimiento para la preparacion de nuevas 1-piperazinil-4h-s-striazolo (3,4c)tieno (2,3e)1,4-diazepinas sustituidas - Google Patents
Procedimiento para la preparacion de nuevas 1-piperazinil-4h-s-striazolo (3,4c)tieno (2,3e)1,4-diazepinas sustituidasInfo
- Publication number
- ES472813A1 ES472813A1 ES472813A ES472813A ES472813A1 ES 472813 A1 ES472813 A1 ES 472813A1 ES 472813 A ES472813 A ES 472813A ES 472813 A ES472813 A ES 472813A ES 472813 A1 ES472813 A1 ES 472813A1
- Authority
- ES
- Spain
- Prior art keywords
- substd
- opt
- halo
- diazepine
- thieno
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 239000002249 anxiolytic agent Substances 0.000 title 1
- 230000000949 anxiolytic effect Effects 0.000 title 1
- 229940005530 anxiolytics Drugs 0.000 title 1
- 229940125723 sedative agent Drugs 0.000 title 1
- 239000000932 sedative agent Substances 0.000 title 1
- -1 tranquillisers Substances 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000005843 halogen group Chemical group 0.000 abstract 3
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 2
- GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical compound C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- GRVDJDISBSALJP-UHFFFAOYSA-N methyloxidanyl Chemical compound [O]C GRVDJDISBSALJP-UHFFFAOYSA-N 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000004076 pyridyl group Chemical group 0.000 abstract 2
- WFCSWCVEJLETKA-UHFFFAOYSA-N 2-piperazin-1-ylethanol Chemical compound OCCN1CCNCC1 WFCSWCVEJLETKA-UHFFFAOYSA-N 0.000 abstract 1
- 241000699670 Mus sp. Species 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 230000034994 death Effects 0.000 abstract 1
- 231100000517 death Toxicity 0.000 abstract 1
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 1
- 150000004908 diazepines Chemical class 0.000 abstract 1
- 125000001475 halogen functional group Chemical group 0.000 abstract 1
- 125000000714 pyrimidinyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
Procedimiento para la preparación de nuevas 1-piperazinil-4H-s-triazolo[33,4c]tieno[2,3e]1,4-diazepinas sustituidas de la fórmula general **(Fórmula)** en la que R1 significa el radical R4 - CO -; R2 significa hidrógeno, fluor, cloro o bromo; R3 significa cloro o bromo o un radical alcohilo; y R4 significa hidrógeno, alcohilo con 1 a 17 átomos de carbono, alcoxi con 1 a 2 átomos de carbono, fenilo, tolilo, metoxifenilo, halogenofenilo, -nitrofenilo y piridilo.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19772732943 DE2732943A1 (de) | 1977-07-21 | 1977-07-21 | Neue substituierte 1-piperazinyl- 4h-s-triazolo eckige klammer auf 3,4c eckige klammer zu thieno eckige klammer auf 2,3e eckige klammer zu 1,4-diazepine, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES472813A1 true ES472813A1 (es) | 1979-02-16 |
Family
ID=6014503
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES472813A Expired ES472813A1 (es) | 1977-07-21 | 1978-08-24 | Procedimiento para la preparacion de nuevas 1-piperazinil-4h-s-striazolo (3,4c)tieno (2,3e)1,4-diazepinas sustituidas |
Country Status (3)
| Country | Link |
|---|---|
| DE (1) | DE2732943A1 (es) |
| ES (1) | ES472813A1 (es) |
| ZA (1) | ZA784122B (es) |
-
1977
- 1977-07-21 DE DE19772732943 patent/DE2732943A1/de not_active Withdrawn
-
1978
- 1978-07-20 ZA ZA784122A patent/ZA784122B/xx unknown
- 1978-08-24 ES ES472813A patent/ES472813A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ZA784122B (en) | 1980-03-26 |
| DE2732943A1 (de) | 1979-02-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19971201 |