ES489628A0 - Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina - Google Patents

Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina

Info

Publication number
ES489628A0
ES489628A0 ES489628A ES489628A ES489628A0 ES 489628 A0 ES489628 A0 ES 489628A0 ES 489628 A ES489628 A ES 489628A ES 489628 A ES489628 A ES 489628A ES 489628 A0 ES489628 A0 ES 489628A0
Authority
ES
Spain
Prior art keywords
piperidina
piridina
tetrahidro
derivatives
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES489628A
Other languages
English (en)
Other versions
ES8104281A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES489628A0 publication Critical patent/ES489628A0/es
Publication of ES8104281A1 publication Critical patent/ES8104281A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/86—Benzo [b] furans; Hydrogenated benzo [b] furans with an oxygen atom directly attached in position 7
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/91—Dibenzofurans; Hydrogenated dibenzofurans

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES489628A 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina Expired ES8104281A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH682378 1978-06-22

Publications (2)

Publication Number Publication Date
ES489628A0 true ES489628A0 (es) 1981-04-01
ES8104281A1 ES8104281A1 (es) 1981-04-01

Family

ID=4315581

Family Applications (3)

Application Number Title Priority Date Filing Date
ES481714A Expired ES481714A1 (es) 1978-06-22 1979-06-20 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina.
ES489627A Granted ES489627A0 (es) 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina
ES489628A Expired ES8104281A1 (es) 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina

Family Applications Before (2)

Application Number Title Priority Date Filing Date
ES481714A Expired ES481714A1 (es) 1978-06-22 1979-06-20 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina.
ES489627A Granted ES489627A0 (es) 1978-06-22 1980-03-17 Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina

Country Status (10)

Country Link
US (1) US4259338A (es)
EP (1) EP0006524A1 (es)
JP (1) JPS552697A (es)
AU (1) AU523656B2 (es)
CA (1) CA1119601A (es)
DD (1) DD144545A5 (es)
DK (1) DK259879A (es)
ES (3) ES481714A1 (es)
NZ (1) NZ190784A (es)
ZA (1) ZA793091B (es)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4495357A (en) * 1981-07-01 1985-01-22 The Upjohn Company Pyridyl-substituted-benzofurans
US4490531A (en) * 1981-07-01 1984-12-25 The Upjohn Company Pyridyl-substituted-benzofurans
US4455427A (en) * 1981-07-01 1984-06-19 The Upjohn Company Pyridyl-substituted-benzofurans
US4452986A (en) * 1982-06-08 1984-06-05 The Upjohn Company Imidazolyl-substituted benzofurans
US4447620A (en) * 1982-06-08 1984-05-08 The Upjohn Company Imidazolyl-substituted benzothiophenes
US4430502A (en) 1982-08-13 1984-02-07 The Upjohn Company Pyridinyl substituted benzimidazoles and quinoxalines
IL69898A0 (en) * 1982-10-08 1984-01-31 Ciba Geigy Ag Furans
US4855435A (en) * 1982-10-12 1989-08-08 The Upjohn Company Pyridyl-substituted benzothiophenes
US4611059A (en) * 1982-10-12 1986-09-09 The Upjohn Company Pyridyl-substituted benzothiophenes
US5296497A (en) * 1989-05-16 1994-03-22 Duphar International Research B.V. 3,4-dehydropiperidine derivatives having psychotropic activity
EP0398413A1 (en) * 1989-05-16 1990-11-22 Duphar International Research B.V "3,4-dehydropiperidine derivatives having psychotropic activity
EP0404721A3 (de) * 1989-06-20 1991-12-27 Ciba-Geigy Ag Mikrobizide Mittel
DE4017211A1 (de) * 1990-05-29 1991-12-05 Merck Patent Gmbh Oxazolidinone
TW222631B (es) * 1991-07-15 1994-04-21 Duphar Int Res
EP0637586B1 (en) * 1993-08-05 1999-06-02 HOECHST MARION ROUSSEL, Inc. 2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)-benzofuran-7-carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors
JPH07320652A (ja) * 1994-05-27 1995-12-08 Toshiba Corp カラー受像管及びシャドウマスクの製造方法
FR2739856B1 (fr) * 1995-10-11 1997-11-14 Synthelabo Derives de 3-benzofuranyloxazolidin-2-one, leur procede de preparation et leur application en therapeutique
EP0891358A1 (fr) * 1995-10-11 1999-01-20 Synthelabo Composes derives d'oxazolidin-2-one, leur procede de preparation et leur application en therapeutique
FR2751653B1 (fr) * 1996-07-25 1998-09-04 Synthelabo Derives de 3-benzofuranyloxazolidin-2-one, leur procede de preparation et leur application en therapeutique
FR2741071B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives de 3-(benzofuran-5-yl)oxazolidin-2-one, leur preparation et leur application en therapeutique
FR2741072B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives d'oxazolidin-2-one, leur preparation et leur application en therapeutique
AR019178A1 (es) * 1998-06-30 2001-12-26 Lilly Co Eli Compuestos de 7-(benzo(b)tiofeno, furan e indolpiridil o tetrahidropiridilo), efectivos sobre sistemas relacionados con la serotonina, composicionesfarmaceuticas formuladas con dichos compuestos; compuestos intermediarios utiles para preparar dichos compuestos de tiofeno, furan e indolpiridilo otetr
GB9912413D0 (en) 1999-05-28 1999-07-28 Pfizer Ltd Compounds useful in therapy
CA2378878A1 (en) * 1999-07-29 2001-02-08 Jeffrey Thomas Mullaney Benzofurylpiperazines and benzofurylhomopiperazines: serotonin agonists
US6881733B1 (en) 1999-07-29 2005-04-19 Eli Lilly And Company Serotonergic benzofurans
DK1204658T3 (da) * 1999-07-29 2003-09-01 Lilly Co Eli Benzofurylpiperazin-serotoninagonister
WO2001009122A2 (en) * 1999-07-29 2001-02-08 Eli Lilly And Company Serotonergic benzofurans
WO2004106317A1 (ja) * 2003-05-29 2004-12-09 The New Industry Research Organization ベンゾフラン化合物、およびそれを含有してなる医薬組成物
JP2005008631A (ja) * 2003-05-29 2005-01-13 New Industry Research Organization ベンゾフラン化合物、およびそれを含有してなる医薬組成物
EP2110374A1 (en) * 2008-04-18 2009-10-21 Merck Sante Benzofurane, benzothiophene, benzothiazol derivatives as FXR modulators
CN101810606A (zh) * 2010-03-12 2010-08-25 南方医科大学 2-(6-羟基-2′,3′-二甲氧基苯基)-6-羟基-7-甲氧基苯骈呋喃在制备单胺氧化酶抑制剂中的应用
CN102381961B (zh) * 2011-09-03 2014-01-15 四川大学 3-苯基戊二酸类化合物、其制备方法和用途
CN118460017B (zh) * 2024-05-11 2024-11-05 广州豫顺新材料科技有限公司 一种覆铜板用改性球形硅微粉及其制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2633468A (en) * 1951-07-26 1953-03-31 Lilly Co Eli Benzooxaheterocyclic bases and acid addition salts thereof
GB1041525A (en) * 1964-11-11 1966-09-07 Belge Produits Chimiques Sa Benzofuran derivatives and processes for preparing the same
GB1139146A (en) 1966-10-10 1969-01-08 Belge Produits Chimiques Sa Benzofuran derivatives and processes for preparing the same
US3751390A (en) * 1971-05-19 1973-08-07 Aldrich Chem Co Inc Substituted dibenzofuran
BE794630A (fr) * 1972-01-26 1973-07-26 Beecham Group Ltd Composes polycycliques antihypertenseurs
CH592656A5 (es) * 1973-03-02 1977-10-31 Ciba Geigy Ag
IE39264B1 (en) * 1973-05-25 1978-08-30 Ciba Geigy Ag New pharmaceutical preparations
CH609054A5 (en) * 1975-11-26 1979-02-15 Ciba Geigy Ag Process for the preparation of a novel piperidine derivative
CH609980A5 (en) * 1974-08-30 1979-03-30 Ciba Geigy Ag Process for the preparation of novel piperidine derivatives
LU76756A1 (es) * 1977-02-11 1978-10-18

Also Published As

Publication number Publication date
US4259338A (en) 1981-03-31
JPS552697A (en) 1980-01-10
ZA793091B (en) 1980-06-25
AU4825779A (en) 1980-01-03
DD144545A5 (de) 1980-10-22
ES481714A1 (es) 1980-06-16
CA1119601A (en) 1982-03-09
NZ190784A (en) 1982-03-16
ES8104280A1 (es) 1981-04-01
ES489627A0 (es) 1981-04-01
ES8104281A1 (es) 1981-04-01
EP0006524A1 (de) 1980-01-09
AU523656B2 (en) 1982-08-05
DK259879A (da) 1979-12-23

Similar Documents

Publication Publication Date Title
AR220704A1 (es) Procedimiento para la preparacion de derivados de indanil y tetrahidronaftil octatrieno
ES489627A0 (es) Procedimiento para la obtencion de derivados de tetrahidro- piridina y piperidina
MX6749E (es) Procedimiento para la preparacion de derivados de tetrazolilalcoxicarboestirilo
ES494634A0 (es) Procedimiento para la preparacion de compuestos de cefem y cefam
MX5631E (es) Procedimiento para la preparacion de acil-anilinas
MX5793E (es) Procedimiento para la preparacion de 4-amino-5-alquilsulfonil-orto-anisamidas
MX5676E (es) Procedimiento mejorado para la preparacion de cicloalcanoles y cicloalcanonas
ES482498A0 (es) Procedimiento para la preparacion de 2-cloro-6-nitroanilinas
AR221355A1 (es) Procedimiento para la preparacion de derivados de pirrolidinil y pirrolidinilmetil-benzamidas
MX5509E (es) Procedimiento para la preparacion de n-halogenoacetil-fenilaminocarboniloximas
AR227379A1 (es) Procedimiento para la preparacion de 1-aril-2-imidazolil vinileteres
MX5898E (es) Procedimiento para la preparacion de 2-amino-4-pirimidonas
AR224784A1 (es) Procedimiento para la preparacion de nuevos derivados de 4-amino-2-piperidinoquinazolina
MX5594E (es) Procedimiento mejorado para la preparacion de derivados de n-trifluoroacetil-n-fosfonometilglicinatos
ES485567A0 (es) Procedimiento para la preparacion de azolilcetales
MX5826E (es) Procedimiento para la obtencion de derivados de fenilimino metil-piridina
MX5672E (es) Procedimiento para la preparacion de acidos 2-piridil y 2-pirimidil-aminobenzoicos
MX5738E (es) Procedimiento para la obtencion de compuestos de iminoeter de benzotiazolina y benzoxazolina-n-substituidos
MX5955E (es) Procedimiento para la preparacion de derivados de piridoxina
MX149694A (es) Procedimiento para la preparacion de trialcoxisilanos de fenoxialquilo
ES484342A0 (es) Procedimiento para la preparacion de propenilensulfona
ES488835A0 (es) Procedimiento para la obtencion de nuevos derivados de la piperacina metanimina
AR227629A1 (es) Procedimiento para la preparacion esteroespecifica o esteroselectiva de derivados de imidazolil-oxi-meteres y derivados de imidazoliloximas
MX6158E (es) Procedimiento para la preparacion de derivados piperazinilbenzoheterociclicos
MX5674E (es) Procedimiento para la preparacion de derivados de la butenofenona