ES544117A0 - Procedimiento para preparar nuevos bencimidazoles - Google Patents

Procedimiento para preparar nuevos bencimidazoles

Info

Publication number
ES544117A0
ES544117A0 ES544117A ES544117A ES544117A0 ES 544117 A0 ES544117 A0 ES 544117A0 ES 544117 A ES544117 A ES 544117A ES 544117 A ES544117 A ES 544117A ES 544117 A0 ES544117 A0 ES 544117A0
Authority
ES
Spain
Prior art keywords
benzmidazoles
procedure
prepare new
prepare
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES544117A
Other languages
English (en)
Other versions
ES8604163A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Publication of ES8604163A1 publication Critical patent/ES8604163A1/es
Publication of ES544117A0 publication Critical patent/ES544117A0/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/18Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ES544117A 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles Expired ES8604163A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3346575A DE3346575A1 (de) 1983-12-23 1983-12-23 Neue benzimidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
ES8604163A1 ES8604163A1 (es) 1986-01-16
ES544117A0 true ES544117A0 (es) 1986-01-16

Family

ID=6217793

Family Applications (5)

Application Number Title Priority Date Filing Date
ES538929A Granted ES538929A0 (es) 1983-12-23 1984-12-21 Procedimiento para preparar bencimidazoles
ES544118A Expired ES8604164A1 (es) 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles
ES544119A Expired ES8604165A1 (es) 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles
ES544116A Expired ES8604162A1 (es) 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles
ES544117A Expired ES8604163A1 (es) 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles

Family Applications Before (4)

Application Number Title Priority Date Filing Date
ES538929A Granted ES538929A0 (es) 1983-12-23 1984-12-21 Procedimiento para preparar bencimidazoles
ES544118A Expired ES8604164A1 (es) 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles
ES544119A Expired ES8604165A1 (es) 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles
ES544116A Expired ES8604162A1 (es) 1983-12-23 1985-06-13 Procedimiento para preparar nuevos bencimidazoles

Country Status (14)

Country Link
EP (1) EP0148431A1 (es)
JP (1) JPS60156676A (es)
KR (1) KR850004467A (es)
AU (1) AU3704284A (es)
DD (1) DD232697A5 (es)
DE (1) DE3346575A1 (es)
DK (1) DK597484A (es)
ES (5) ES538929A0 (es)
FI (1) FI845084A7 (es)
HU (1) HU193073B (es)
IL (1) IL73897A0 (es)
NO (1) NO845169L (es)
PT (1) PT79718B (es)
ZA (1) ZA849972B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU85544A1 (fr) * 1984-09-19 1986-04-03 Cird Derives heterocycliques aromatiques,leur procede de preparation et leur application dans les domaines therapeutique et cosmetique
DE3522230A1 (de) * 1985-06-21 1987-01-02 Thomae Gmbh Dr K Neue 2-arylimidazole, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung
FR2677020B1 (fr) * 1991-05-31 1993-08-27 Cird Galderma Composes derives de benzimidazole, leur procede de preparation et leur utilisation dans les domaines therapeutique et cosmetique.
US5821258A (en) * 1994-12-27 1998-10-13 Mitsui Chemicals, Inc. Phenylbenzimidazole derivatives
PT841924E (pt) * 1995-08-02 2003-02-28 Univ Newcastle Ventures Ltd Compostos de benzimidazolo
US5942532A (en) * 1997-09-05 1999-08-24 Ortho Pharmaceutical Corporation 2-substituted phenyl-benzimidazole antibacterial agents
DE60221866T2 (de) 2001-10-19 2008-05-29 Ortho-Mcneil Pharmaceutical, Inc. 2-PHENYL BENZIMIDAZOLE UND IMIDAZO-i4,5ö-PYRIDINE ALS CDS1/CHK2-INHIBITOREN UND ADJUVANTIEN IN DER CHEMOTHERAPIE ODER STRAHLUNGSTHERAPIE ZUR BEHANDLUNG VON KREBS
JP2006513159A (ja) * 2002-11-01 2006-04-20 メルク エンド カムパニー インコーポレーテッド アンドロゲン受容体モジュレーターとしてのカルボニルアミノ−ベンズイミダゾール誘導体
DE602004006852D1 (de) 2003-04-17 2007-07-19 Janssen Pharmaceutica Nv 2-phenyl-benzimidazol und 2-phenyl-imidazo-4,5ü-pyridin-derivate als checkpoint-kinase-cds1 (chk2)-hemmer zur behandlung von krebs
DE602005027739D1 (de) 2004-06-30 2011-06-09 Janssen Pharmaceutica Nv Arylsubstituiertes benzimidazol- und imidazopyridinether als wirkstoffe gegen krebs
BR112013016022B1 (pt) 2010-12-24 2019-05-07 Sumitomo Chemical Company, Limited Composto heterocíclico fundido e uso do mesmo para controle de peste.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH350763A (de) * 1958-10-14 1960-12-15 Ciba Geigy Verwendung von Azolverbindungen als Schutzmittel gegen ultraviolette Strahlung
DE1447733B2 (de) * 1963-12-23 1977-04-21 Hoechst Ag, 6000 Frankfurt 2-(3,5-dihydroxyphenyl)-benzimidazolderivate
IL23847A (en) * 1964-08-07 1969-02-27 Merck & Co Inc Benzimidazoles useful as antifungals
FR1569337A (es) * 1968-06-18 1969-05-30
DE2742093A1 (de) * 1977-09-19 1979-03-29 Cassella Ag Verfahren zur herstellung von 2-(3'- bzw. 4'-aminophenyl)-5(bzw. 6) -aminobenzimidazolen
DE2927987A1 (de) * 1979-07-11 1981-02-05 Thomae Gmbh Dr K Neue 2-alkoxyphenyl-imidazo eckige klammer auf 4,5-b eckige klammer zu pyridine, deren herstellung und deren verwendung als arzneimittel
DE3224512A1 (de) * 1982-07-01 1984-01-05 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazolderivate, ihre herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
AU3704284A (en) 1985-07-04
ES544116A0 (es) 1986-01-16
ES8604163A1 (es) 1986-01-16
ES544119A0 (es) 1986-01-16
FI845084A0 (fi) 1984-12-21
DK597484A (da) 1985-06-24
ES8604164A1 (es) 1986-01-16
ES8601913A1 (es) 1985-11-16
ES8604162A1 (es) 1986-01-16
PT79718A (de) 1985-01-01
DE3346575A1 (de) 1985-07-04
ES538929A0 (es) 1985-11-16
EP0148431A1 (de) 1985-07-17
HUT37763A (en) 1986-02-28
JPS60156676A (ja) 1985-08-16
KR850004467A (ko) 1985-07-15
NO845169L (no) 1985-06-24
PT79718B (de) 1986-12-30
DD232697A5 (de) 1986-02-05
ES8604165A1 (es) 1986-01-16
FI845084L (fi) 1985-06-24
FI845084A7 (fi) 1985-06-24
ES544118A0 (es) 1986-01-16
IL73897A0 (en) 1985-03-31
ZA849972B (en) 1986-08-27
HU193073B (en) 1987-08-28
DK597484D0 (da) 1984-12-13

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