ES540332A0 - Procedimiento para preparar nuevos pirimido (2,1-b) benzo- tiazoles - Google Patents

Procedimiento para preparar nuevos pirimido (2,1-b) benzo- tiazoles

Info

Publication number: ES540332A0
Authority: ES; Spain
Prior art keywords: group; branched; straight; hydrogen atom; alkyl
Prior art date: 1984-02-13
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

ES540332A

Other languages

English (en)

Other versions

ES8702421A1 (es

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sanofi Aventis France

Original Assignee

Roussel Uclaf SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-02-13

Filing date

1985-02-12

Publication date

1986-12-16

1985-02-12 Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA

1986-12-16 Publication of ES540332A0 publication Critical patent/ES540332A0/es

1986-12-16 Publication of ES8702421A1 publication Critical patent/ES8702421A1/es

Status Expired legal-status Critical Current

Links

125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 2
125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
239000000043 antiallergic agent Substances 0.000 abstract 1
125000003710 aryl alkyl group Chemical group 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
229910052799 carbon Inorganic materials 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
125000001072 heteroaryl group Chemical group 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
125000000587 piperidin-1-yl group Chemical group [H]C1([H])N(*)C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pulmonology (AREA)
Public Health (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Luminescent Compositions (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Saccharide Compounds (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Polymerisation Methods In General (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Indole Compounds (AREA)
Compositions Of Macromolecular Compounds (AREA)

ES540332A 1984-02-13 1985-02-12 Procedimiento para preparar nuevos pirimido (2,1-b) benzo- tiazoles Expired ES8702421A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB848403739A GB8403739D0 (en)	1984-02-13	1984-02-13	Chemical compounds

Publications (2)

Publication Number	Publication Date
ES540332A0 true ES540332A0 (es)	1986-12-16
ES8702421A1 ES8702421A1 (es)	1986-12-16

Family

ID=10556508

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
ES540332A Expired ES8702421A1 (es)	1984-02-13	1985-02-12	Procedimiento para preparar nuevos pirimido (2,1-b) benzo- tiazoles
ES553574A Expired ES8800243A1 (es)	1984-02-13	1986-04-01	Procedimiento para preparar nuevos pirimido(2,1-b)benzotiazoles

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
ES553574A Expired ES8800243A1 (es)	1984-02-13	1986-04-01	Procedimiento para preparar nuevos pirimido(2,1-b)benzotiazoles

Country Status (16)

Country	Link
EP (1)	EP0153230B1 (es)
JP (1)	JPS60184086A (es)
KR (1)	KR850005847A (es)
AT (1)	ATE44745T1 (es)
AU (1)	AU574131B2 (es)
CA (1)	CA1257259A (es)
DE (1)	DE3571621D1 (es)
DK (1)	DK63385A (es)
ES (2)	ES8702421A1 (es)
FI (1)	FI79323C (es)
GB (2)	GB8403739D0 (es)
GR (1)	GR850369B (es)
HU (1)	HU192318B (es)
NZ (1)	NZ211104A (es)
PT (1)	PT79955B (es)
ZA (1)	ZA85696B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8519261D0 (en) *	1985-07-31	1985-09-04	Roussel Lab Ltd	Chemical compounds
US4762840A (en) *	1984-02-13	1988-08-09	Roussel Uclaf	Pyrimido[2,1-b]benzothiazoles having antiallergic activity
AP2013006706A0 (en)	2010-07-02	2013-02-28	Gilead Sciences Inc	Napht-2-ylacetic acid derivatives to treat AIDS
KR20130124291A (ko)	2010-07-02	2013-11-13	길리애드 사이언시즈, 인코포레이티드	Ｈｉｖ 항바이러스 화합물로서의 2-퀴놀리닐-아세트산 유도체
BR112013027096A2 (pt)	2011-04-21	2016-12-27	Gilead Sciences Inc	compostos de benzotiazol e seu uso farmacêutico
US9284323B2 (en)	2012-01-04	2016-03-15	Gilead Sciences, Inc.	Naphthalene acetic acid derivatives against HIV infection
WO2013103724A1 (en)	2012-01-04	2013-07-11	Gilead Sciences, Inc.	2- (tert - butoxy) -2- (7 -methylquinolin- 6 - yl) acetic acid derivatives for treating aids
ES2571479T3 (es)	2012-04-20	2016-05-25	Gilead Sciences Inc	Derivados del ácido benzotiazol-6-il acético y su uso para tratar una infección por VIH

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3919201A (en) *	1970-09-30	1975-11-11	Lilly Industries Ltd	2-({62 -Aminoacryloyl)iminobenzothiazolines
DE2810863A1 (de) *	1978-03-13	1979-09-27	Boehringer Mannheim Gmbh	1-oxo-1h-pyrimido eckige klammer auf 6,1-b eckige klammer zu benzthiazol-derivate und verfahren zu ihrer herstellung
GB8519261D0 (en) *	1985-07-31	1985-09-04	Roussel Lab Ltd	Chemical compounds

1984
- 1984-02-13 GB GB848403739A patent/GB8403739D0/en active Pending
1985
- 1985-01-13 KR KR1019850000879A patent/KR850005847A/ko not_active Ceased
- 1985-01-29 ZA ZA85696A patent/ZA85696B/xx unknown
- 1985-02-11 DE DE8585400219T patent/DE3571621D1/de not_active Expired
- 1985-02-11 EP EP85400219A patent/EP0153230B1/fr not_active Expired
- 1985-02-11 AT AT85400219T patent/ATE44745T1/de not_active IP Right Cessation
- 1985-02-12 NZ NZ211104A patent/NZ211104A/en unknown
- 1985-02-12 FI FI850582A patent/FI79323C/fi not_active IP Right Cessation
- 1985-02-12 JP JP60023706A patent/JPS60184086A/ja active Pending
- 1985-02-12 HU HU85529A patent/HU192318B/hu not_active IP Right Cessation
- 1985-02-12 ES ES540332A patent/ES8702421A1/es not_active Expired
- 1985-02-12 GB GB08503541A patent/GB2154583B/en not_active Expired
- 1985-02-12 CA CA000474113A patent/CA1257259A/en not_active Expired
- 1985-02-12 GR GR850369A patent/GR850369B/el unknown
- 1985-02-12 PT PT79955A patent/PT79955B/pt not_active IP Right Cessation
- 1985-02-12 DK DK63385A patent/DK63385A/da not_active Application Discontinuation
- 1985-02-13 AU AU38672/85A patent/AU574131B2/en not_active Ceased
1986
- 1986-04-01 ES ES553574A patent/ES8800243A1/es not_active Expired

Also Published As

Publication number	Publication date
HUT38649A (en)	1986-06-30
DK63385D0 (da)	1985-02-12
GR850369B (es)	1985-06-14
GB2154583A (en)	1985-09-11
FI79323C (fi)	1989-12-11
NZ211104A (en)	1987-08-31
FI850582L (fi)	1985-08-14
CA1257259A (en)	1989-07-11
PT79955A (en)	1985-03-01
KR850005847A (ko)	1985-09-26
ZA85696B (en)	1986-03-26
ES8800243A1 (es)	1987-10-16
DE3571621D1 (en)	1989-08-24
JPS60184086A (ja)	1985-09-19
PT79955B (en)	1987-02-02
ES553574A0 (es)	1987-10-16
GB2154583B (en)	1987-10-28
ATE44745T1 (de)	1989-08-15
EP0153230B1 (fr)	1989-07-19
HU192318B (en)	1987-05-28
EP0153230A3 (en)	1986-10-01
FI850582A0 (fi)	1985-02-12
FI79323B (fi)	1989-08-31
GB8503541D0 (en)	1985-03-13
AU574131B2 (en)	1988-06-30
ES8702421A1 (es)	1986-12-16
GB8403739D0 (en)	1984-03-14
DK63385A (da)	1985-08-14
AU3867285A (en)	1985-08-22
EP0153230A2 (fr)	1985-08-28

Legal Events

Date	Code	Title	Description
1996-08-16	FD1A	Patent lapsed	Effective date: 19960603

Publication	Publication Date	Title
DE3588100D1 (de)	1996-05-23	Carbamidsäureester-Derivate, Mittel und Herstellungsverfahren
ES533916A0 (es)	1985-12-01	Un metodo para producir acidos 1,4-dihidro-4-oxo-quinolin-3-carboxilico
ES540332A0 (es)	1986-12-16	Procedimiento para preparar nuevos pirimido (2,1-b) benzo- tiazoles
ES8604543A1 (es)	1986-02-01	Procedimiento para la obtencion de derivados piperazinicos
ATE28639T1 (de)	1987-08-15	Derivate von 4-(3-alkynyloxy-2-hydroxy-propyl)piperazin-1-yl-n-phenylacetamid, ihre herstellung und ihre therapeutische verwendung.
ATE30415T1 (de)	1987-11-15	Enkephalinas-inhibitoren.
AU586010B2 (en)	1989-06-29	Pyrimido``2,1-b`` benzothiazole derivatives
FI824298L (fi)	1983-06-15	N,n-disubstituerade alkenamider och fenylalkenamider, deras framstaellningsfoerfaranden och anvaendning som laekemedel