ES8601152A1 - Procedimiento para la obtencion de derivados de acido barbi-turico - Google Patents

Procedimiento para la obtencion de derivados de acido barbi-turico

Info

Publication number
ES8601152A1
ES8601152A1 ES540037A ES540037A ES8601152A1 ES 8601152 A1 ES8601152 A1 ES 8601152A1 ES 540037 A ES540037 A ES 540037A ES 540037 A ES540037 A ES 540037A ES 8601152 A1 ES8601152 A1 ES 8601152A1
Authority
ES
Spain
Prior art keywords
image
acid derivatives
barbituric acid
zooparasitic
helminths
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES540037A
Other languages
English (en)
Other versions
ES540037A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES540037A0 publication Critical patent/ES540037A0/es
Publication of ES8601152A1 publication Critical patent/ES8601152A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60—Three or more oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60—Three or more oxygen or sulfur atoms
    • C07D239/62—Barbituric acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Agronomy & Crop Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DEL ACIDO BARBITURICO DE SUS FORMAS TAUTOMERAS Y DE SUS SALES DE FORMULA (I) EN LA QUE X REPRESENTA OXIGENO O AZUFRE; Y R1 R2 R3 R4 Y R5 PUEDEN SER VARIOS TIPOS DE RADICALES. COMPRENDE LA REACCION DE CONDENSACION DE UN ACIDO BARBITURICO SUSTITUIDO DE FORMULA (II) CON UNA BENZOILAZIDA SUSTITUIDA DE FORMULA (III) EN LAS QUE TODOS LOS SIMBOLOS TIENEN LOS MISMOS SIGNIFICADOS QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO EN UN DISOLVENTE ORGANICO INERTE EN PRESENCIA DE UNA BASE A UNA TEMPERATURA COMPRENDIDA ENTRE 0JC Y 200JC. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS PARA EL TRATAMIENTO DE LOS HELMINTOS.
ES540037A 1983-08-19 1985-02-01 Procedimiento para la obtencion de derivados de acido barbi-turico Expired ES8601152A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH453583 1983-08-19
CH352684 1984-07-20

Publications (2)

Publication Number Publication Date
ES540037A0 ES540037A0 (es) 1985-11-01
ES8601152A1 true ES8601152A1 (es) 1985-11-01

Family

ID=25693240

Family Applications (3)

Application Number Title Priority Date Filing Date
ES535293A Expired ES8506290A1 (es) 1983-08-19 1984-08-20 Procedimiento para la obtencion de derivados de acido barbiturico
ES540040A Granted ES540040A0 (es) 1983-08-19 1985-02-01 Procedimiento para la obtencion de derivados de acido barbi-turico
ES540037A Expired ES8601152A1 (es) 1983-08-19 1985-02-01 Procedimiento para la obtencion de derivados de acido barbi-turico

Family Applications Before (2)

Application Number Title Priority Date Filing Date
ES535293A Expired ES8506290A1 (es) 1983-08-19 1984-08-20 Procedimiento para la obtencion de derivados de acido barbiturico
ES540040A Granted ES540040A0 (es) 1983-08-19 1985-02-01 Procedimiento para la obtencion de derivados de acido barbi-turico

Country Status (18)

Country Link
US (1) US4748178A (es)
EP (1) EP0135155B1 (es)
KR (1) KR850001907A (es)
AU (1) AU583796B2 (es)
CA (1) CA1264745A (es)
DD (1) DD222876A5 (es)
DE (1) DE3483294D1 (es)
DK (1) DK396384A (es)
EG (1) EG17262A (es)
ES (3) ES8506290A1 (es)
GB (1) GB2145087B (es)
HU (1) HU192991B (es)
IL (1) IL72716A (es)
MX (1) MX160630A (es)
MY (1) MY101864A (es)
NZ (1) NZ209267A (es)
PH (1) PH23080A (es)
ZW (1) ZW13584A1 (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2145087B (en) * 1983-08-19 1987-02-04 Ciba Geigy Ag Barbituric acid derivatives
CH657015A5 (de) * 1984-06-27 1986-08-15 Ciba Geigy Ag Motten- und kaeferschutzmittel.
US4753940A (en) * 1985-02-15 1988-06-28 Ciba-Geigy Corporation Barbituric acid derivatives
GB2171099B (en) * 1985-02-15 1988-10-19 Ciba Geigy Ag 5-(azolyloxphenylcarbamoyl)barbituric acid derivatives as anthelmintics
GB8531815D0 (en) * 1985-12-24 1986-02-05 Wellcome Found Insecticidal compounds
EP0430885A3 (en) * 1989-12-01 1991-11-06 Ciba-Geigy Ag Anthelmintical compounds
NL9001075A (es) * 1990-05-04 1991-12-02 Duphar Int Res
AUPO190596A0 (en) 1996-08-26 1996-09-19 Alchemia Pty Ltd Oligosaccharide synthesis
AUPO937597A0 (en) * 1997-09-24 1997-10-16 Alchemia Pty Ltd Protecting and linking groups for organic synthesis
KR101272098B1 (ko) * 2005-02-08 2013-06-07 가부시키가이샤 한도오따이 에네루기 켄큐쇼 발광소자, 발광장치 및 전자기기
AR125350A1 (es) * 2021-04-16 2023-07-12 Orion Corp Inhibidores tead

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2405733C2 (de) * 1974-02-07 1984-12-13 Bayer Ag, 5090 Leverkusen Amidocarbonylthiobarbitursäurederivate und deren Salze, Verfahren zu ihrer Herstellung sowie ihre Verwendung zur Bekämpfung von Insekten, Milben und Pilzen
PL103086B1 (pl) * 1976-05-06 1979-05-31 Ciba Geigy Ag Srodek owadobojczy
DE2832698A1 (de) * 1978-07-26 1980-02-07 Bayer Ag Substituierte 5-phenylcarbamoyl- barbitursaeuren, verfahren zu ihrer herstellung und ihre verwendung als insektizide
US4283444A (en) * 1978-09-12 1981-08-11 Ciba-Geigy Corporation Method of protecting keratinous material from attack by insects that feed on keratin by treatment with 5-phenylcarbamoylbarbituric acid compounds
GB2126582B (en) * 1982-08-26 1986-03-05 Ciba Geigy Ag Phenyl carbamoyl barbituric acid anthelmintics
CH658770A5 (de) * 1982-08-26 1986-12-15 Ciba Geigy Ag Motten- und kaeferschutzmittel.
GB2145087B (en) * 1983-08-19 1987-02-04 Ciba Geigy Ag Barbituric acid derivatives
IL73840A (en) * 1983-12-19 1988-11-15 Uniroyal Chem Co Inc 2-thio-5-(thio)carbamoyl barbituric acid derivatives,their preparation and pharmaceutical compositions containing them
CH657015A5 (de) * 1984-06-27 1986-08-15 Ciba Geigy Ag Motten- und kaeferschutzmittel.
EP0167491A3 (de) * 1984-07-06 1986-12-30 Ciba-Geigy Ag Thiobarbitursäurederivate
GB2171099B (en) * 1985-02-15 1988-10-19 Ciba Geigy Ag 5-(azolyloxphenylcarbamoyl)barbituric acid derivatives as anthelmintics

Also Published As

Publication number Publication date
DD222876A5 (de) 1985-05-29
KR850001907A (ko) 1985-04-10
ES8601153A1 (es) 1985-11-01
IL72716A0 (en) 1984-11-30
CA1264745A (en) 1990-01-23
MX160630A (es) 1990-03-29
US4748178A (en) 1988-05-31
ES535293A0 (es) 1985-07-16
EP0135155A3 (en) 1986-01-02
ES540037A0 (es) 1985-11-01
GB8420712D0 (en) 1984-09-19
EP0135155B1 (de) 1990-09-26
HU192991B (en) 1987-08-28
GB2145087A (en) 1985-03-20
PH23080A (en) 1989-04-10
DK396384D0 (da) 1984-08-17
AU3204084A (en) 1985-02-21
MY101864A (en) 1992-01-31
EP0135155A2 (de) 1985-03-27
EG17262A (en) 1991-08-30
ZW13584A1 (en) 1985-03-06
IL72716A (en) 1987-10-20
NZ209267A (en) 1988-01-08
GB2145087B (en) 1987-02-04
DK396384A (da) 1985-02-20
ES8506290A1 (es) 1985-07-16
HUT35653A (en) 1985-07-29
ES540040A0 (es) 1985-11-01
DE3483294D1 (de) 1990-10-31
AU583796B2 (en) 1989-05-11

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