ES494955A0 - Un procedimiento para preparar derivados de fenilpiperidina - Google Patents
Un procedimiento para preparar derivados de fenilpiperidinaInfo
- Publication number
- ES494955A0 ES494955A0 ES494955A ES494955A ES494955A0 ES 494955 A0 ES494955 A0 ES 494955A0 ES 494955 A ES494955 A ES 494955A ES 494955 A ES494955 A ES 494955A ES 494955 A0 ES494955 A0 ES 494955A0
- Authority
- ES
- Spain
- Prior art keywords
- preparing
- procedure
- phenylpiperidine derivatives
- derivatives
- intermediates
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- LLSKXGRDUPMXLC-UHFFFAOYSA-N 1-phenylpiperidine Chemical class C1CCCCN1C1=CC=CC=C1 LLSKXGRDUPMXLC-UHFFFAOYSA-N 0.000 title 1
- 229940051803 opioid analgesics phenylpiperidine derivative Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000000543 intermediate Substances 0.000 abstract 2
- 230000000202 analgesic effect Effects 0.000 abstract 1
- 230000001430 anti-depressive effect Effects 0.000 abstract 1
- 239000000935 antidepressant agent Substances 0.000 abstract 1
- 229940005513 antidepressants Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
-
- H—ELECTRICITY
- H10—SEMICONDUCTOR DEVICES; ELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
- H10D—INORGANIC ELECTRIC SEMICONDUCTOR DEVICES
- H10D30/00—Field-effect transistors [FET]
- H10D30/01—Manufacture or treatment
- H10D30/021—Manufacture or treatment of FETs having insulated gates [IGFET]
- H10D30/028—Manufacture or treatment of FETs having insulated gates [IGFET] of double-diffused metal oxide semiconductor [DMOS] FETs
- H10D30/0291—Manufacture or treatment of FETs having insulated gates [IGFET] of double-diffused metal oxide semiconductor [DMOS] FETs of vertical DMOS [VDMOS] FETs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/54—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/014,548 US4216218A (en) | 1979-02-23 | 1979-02-23 | Antidepressant and analgesic 4-aryloxy- and 4-arylthio-3-phenylpiperidines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES494955A0 true ES494955A0 (es) | 1981-09-01 |
| ES8106892A1 ES8106892A1 (es) | 1981-09-01 |
Family
ID=21766108
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES488708A Granted ES488708A0 (es) | 1979-02-23 | 1980-02-18 | Un procedimiento para preparar derivados de fenilpiperidina |
| ES494955A Expired ES8106892A1 (es) | 1979-02-23 | 1980-09-11 | Un procedimiento para preparar derivados de fenilpiperidina |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES488708A Granted ES488708A0 (es) | 1979-02-23 | 1980-02-18 | Un procedimiento para preparar derivados de fenilpiperidina |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US4216218A (es) |
| EP (1) | EP0014997B1 (es) |
| JP (1) | JPS55147258A (es) |
| AT (1) | ATE4203T1 (es) |
| CA (1) | CA1142522A (es) |
| DE (1) | DE3064183D1 (es) |
| ES (2) | ES488708A0 (es) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4312876A (en) * | 1979-02-23 | 1982-01-26 | Hoechst-Roussel Pharmaceuticals Incorporated | Antidepressive and analgesic 4-aryloxy- and 4-arylthio-3-phenylpiperidines |
| US4333942A (en) * | 1979-08-03 | 1982-06-08 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Anti-depressant and analgesic 4-phenoxypiperidines |
| US4387230A (en) * | 1979-09-06 | 1983-06-07 | John Wyeth And Brother Limited | Process for preparing a dihydropyridine derivative |
| US4496732A (en) * | 1983-03-14 | 1985-01-29 | Hoechst-Roussel Pharmaceuticals Inc. | Stereoselective reduction of 2- or 3-substituted 4-piperidones with sodium borohydride |
| US4529732A (en) * | 1983-03-14 | 1985-07-16 | Pfizer Inc. | 2-[2-Hydroxy-4-(substituted)phenyl]piperidines |
| GB8321157D0 (en) * | 1983-08-05 | 1983-09-07 | Fordonal Sa | Piperidine derivatives |
| US6162927A (en) * | 1994-08-19 | 2000-12-19 | Abbott Laboratories | Endothelin antagonists |
| US7208517B1 (en) | 1994-08-19 | 2007-04-24 | Abbott Labortories | Endothelin antagonists |
| US6124341A (en) * | 1996-02-13 | 2000-09-26 | Abbott Laboratories | Endothelin antagonists |
| CN1222513C (zh) | 1997-02-03 | 2005-10-12 | 富士写真菲林株式会社 | 卤化银彩色照相感光材料和其中所用的菲尼酮化合物以及这类化合物的制备方法 |
| US20020055457A1 (en) * | 2000-08-07 | 2002-05-09 | Janus Todd J. | Methods of treating cancer and the pain associated therewith using endothelin antagonists |
| DE10201550A1 (de) * | 2002-01-17 | 2003-07-31 | Merck Patent Gmbh | Phenoxy-Piperidine |
| JP2007537233A (ja) * | 2004-05-12 | 2007-12-20 | ファイザー・プロダクツ・インク | Ｎｋ１及びｎｋ３アンタゴニストとしてのピペリジン誘導体 |
| US8865906B2 (en) * | 2009-05-15 | 2014-10-21 | Sanofi | Process for the preparation of a compound useful as an inhibitor of TAFIa |
| CN116057038B (zh) * | 2020-09-11 | 2025-12-12 | 大金工业株式会社 | 丙烯酸衍生物的制造方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3542794A (en) * | 1969-11-07 | 1970-11-24 | Grover Cleveland Helsley | 1-carbamoyl-4-phenoxypiperidines |
| DE2116316A1 (de) * | 1970-04-08 | 1971-10-28 | Sandoz Ag, Basel (Schweiz) | Verfahren zur Herstellung neuer heterocyclischer Verbindungen |
| US3743645A (en) * | 1970-10-19 | 1973-07-03 | Robins Co Inc A H | 1-substituted-4-phenoxypiperidines |
| US4132709A (en) * | 1976-12-20 | 1979-01-02 | Ayerst, Mckenna & Harrison, Ltd. | [2]Benzopyrano[4,3-c]pyridine derivatives and process therefor |
| US4147872A (en) * | 1977-09-13 | 1979-04-03 | Pfizer Inc. | 3-[2-Hydroxy-4-(substituted)-phenyl]azacycloalkanes and derivatives thereof as analgesic agents and intermediates therefor |
-
1979
- 1979-02-23 US US06/014,548 patent/US4216218A/en not_active Expired - Lifetime
-
1980
- 1980-02-18 ES ES488708A patent/ES488708A0/es active Granted
- 1980-02-20 EP EP80100838A patent/EP0014997B1/en not_active Expired
- 1980-02-20 DE DE8080100838T patent/DE3064183D1/de not_active Expired
- 1980-02-20 AT AT80100838T patent/ATE4203T1/de not_active IP Right Cessation
- 1980-02-22 JP JP2067280A patent/JPS55147258A/ja active Granted
- 1980-02-22 CA CA000346309A patent/CA1142522A/en not_active Expired
- 1980-09-11 ES ES494955A patent/ES8106892A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| JPH0243740B2 (es) | 1990-10-01 |
| ES8106892A1 (es) | 1981-09-01 |
| US4216218A (en) | 1980-08-05 |
| EP0014997A1 (en) | 1980-09-03 |
| ES8102097A1 (es) | 1980-12-16 |
| ATE4203T1 (de) | 1983-08-15 |
| CA1142522A (en) | 1983-03-08 |
| ES488708A0 (es) | 1980-12-16 |
| EP0014997B1 (en) | 1983-07-20 |
| DE3064183D1 (en) | 1983-08-25 |
| JPS55147258A (en) | 1980-11-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Patent lapsed |
Effective date: 19960506 |