ES8205209A1 - Un procedimiento para la preparacion de un derivado de ben- zamida - Google Patents

Un procedimiento para la preparacion de un derivado de ben- zamida

Info

Publication number
ES8205209A1
ES8205209A1 ES505518A ES505518A ES8205209A1 ES 8205209 A1 ES8205209 A1 ES 8205209A1 ES 505518 A ES505518 A ES 505518A ES 505518 A ES505518 A ES 505518A ES 8205209 A1 ES8205209 A1 ES 8205209A1
Authority
ES
Spain
Prior art keywords
isoxazolylbenzamides
benzisoxazolyl
insecticides
isoxazolyl
directed
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES505518A
Other languages
English (en)
Other versions
ES505518A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES8205209A1 publication Critical patent/ES8205209A1/es
Publication of ES505518A0 publication Critical patent/ES505518A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/12—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines
    • C07C259/18—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines having carbon atoms of hydroxamidine groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/14—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE BENZAMIDA DE FORMULA (I), EN LA QUE R, R1 Y R2 PUEDEN SER VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE CONDENSACION DE UN HALURO DE BENZOILO DE FORMULA (II) CON UN AMINOISOXAZOL DE FORMULA HNR1R2, EN LAS QUE R, R1 Y R2 TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I) Y X ES HALOGENO. LA REACCION SE LLEVA A CABO EN UN DISOLVENTE ORGANICO INERTE EN PRESENCIA DE UN ACEPTOR DE ACIDO TAL COMO TRIETILAMINA O PIRIDINA Y A TEMPERATURAS ENTRE 10 Y 120 GRADOS CENTIGRADOS. ESTOS COMPUESTOS TIENEN APLICACIONES EN AGRICULTURA COMO INSECTICIDAS.
ES505518A 1980-09-16 1981-09-15 Un procedimiento para la preparacion de un derivado de ben- zamida Granted ES505518A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/187,677 US4322429A (en) 1980-09-16 1980-09-16 Isoxazolylbenzamides as insecticides

Publications (2)

Publication Number Publication Date
ES8205209A1 true ES8205209A1 (es) 1982-06-01
ES505518A0 ES505518A0 (es) 1982-06-01

Family

ID=22689988

Family Applications (1)

Application Number Title Priority Date Filing Date
ES505518A Granted ES505518A0 (es) 1980-09-16 1981-09-15 Un procedimiento para la preparacion de un derivado de ben- zamida

Country Status (19)

Country Link
US (1) US4322429A (es)
EP (1) EP0048162A1 (es)
JP (1) JPS5781476A (es)
KR (1) KR830007589A (es)
AR (1) AR231443A1 (es)
AU (1) AU7525681A (es)
BR (1) BR8105874A (es)
CA (1) CA1164871A (es)
ES (1) ES505518A0 (es)
GB (1) GB2084139B (es)
GR (1) GR75336B (es)
IL (1) IL63838A0 (es)
MA (1) MA19268A1 (es)
PT (1) PT73671B (es)
RO (1) RO83215B (es)
TR (1) TR20923A (es)
YU (1) YU221581A (es)
ZA (1) ZA816394B (es)
ZW (1) ZW23081A1 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5086184A (en) * 1980-09-16 1992-02-04 Dowelanco N-heterocyclic benzamides
US4636243A (en) * 1980-09-16 1987-01-13 Eli Lilly And Company Benzamides, compositions and agricultural method
US4943634A (en) * 1980-09-16 1990-07-24 Eli Lilly And Company N-heterocyclic benzamides
US4716233A (en) * 1985-08-15 1987-12-29 International Minerals & Chemical Corp. Process for preparing phthalimido isoxazoles
US4593024A (en) * 1985-08-15 1986-06-03 International Minerals & Chemical Corp. Dihydroisoxazole compounds and anthelmintic use
US4694016A (en) * 1985-10-18 1987-09-15 International Minerals & Chemical Corp. Phthalamide derivatives with anthelmintic activity
US4636517A (en) * 1985-10-18 1987-01-13 International Minerals & Chemical Corp. 3-tolylthio-4-amino-4,5-dihydro isoxazole as anthelmintic
FR2639636B1 (fr) * 1988-11-30 1994-03-04 Novapharme Nouveaux composes heterocycliques a activite anticonvulsivante, procede de preparation et compositions therapeutiques les contenant
FR2662692B1 (fr) * 1990-05-30 1995-04-28 Novapharme Derives heterocycliques doues d'activite anticonvulsivante, procede de preparation et composition pharmaceutique.
US5258397A (en) * 1988-11-30 1993-11-02 Novapharme 3-Isoxazoyl derivatives endowed with anticonvulsant activity, procedure for their preparation and their pharmaceutical compositions
JP2000514788A (ja) 1996-06-25 2000-11-07 イーライ・リリー・アンド・カンパニー 抗凝固剤
US6200967B1 (en) 1996-06-25 2001-03-13 Eli Lilly And Company Anticoagulant agents
JP3191943B2 (ja) * 1997-02-04 2001-07-23 ドン ワ ファーマシューティカル インダストリアル カンパニー リミテッド ３−アミノ−１，２−ベンゾイソオキサゾール誘導体類とその製造方法及び用途
DE102005026194A1 (de) * 2005-06-06 2006-12-07 Grünenthal GmbH Substituierte N-Benzo[d]isoxazol-3-yl-amin-Derivate und deren Verwendung zur Herstellung von Arzneimitteln
US7504513B2 (en) * 2006-02-27 2009-03-17 Hoffman-La Roche Inc. Thiazolyl-benzimidazoles
JP4518066B2 (ja) * 2006-10-25 2010-08-04 宇部興産株式会社 ジアルコキシニトリル誘導体及びその製法
JP2012512223A (ja) * 2008-12-18 2012-05-31 エフ．ホフマン−ラ ロシュ アーゲー チアゾリル−ベンズイミダゾール類

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3360516A (en) * 1961-06-23 1967-12-26 Dow Chemical Co N-[4-(2, 6-dimethylpyrimidyl)]3, 5-dinitrobenzamide
DE1668723A1 (de) 1966-09-16 1971-04-08 Toyo Jozo Kk Verfahren zum Herstellen von Verbindungen mit Saeureamid-Bindung
FR2088826A5 (en) * 1970-04-27 1972-01-07 Aries Robert Salicylamido isoxazoles - as antiseptics and antiparasitics from aminoisoxazoles and benzoyl halide derivs
US4062861A (en) * 1973-07-27 1977-12-13 Shionogi & Co., Ltd. 3-Isoxazolylurea derivatives
GB1548397A (en) * 1976-06-01 1979-07-11 Lilly Industries Ltd Acylated amino-isoxazoles and aminoisothiazoles

Also Published As

Publication number Publication date
YU221581A (en) 1983-09-30
GB2084139B (en) 1984-07-25
GB2084139A (en) 1982-04-07
IL63838A0 (en) 1981-12-31
JPS5781476A (en) 1982-05-21
ZW23081A1 (en) 1981-12-09
MA19268A1 (fr) 1982-04-01
TR20923A (tr) 1983-01-11
RO83215A (ro) 1984-02-21
PT73671A (en) 1981-10-01
EP0048162A1 (en) 1982-03-24
RO83215B (ro) 1984-02-28
GR75336B (es) 1984-07-13
ZA816394B (en) 1983-04-27
ES505518A0 (es) 1982-06-01
PT73671B (en) 1982-11-22
BR8105874A (pt) 1982-06-08
US4322429A (en) 1982-03-30
KR830007589A (ko) 1983-11-04
AR231443A1 (es) 1984-11-30
AU7525681A (en) 1982-03-25
CA1164871A (en) 1984-04-03

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