ES556754A0 - Un procedimiento para preparar derivados de acido piridoncarboxilico - Google Patents

Un procedimiento para preparar derivados de acido piridoncarboxilico

Info

Publication number: ES556754A0
Authority: ES; Spain
Prior art keywords: sup; sub; acid; piridoncarboxilico; procedure
Prior art date: 1985-06-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

ES556754A

Other languages

English (en)

Other versions

ES8707520A1 (es

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Daiichi Pharmaceutical Co Ltd

Original Assignee

Daiichi Pharmaceutical Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-06-26

Filing date

1986-06-25

Publication date

1987-08-01

1986-06-25 Application filed by Daiichi Pharmaceutical Co Ltd filed Critical Daiichi Pharmaceutical Co Ltd

1987-08-01 Publication of ES556754A0 publication Critical patent/ES556754A0/es

1987-08-01 Publication of ES8707520A1 publication Critical patent/ES8707520A1/es

Status Expired legal-status Critical Current

Links

239000002253 acid Substances 0.000 title abstract 2
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
125000004777 2-fluoroethyl group Chemical group [H]C([H])(F)C([H])([H])* 0.000 abstract 1
125000006414 CCl Chemical group ClC* 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
230000000845 anti-microbial effect Effects 0.000 abstract 1
125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 abstract 1
125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
125000000555 isopropenyl group Chemical group [H]\C([H])=C(\*)C([H])([H])[H] 0.000 abstract 1
125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 abstract 1
229920002554 vinyl polymer Polymers 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Table Devices Or Equipment (AREA)
Stringed Musical Instruments (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

ES556754A 1985-06-26 1986-06-25 Un procedimiento para preparar derivados de acido piridoncarboxilico Expired ES8707520A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP13983085		1985-06-26
JP27999185		1985-12-12

Publications (2)

Publication Number	Publication Date
ES556754A0 true ES556754A0 (es)	1987-08-01
ES8707520A1 ES8707520A1 (es)	1987-08-01

Family

ID=26472527

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ES556754A Expired ES8707520A1 (es)	1985-06-26	1986-06-25	Un procedimiento para preparar derivados de acido piridoncarboxilico

Country Status (18)

Country	Link
US (4)	US5098912A (es)
EP (1)	EP0207420B1 (es)
JP (2)	JPH0745491B2 (es)
KR (1)	KR930005001B1 (es)
AT (1)	ATE75740T1 (es)
AU (1)	AU589978B2 (es)
CA (1)	CA1301760C (es)
DE (1)	DE3685157D1 (es)
DK (1)	DK170641B1 (es)
ES (1)	ES8707520A1 (es)
FI (1)	FI87071C (es)
GR (1)	GR861649B (es)
IE (1)	IE59188B1 (es)
IL (1)	IL79189A (es)
NO (1)	NO167090C (es)
PH (1)	PH24886A (es)
PT (1)	PT82839B (es)
YU (1)	YU46526B (es)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3508816A1 (de) *	1985-01-10	1986-07-10	Bayer Ag, 5090 Leverkusen	6,7-disubstituierte 1-cyclopropyl-1,4-dihydro-4-oxo-1,8-naphtyridin-3-carbonsaeuren
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents
US5585491A (en) *	1988-01-25	1996-12-17	Otsuka Pharmaceutical Co., Ltd.	Antibacterial agents
CA1332605C (en) *	1988-10-03	1994-10-18	Yasuhiro Nishitani	Pyridonecarboxylic acids
US5364861A (en) *	1990-11-30	1994-11-15	Warner-Lambert Company	Optical isomers of 7-[3-(1,1-dialkylmethyl-1-amino-1-pyrrolidinyl]-quinolones and naphthyridones as antibacterial agents
DE69131428T2 (de) *	1990-11-30	2000-01-05	Warner-Lambert Co., Ann Arbor	Individuelle stereoisomere von 7-[3-(aminoalkyl)-1-pyrrolidinyl]-quinolone und naphthyridone als antibakterielle wirkstoffe
US5157128A (en) *	1990-11-30	1992-10-20	Warner-Lambert Company	Certain optically active substituted α,α-dialkyl-pyrrolidine-3-methamines useful as intermediates
US5258528A (en) *	1990-11-30	1993-11-02	Warner-Lambert Company	Individual stereoisomers of pyrrolidine methanamines substituted on the ring nitrogen by a 1-phenylethyl group
EP0550016A1 (en) *	1991-12-31	1993-07-07	Korea Research Institute Of Chemical Technology	Novel quinolone carboxylic acid derivatives and processes for preparing same
PT807630E (pt) *	1995-02-02	2003-08-29	Daiichi Seiyaku Co	Compostos heterociclicos
JP4040091B2 (ja) *	1995-11-22	2008-01-30	第一三共株式会社	置換アミノシクロアルキルピロリジン誘導体
US6121285A (en)	1995-11-22	2000-09-19	Daiichi Pharmaceutical Co., Ltd.	Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
AU3459797A (en)	1996-07-12	1998-02-09	Daiichi Pharmaceutical Co., Ltd.	Cis-substituted aminocyclopropane derivatives
CN1263527A (zh) *	1997-05-21	2000-08-16	第一制药株式会社	顺式取代－取代氨基环烷基吡咯烷衍生物
MY119816A (en) *	1997-05-30	2005-07-29	Daiichi Seiyaku Co	Substituted cyclobutylamine derivatives
US6387928B1 (en)	1997-09-15	2002-05-14	The Procter & Gamble Co.	Antimicrobial quinolones, their compositions and uses
CN1264837C (zh) *	1997-09-15	2006-07-19	普罗克特和甘保尔公司	喹诺酮抗微生物剂、其组合物和应用
EP1082300B1 (en) *	1998-05-29	2003-09-10	PHARMACIA & UPJOHN COMPANY	3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidine monomethanesulfonate
CN1258531C (zh)	1999-03-10	2006-06-07	第一制药株式会社	芳香族取代基取代的氨基甲基吡咯烷衍生物
US6569686B2 (en) *	2000-01-28	2003-05-27	Pion, Inc.	Measurement of solubility-pH profiles
PT1336611E (pt) *	2000-11-20	2007-12-06	Daiichi Sankyo Co Ltd	Compostos desalogenados
PL1666477T3 (pl)	2003-09-10	2013-11-29	Kyorin Seiyaku Kk	Pochodna kwasu 7-(4-podstawionego-3-cyklopropyloaminometylo-1- pirolidynylo)chinolonokarboksylowego
WO2005030752A1 (ja) *	2003-09-29	2005-04-07	Daiichi Pharmaceutical Co., Ltd.	８−シアノキノロンカルボン酸誘導体
ES2366150T3 (es) *	2006-03-28	2011-10-17	Warner Chilcott Company, Llc	Malatos de polimorfos de ácido (3s,5s)-7-[3-amino-5-metil-piperidinil]-1-ciclopropil-1,4-dihidro-8-metoxi-4-oxo-3-quinolinocarboxílico.
CA2647454A1 (en) *	2006-03-28	2007-10-04	The Procter & Gamble Company	A coupling process for preparing quinolone intermediates
BRPI0709209A2 (pt) *	2006-03-28	2011-06-28	Procter & Gamble	processo de redução de hidreto para preparo de intermediários de quinolona
JP5322927B2 (ja) *	2007-05-24	2013-10-23	杏林製薬株式会社	１４位置換基に複素芳香環カルボン酸構造を有するムチリン誘導体
CN116606280A (zh) *	2023-03-13	2023-08-18	广东工业大学	一种氟喹诺酮类化合物及其在制备抗菌药物中的应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4665079A (en) *	1984-02-17	1987-05-12	Warner-Lambert Company	Antibacterial agents
IE55898B1 (en) *	1982-09-09	1991-02-14	Warner Lambert Co	Antibacterial agents
DE3318145A1 (de) *	1983-05-18	1984-11-22	Bayer Ag, 5090 Leverkusen	7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
JPS60228479A (ja) *	1984-04-26	1985-11-13	Toyama Chem Co Ltd	１，４−ジヒドロ−４−オキソナフチリジン誘導体およびその塩
IE58742B1 (en) *	1984-07-20	1993-11-05	Warner Lambert Co	Substituted-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7h-pyrido[1,2,3-de] [1,4]benzoxauine-6-carboxylic acids; sibstituted-5-amino-6-6fluoro-4-oxo.1,4-dihydroquinoline-3 carboxylic acids; substituted-5-amino-6-fluoro-1,4-dihydro-4-oxo-1.8-naphthyridine-3-carboxylic acids; derivatives thereof; pharmaceutical compositions comprising the compounds; and processes for producing the compounds
DE3509546A1 (de) *	1985-03-16	1986-09-25	Bayer Ag, 5090 Leverkusen	7-amino-1-(subst.cyclopropyl)-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
US4657913A (en) *	1985-04-18	1987-04-14	Warner-Lambert Company	Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents
EP0242789A3 (en) *	1986-04-25	1990-09-05	Dainippon Pharmaceutical Co., Ltd.	Novel quinoline derivates and processes for preparation thereof
US4851418A (en) *	1987-08-21	1989-07-25	Warner-Lambert Company	Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents

1986
- 1986-06-23 AT AT86108547T patent/ATE75740T1/de not_active IP Right Cessation
- 1986-06-23 EP EP86108547A patent/EP0207420B1/en not_active Expired - Lifetime
- 1986-06-23 DE DE8686108547T patent/DE3685157D1/de not_active Expired - Lifetime
- 1986-06-23 IL IL79189A patent/IL79189A/xx not_active IP Right Cessation
- 1986-06-24 FI FI862688A patent/FI87071C/fi not_active IP Right Cessation
- 1986-06-25 PT PT82839A patent/PT82839B/pt unknown
- 1986-06-25 AU AU59245/86A patent/AU589978B2/en not_active Expired
- 1986-06-25 GR GR861649A patent/GR861649B/el unknown
- 1986-06-25 IE IE169686A patent/IE59188B1/en not_active IP Right Cessation
- 1986-06-25 CA CA000512446A patent/CA1301760C/en not_active Expired - Lifetime
- 1986-06-25 ES ES556754A patent/ES8707520A1/es not_active Expired
- 1986-06-25 NO NO862559A patent/NO167090C/no not_active IP Right Cessation
- 1986-06-26 YU YU112086A patent/YU46526B/sh unknown
- 1986-06-26 KR KR1019860005150A patent/KR930005001B1/ko not_active Expired - Lifetime
- 1986-06-26 DK DK304686A patent/DK170641B1/da not_active IP Right Cessation
- 1986-06-26 PH PH33956A patent/PH24886A/en unknown
- 1986-06-26 JP JP61150581A patent/JPH0745491B2/ja not_active Expired - Lifetime
1989
- 1989-12-12 US US07/449,160 patent/US5098912A/en not_active Expired - Lifetime
1991
- 1991-12-24 US US07/812,830 patent/US5416222A/en not_active Expired - Lifetime
1993
- 1993-06-21 JP JP5148887A patent/JP2686705B2/ja not_active Expired - Lifetime
1994
- 1994-03-04 US US08/205,638 patent/US5380874A/en not_active Expired - Lifetime
1995
- 1995-03-20 US US08/406,594 patent/US5476950A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
FI87071B (fi)	1992-08-14
DK304686A (da)	1987-02-23
JPH09143157A (ja)	1997-06-03
JPS62234082A (ja)	1987-10-14
KR870000321A (ko)	1987-02-17
US5380874A (en)	1995-01-10
EP0207420A3 (en)	1988-04-20
PT82839B (pt)	1988-04-21
US5416222A (en)	1995-05-16
YU46526B (sh)	1993-11-16
EP0207420B1 (en)	1992-05-06
AU589978B2 (en)	1989-10-26
FI87071C (fi)	1992-11-25
IL79189A0 (en)	1986-09-30
AU5924586A (en)	1987-01-08
ATE75740T1 (de)	1992-05-15
PT82839A (en)	1986-07-01
NO167090B (no)	1991-06-24
YU112086A (en)	1991-04-30
IE861696L (en)	1986-12-26
EP0207420A2 (en)	1987-01-07
DE3685157D1 (de)	1992-06-11
NO862559L (no)	1986-12-29
IE59188B1 (en)	1994-01-26
IL79189A (en)	1990-07-12
DK304686D0 (da)	1986-06-26
PH24886A (en)	1990-12-26
GR861649B (en)	1986-10-30
FI862688L (fi)	1986-12-27
JPH0745491B2 (ja)	1995-05-17
JP2686705B2 (ja)	1997-12-08
NO862559D0 (no)	1986-06-25
FI862688A0 (fi)	1986-06-24
DK170641B1 (da)	1995-11-20
KR930005001B1 (ko)	1993-06-11
NO167090C (no)	1991-10-02
CA1301760C (en)	1992-05-26
ES8707520A1 (es)	1987-08-01
US5098912A (en)	1992-03-24
US5476950A (en)	1995-12-19

Legal Events

Date	Code	Title	Description
2008-06-16	FD1A	Patent lapsed	Effective date: 20070530

Publication	Publication Date	Title
PT82839B (pt)	1988-04-21	Processo para a preparacao de derivados de acido piridonocarboxilico
IL81002A0 (en)	1987-03-31	Pyrazoline derivatives,processes for their preparation and pesticidal compositions containing the same
ES8502106A1 (es)	1980-07-16	Un procedimiento para la preparacion de derivados de diben- zopirano
ES8702371A1 (es)	1986-12-16	Un procedimiento para preparar nuevos derivados de 6-(4-fenilo sustituido -3(2h) piradazinona.
ES2008962A6 (es)	1989-08-16	Proceso para la preparacion de nuevos compuestos de 2-guanidinotiazol
ES8505956A1 (es)	1985-06-01	Procedimiento para la preparacion de nuevas 5-acil-2-(1h)-piridinonas.
DE3672446D1 (en)	1990-08-09	Pantothenolderivate.
GB2162182B (en)	1989-04-12	Pharmaceutical compounds and their preparation
IT8621229A0 (it)	1986-07-23	Procedimento per la preparazione di nitrato di potassio.
ES2001670A6 (es)	1988-06-01	Procedimiento para preparar derivados de fenoxiftalida y composiciones herbicidas que los contienen
EP0210642A3 (en)	1989-02-22	Surfactants derived from succinic acid
IT8024975A0 (it)	1980-09-26	Preparazione di acido 2,5-dichetogluconico.
DE3070667D1 (en)	1985-06-27	Pyrimidine compounds, their preparation, herbicidal compositions containing them as active compounds and intermediates thereof
BR8600034A (pt)	1986-09-23	Composto de eter de fenila e processo de preparacao
ES8601931A1 (es)	1985-11-16	Procedimiento para preparar imidazoles y triazoles con es- tructura de enoleter
ES542611A0 (es)	1987-06-01	Procedimiento de preparacion de nuevas composiciones sinergeticas antimicrobianas que contienen aritetraciclina y un acido organico de acitividad antimicrobiana.
IL67526A (en)	1986-07-31	Fluorophenoxybenzyl-2,2-dimethyl-3-oximino-methyl cyclopropane derivatives,their preparation and pesticidal compositions containing them
SU1363769A1 (ru)	1999-08-27	Метиловый эфир 4-дифенилметилиденгидразино-2-оксо-4-фенил-3-бутеновой кислоты, проявляющий противовоспалительную активность
EP0143381A3 (en)	1986-04-02	Biphenylylalkanoic acid derivatives, methods of preparation and pharmaceutical compositions therefrom
FR2515649B1 (es)	1984-06-29
FI852260A0 (fi)	1985-06-05	Reglerbar baeranordning foer kastredskap.
JO1183B1 (en)	1983-11-30	Benzodine isoxazolyl compounds
SU892892A1 (ru)	2006-12-27	3-Дицианметилпиримидо-[4,5-е][1,2,4]-триазин-6,8-дион гидрат, обладающий противовоспалительной активностью