ES533537A0 - Triazol (2,3-c)pirimidin-aminas(-amidas) - Google Patents

Triazol (2,3-c)pirimidin-aminas(-amidas)

Info

Publication number
ES533537A0
ES533537A0 ES533537A ES533537A ES533537A0 ES 533537 A0 ES533537 A0 ES 533537A0 ES 533537 A ES533537 A ES 533537A ES 533537 A ES533537 A ES 533537A ES 533537 A0 ES533537 A0 ES 533537A0
Authority
ES
Spain
Prior art keywords
pirimidin
amids
triazol
amines
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES533537A
Other languages
English (en)
Other versions
ES8506714A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GD Searle LLC
Original Assignee
GD Searle LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by GD Searle LLC filed Critical GD Searle LLC
Publication of ES533537A0 publication Critical patent/ES533537A0/es
Publication of ES8506714A1 publication Critical patent/ES8506714A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES533537A 1983-06-20 1984-06-19 Triazol (2,3-c)pirimidin-aminas(-amidas) Expired ES8506714A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/506,157 US4483987A (en) 1983-06-20 1983-06-20 8-Substituted 7-phenyl-1,2,4-triazolo[2,3-c]pyrimidines-5-amines and amides

Publications (2)

Publication Number Publication Date
ES533537A0 true ES533537A0 (es) 1985-08-01
ES8506714A1 ES8506714A1 (es) 1985-08-01

Family

ID=24013440

Family Applications (1)

Application Number Title Priority Date Filing Date
ES533537A Expired ES8506714A1 (es) 1983-06-20 1984-06-19 Triazol (2,3-c)pirimidin-aminas(-amidas)

Country Status (7)

Country Link
US (1) US4483987A (es)
EP (1) EP0129247A1 (es)
JP (1) JPS6013792A (es)
AU (1) AU566670B2 (es)
CA (1) CA1204741A (es)
ES (1) ES8506714A1 (es)
ZA (1) ZA844669B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3130633A1 (de) * 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
US4562192A (en) * 1984-02-03 1985-12-31 G. D. Searle & Co. 6-Substituted-5-phenyltetrazolo[1,5-a][1,2,4]triazole[1,5-c]pyrimidines, and pharmaceutical compositions containing them
JPS62107954A (ja) * 1985-11-05 1987-05-19 Tomiji Saito 可塑性研磨材料
EP0244948A3 (en) * 1986-04-30 1989-03-15 Schering Agrochemicals Limited Triazolopyrimidine herbicides
JPH07115284B2 (ja) * 1986-07-18 1995-12-13 株式会社東芝 非球面部材のみがき装置
US5338743A (en) * 1988-06-06 1994-08-16 Fujisawa Pharmaceutical Co., Ltd. New use of the adenosine antagonist
US4866063A (en) * 1988-12-22 1989-09-12 G. D. Searle & Co. Diol metabolites of 7-phenyl-1,2,4-triazolo[2,3-c]pyrimidines-5-amines
FR2687676B1 (fr) * 1992-02-24 1994-07-08 Union Pharma Scient Appl Nouveaux derives de polyazaindenes antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.
WO1998042711A1 (en) * 1997-03-24 1998-10-01 Kyowa Hakko Kogyo Co., Ltd. [1,2,4]TRIAZOLO[1,5-c]PYRIMIDINE DERIVATIVES
KR20010087361A (ko) 1998-09-22 2001-09-15 히라타 다다시 [1,2,4]트리아졸로[1,5-c]피리미딘 유도체
JP2001302667A (ja) * 2000-04-28 2001-10-31 Bayer Ag イミダゾピリミジン誘導体およびトリアゾロピリミジン誘導体
US6998148B1 (en) 2001-03-28 2006-02-14 Shipley Company, L.L.C. Porous materials
EP2292278B1 (en) * 2001-11-16 2013-04-24 Children's Medical Center Corporation Augmentation of organ function
AU2003272886A1 (en) * 2002-09-24 2004-04-19 Kyowa Hakko Kogyo Co., Ltd. (1,2,4)-TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVE
US12414952B2 (en) 2018-11-20 2025-09-16 Merck Sharp & Dohme Llc Substituted amino triazolopyrimidine and amino triazolopyrazine adenosine receptor antagonists, pharmaceutical compositions and their use

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3053844A (en) * 1959-04-13 1962-09-11 Ici Ltd Mono-acyl derivatives of s-triazolo [2, 3-c] pyrimidines
US3046276A (en) * 1959-06-15 1962-07-24 Ici Ltd S-triazolo-[2, 3-c] pyrimidine derivatives
US4205169A (en) * 1979-04-09 1980-05-27 G. D. Searle & Co. N-[4-Azido-5-(2-ethoxyethyl)-6-phenyl-2-pyrimidinyl]acetamide and congeners
US4405780A (en) * 1979-08-08 1983-09-20 G. D. Searle & Co. 8-Substituted 7-phenyl-1,2,4,-triazolo[4,3-c]/[2,3-c]pyrimidines-5-amines and amides
DE3029871C2 (de) * 1979-08-08 1987-01-15 G.D. Searle & Co., Skokie, Ill. 8-(2-Ethoxyethyl)-7-phenyl-1,2,4-triazolo[1,5-c]pyrimidin-5-amin, Verfahren zu dessen Herstellung und pharmazeutische Zubereitung, die diese Verbindung enthält
US4269980A (en) * 1979-12-17 1981-05-26 American Cyanamid Company (Substituted-phenyl)-1,2,4-triazolo[4,3-c]pyrimidines and (substituted-phenyl)-1,2,4-triazolo[1,5-c]pyrimidines

Also Published As

Publication number Publication date
AU566670B2 (en) 1987-10-29
ZA844669B (en) 1985-08-28
JPH0471074B2 (es) 1992-11-12
AU2949484A (en) 1985-01-03
ES8506714A1 (es) 1985-08-01
EP0129247A1 (en) 1984-12-27
CA1204741A (en) 1986-05-20
JPS6013792A (ja) 1985-01-24
US4483987A (en) 1984-11-20

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970505