ES512045A0 - "procedimiento de preparar compuestos benzoxepinicos y analogos". - Google Patents

"procedimiento de preparar compuestos benzoxepinicos y analogos".

Info

Publication number
ES512045A0
ES512045A0 ES512045A ES512045A ES512045A0 ES 512045 A0 ES512045 A0 ES 512045A0 ES 512045 A ES512045 A ES 512045A ES 512045 A ES512045 A ES 512045A ES 512045 A0 ES512045 A0 ES 512045A0
Authority
ES
Spain
Prior art keywords
benzoxepinic
preparing
procedure
analog compounds
analog
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES512045A
Other languages
English (en)
Other versions
ES8303395A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pierre Fabre SA
Original Assignee
Pierre Fabre SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8207693A external-priority patent/FR2526429A1/fr
Application filed by Pierre Fabre SA filed Critical Pierre Fabre SA
Publication of ES512045A0 publication Critical patent/ES512045A0/es
Publication of ES8303395A1 publication Critical patent/ES8303395A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
    • C07D313/02—Seven-membered rings
    • C07D313/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D313/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES512045A 1981-05-11 1982-05-10 "procedimiento de preparar compuestos benzoxepinicos y analogos". Expired ES8303395A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8109327 1981-05-11
FR8207693A FR2526429A1 (fr) 1982-05-04 1982-05-04 Nouveaux composes de la serie des benzoxepines et analogues soufres et azotes, leurs procedes de preparation et utilisations en tant que medicament

Publications (2)

Publication Number Publication Date
ES512045A0 true ES512045A0 (es) 1983-03-01
ES8303395A1 ES8303395A1 (es) 1983-03-01

Family

ID=26222386

Family Applications (1)

Application Number Title Priority Date Filing Date
ES512045A Expired ES8303395A1 (es) 1981-05-11 1982-05-10 "procedimiento de preparar compuestos benzoxepinicos y analogos".

Country Status (6)

Country Link
US (1) US4436749A (es)
EP (1) EP0067086B1 (es)
AU (1) AU548253B2 (es)
CA (1) CA1196637A (es)
DE (1) DE3267884D1 (es)
ES (1) ES8303395A1 (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2538250A1 (fr) * 1982-12-28 1984-06-29 Fabre Sa Pierre Nouvel extrait de ruscus, son procede de preparation et son application en tant que principe actif veinotonique
GB8523776D0 (en) * 1985-09-26 1985-10-30 Scras Catechol derivatives
US4824831A (en) * 1987-12-21 1989-04-25 E. R. Squibb & Sons, Inc. 4,5-dihydro-1H-benzazepine-3-carboxylic acid esters which are useful as anti-hypertensive agents
US6642268B2 (en) 1994-09-13 2003-11-04 G.D. Searle & Co. Combination therapy employing ileal bile acid transport inhibiting benzothipines and HMG Co-A reductase inhibitors
US6262277B1 (en) 1994-09-13 2001-07-17 G.D. Searle And Company Intermediates and processes for the preparation of benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
US6268392B1 (en) 1994-09-13 2001-07-31 G. D. Searle & Co. Combination therapy employing ileal bile acid transport inhibiting benzothiepines and HMG Co-A reductase inhibitors
US6221897B1 (en) * 1998-06-10 2001-04-24 Aventis Pharma Deutschland Gmbh Benzothiepine 1,1-dioxide derivatives, a process for their preparation, pharmaceuticals comprising these compounds, and their use
AU2157500A (en) 1998-12-23 2000-07-31 G.D. Searle Llc Combinations of cholesteryl ester transfer protein inhibitors and bile acid sequestering agents for cardiovascular indications
DK1140189T3 (da) 1998-12-23 2003-09-15 Searle Llc Kombinationer af ileal galdesyre-transportinhibitorer og fibrinsyrederivater til cardiovaskulære indikationer
BR9916486A (pt) 1998-12-23 2002-02-05 Searle Llc Combinações de inibidores do transporte de ácidos biliares no ìleo e inibidores da proteìna de transferência do ester colesteril para indicações cardiovasculares
EA004877B1 (ru) 1998-12-23 2004-08-26 Джи.Ди.Сирл Ллс Сочетания ингибиторов транспорта желчных кислот в подвздошной кишке и агентов, секвестрирующих желчные кислоты, для сердечно-сосудистых показаний
US6458850B1 (en) 1998-12-23 2002-10-01 G.D. Searle, Llc Combinations of cholesteryl ester transfer protein inhibitors and fibric acid derivatives for cardiovascular indications
AU2157400A (en) 1998-12-23 2000-07-31 G.D. Searle & Co. Combinations of cholesteryl ester transfer protein inhibitors and hmg coa reductase inhibitors for cardiovascular indications
AU3103800A (en) 1998-12-23 2000-07-31 G.D. Searle Llc Combinations of cholesteryl ester transfer protein inhibitors and nicotinic acidderivatives for cardiovascular indications
WO2000069845A1 (en) 1999-05-18 2000-11-23 Takeda Chemical Industries, Ltd. Processes for the preparation of 2,3-dihydrothiepine derivatives
EP1286984A2 (en) 2000-03-10 2003-03-05 Pharmacia Corporation Method for the preparation of tetrahydrobenzothiepines
BR0213501A (pt) 2001-11-02 2004-08-24 Searle Llc Compostos de benzotiepina mono- e di-fluorada como inibidores de transporte de ácido biliar co-dependente de sódio apical (asbt) e captação de taurocolato
MXPA04006255A (es) 2002-01-17 2004-09-27 Pharmacia Corp Compuestos novedosos de alquil/aril hidroxi o ceto tiepina como inhibidores del transporte del acido biliar codependiente del sodio apical y la captacion de taurocolato.
JP6217938B2 (ja) 2011-10-28 2017-10-25 ルメナ ファーマシューティカルズ エルエルシー 小児の胆汁うっ滞性肝疾患の処置のための胆汁酸再循環阻害剤
EA038594B1 (ru) 2011-10-28 2021-09-21 Шайр Хьюман Дженетик Терапис, Инк. Ингибиторы рециркуляции желчных кислот для лечения гиперхолемии и холестатического заболевания печени
CN111087305B (zh) * 2019-12-13 2021-08-27 南京工业大学 一种β-氟烷基肉桂酸酯类化合物及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL301813A (es) * 1962-12-14 1900-01-01
US3374245A (en) 1964-04-01 1968-03-19 Ciba Geigy Corp Unsaturated oxacycles
US3444176A (en) * 1967-04-28 1969-05-13 Mcneilab Inc Certain 4-diloweralkylamino-lower alkyl - 5 - pyridyl (or phenyl)-2,3-dihydro - 1 - benzothiepins and derivatives thereof

Also Published As

Publication number Publication date
EP0067086B1 (fr) 1985-12-11
EP0067086A1 (fr) 1982-12-15
AU8341782A (en) 1982-11-18
ES8303395A1 (es) 1983-03-01
DE3267884D1 (en) 1986-01-23
CA1196637A (fr) 1985-11-12
US4436749A (en) 1984-03-13
AU548253B2 (en) 1985-12-05

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