ES8604501A2 - Procedimiento de obtencion de sulfonamidinas - Google Patents
Procedimiento de obtencion de sulfonamidinasInfo
- Publication number
- ES8604501A2 ES8604501A2 ES540192A ES540192A ES8604501A2 ES 8604501 A2 ES8604501 A2 ES 8604501A2 ES 540192 A ES540192 A ES 540192A ES 540192 A ES540192 A ES 540192A ES 8604501 A2 ES8604501 A2 ES 8604501A2
- Authority
- ES
- Spain
- Prior art keywords
- formula
- obtaining
- alkyl
- sulphonamidines
- thio
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- -1 2-[[[2-[(aminoiminomethyl)amino]-4- thiazolyl]methyl]thio]ethyl Chemical group 0.000 abstract 1
- 102000000543 Histamine Receptors Human genes 0.000 abstract 1
- 108010002059 Histamine Receptors Proteins 0.000 abstract 1
- 230000009858 acid secretion Effects 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- 125000004656 alkyl sulfonylamino group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 230000008485 antagonism Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 1
- CEIPQQODRKXDSB-UHFFFAOYSA-N ethyl 3-(6-hydroxynaphthalen-2-yl)-1H-indazole-5-carboximidate dihydrochloride Chemical compound Cl.Cl.C1=C(O)C=CC2=CC(C3=NNC4=CC=C(C=C43)C(=N)OCC)=CC=C21 CEIPQQODRKXDSB-UHFFFAOYSA-N 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- FDDDEECHVMSUSB-UHFFFAOYSA-N sulfanilamide Chemical compound NC1=CC=C(S(N)(=O)=O)C=C1 FDDDEECHVMSUSB-UHFFFAOYSA-N 0.000 abstract 1
- 229940124530 sulfonamide Drugs 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE SULFONAMIDINAS Y DE SUS SALES FISIOLOGICAMENTE COMPATIBLES, DE FORMULA (I), EN LA QUE R REPRESENTA UN RADICAL 2-Y2-(AMINO-IMINOMETIL)AMINO-4-TIAZOLILMETILTIOZETIL Y R1 PUEDE SER UNO DE VARIOS TIPOS DE RADICALES (CERTIFICADO DE ADICION DE LA PATENTE NUM. 532.242). CONSISTE EN LA REACCION DE UNA AMINA DE FORMULA R-NH2 CON UN EXCESO DE ORTOFORMIATO DE FORMULA H-C(OR2)3, EN LAS QUE R2 PUEDE SER VARIOS TIPOS DE RADICALES Y R ES EL MISMO QUE EN LA FORMULA (I), A UNA TEMPERATURA COMPRENDIDA ENTRE 85JC Y LA DE EBULLICION DE LA MEZCLA; SEGUIDA DE LA REACCION DEL COMPUESTO FORMADO CON UNA SULFONAMIDA DE FORMULA H2N-SO2-R1, EN UN ALCANOL C1-4, A LA TEMPERATURA AMBIENTE. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS COMO INHIBIDORES DE LA SECRECION GASTRICA.
Priority Applications (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES540192A ES540192A0 (es) | 1985-01-25 | 1985-01-25 | Procedimiento de obtencion de sulfonamidinas |
| CA000477755A CA1269382A (en) | 1984-04-18 | 1985-03-28 | Anti-ulceric sulfonamidines |
| PH32140A PH21779A (en) | 1984-04-18 | 1985-04-15 | Sulfonomidines and pharmaceutical compositions containing the same |
| EP85104577A EP0159012B1 (en) | 1984-04-18 | 1985-04-16 | Sulfonamidines, a process for preparing them and pharmaceutical compositions containing them |
| DE8585104577T DE3568041D1 (en) | 1984-04-18 | 1985-04-16 | Sulfonamidines, a process for preparing them and pharmaceutical compositions containing them |
| US06/724,784 US4728655A (en) | 1984-04-18 | 1985-04-18 | Sulfonamidines, process for the production thereof and pharmaceutical compositions containing the same |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES540192A ES540192A0 (es) | 1985-01-25 | 1985-01-25 | Procedimiento de obtencion de sulfonamidinas |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8604501A2 true ES8604501A2 (es) | 1986-02-01 |
| ES540192A0 ES540192A0 (es) | 1986-02-01 |
Family
ID=8488664
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES540192A Granted ES540192A0 (es) | 1984-04-18 | 1985-01-25 | Procedimiento de obtencion de sulfonamidinas |
Country Status (1)
| Country | Link |
|---|---|
| ES (1) | ES540192A0 (es) |
-
1985
- 1985-01-25 ES ES540192A patent/ES540192A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| ES540192A0 (es) | 1986-02-01 |
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