ES8604530A1 - Procedimiento para la preparacion de derivados de n-(2-ni- trofenil)-2-aminopirimidina - Google Patents

Procedimiento para la preparacion de derivados de n-(2-ni- trofenil)-2-aminopirimidina

Info

Publication number
ES8604530A1
ES8604530A1 ES544463A ES544463A ES8604530A1 ES 8604530 A1 ES8604530 A1 ES 8604530A1 ES 544463 A ES544463 A ES 544463A ES 544463 A ES544463 A ES 544463A ES 8604530 A1 ES8604530 A1 ES 8604530A1
Authority
ES
Spain
Prior art keywords
substd
halogen
alkoxy
opt
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES544463A
Other languages
English (en)
Other versions
ES544463A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES544463A0 publication Critical patent/ES544463A0/es
Publication of ES8604530A1 publication Critical patent/ES8604530A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Health & Medical Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Dental Preparations (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE N-(2-NITROFENIL)-2-AMINOPIRIMIDINA, DE FORMULA (I), EN LA QUE R1, R2, R3, R4, R5, R6 Y R7 PUEDEN SER VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE UN COMPUESTO DE FORMULA (II) CON UN DERIVADO DE PIRIMIDINA DE FORMULA (III), EN PRESENCIA DE UNA BASE; SEGUIDA DEL TRATAMIENTO DEL COMPUESTO FORMADO CON UN DERIVADO REACTIVO DEL ACIDO CARBOXILICO DE FORMULA R4COOH, EN LAS QUE Z E Y REPRESENTAN, UNO DE ELLOS HALOGENO Y EL OTRO GRUPO NH2, Y TODOS LOS DEMAS SIMBOLOS TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). ESTOS COMPUESTOS TIENEN APLICACIONES EN AGRICULTURA PARA COMBATIR LOS HONGOS Y LAS BACTERIAS QUE PERJUDICAN A LAS PLANTAS.
ES544463A 1984-06-25 1985-06-22 Procedimiento para la preparacion de derivados de n-(2-ni- trofenil)-2-aminopirimidina Expired ES8604530A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH305584 1984-06-25

Publications (2)

Publication Number Publication Date
ES544463A0 ES544463A0 (es) 1986-02-01
ES8604530A1 true ES8604530A1 (es) 1986-02-01

Family

ID=4247600

Family Applications (1)

Application Number Title Priority Date Filing Date
ES544463A Expired ES8604530A1 (es) 1984-06-25 1985-06-22 Procedimiento para la preparacion de derivados de n-(2-ni- trofenil)-2-aminopirimidina

Country Status (14)

Country Link
US (1) US4694009A (es)
EP (1) EP0172786B1 (es)
JP (1) JPS6115877A (es)
AT (1) ATE60591T1 (es)
AU (1) AU585867B2 (es)
BR (1) BR8503024A (es)
DE (1) DE3581570D1 (es)
DK (1) DK285285A (es)
ES (1) ES8604530A1 (es)
GR (1) GR851534B (es)
IL (1) IL75612A (es)
PH (1) PH22765A (es)
PT (1) PT80683B (es)
ZA (1) ZA854738B (es)

Families Citing this family (35)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4659363A (en) * 1983-07-25 1987-04-21 Ciba-Geigy Corporation N-(2-nitrophenyl)-2-aminopyrimidine derivatives, the preparation and use thereof
PH21918A (en) * 1983-07-25 1988-04-08 Ciba Geigy Ag N-(2-nitrophenyl)-5-aminopyrimidine derivatives,the preparation and use thereof
GR80171B (en) * 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
DE3614060A1 (de) * 1986-04-23 1987-10-29 Schering Ag Pyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
EP0264348B1 (de) * 1986-10-13 1993-12-15 Ciba-Geigy Ag Harnstoffe
JPH0784445B2 (ja) * 1986-12-03 1995-09-13 クミアイ化学工業株式会社 ピリミジン誘導体および農園芸用殺菌剤
ES2058332T3 (es) * 1987-06-11 1994-11-01 Ciba Geigy Ag Microbicidas.
ES2054867T3 (es) * 1987-09-28 1994-08-16 Ciba Geigy Ag Plaguicidas y pesticidas.
CN1034255C (zh) * 1987-09-28 1997-03-19 希巴-盖吉股份公司 控制或预防有害昆虫或微生物侵害的组合物
US5153200A (en) * 1987-09-28 1992-10-06 Ciba-Geigy Corporation Pesticides
US4966622A (en) * 1988-04-12 1990-10-30 Ciba-Geigy Corporation N-phenyl-N-pyrimidin-2-ylureas
US4973690A (en) * 1988-04-12 1990-11-27 Ciba-Geigy Corporation Novel ureas
DE58905007D1 (de) * 1988-04-12 1993-09-02 Ciba Geigy Ag Harnstoffe.
US4897396A (en) * 1988-06-03 1990-01-30 Ciba-Geigy Corporation 2-phenylamino pyrimidine derivatives and their uses as microbicides
US5521184A (en) * 1992-04-03 1996-05-28 Ciba-Geigy Corporation Pyrimidine derivatives and processes for the preparation thereof
GB9304919D0 (en) * 1993-03-10 1993-04-28 Celltech Ltd Chemical compounds
US5786354A (en) * 1994-06-21 1998-07-28 Celltech Therapeutics, Limited Tri-substituted phenyl derivatives and processes for their preparation
US6245774B1 (en) 1994-06-21 2001-06-12 Celltech Therapeutics Limited Tri-substituted phenyl or pyridine derivatives
GB9412571D0 (en) 1994-06-22 1994-08-10 Celltech Ltd Chemical compounds
GB9412573D0 (en) 1994-06-22 1994-08-10 Celltech Ltd Chemical compounds
GB9523675D0 (en) 1995-11-20 1996-01-24 Celltech Therapeutics Ltd Chemical compounds
GB9622363D0 (en) 1996-10-28 1997-01-08 Celltech Therapeutics Ltd Chemical compounds
AU5330698A (en) * 1996-12-23 1998-07-17 Celltech Therapeutics Limited Fused polycyclic 2-aminopyrimidine derivatives, their preparation and their use as protein tyrosine kinase inhibitors
GB9705361D0 (en) * 1997-03-14 1997-04-30 Celltech Therapeutics Ltd Chemical compounds
GB9713087D0 (en) * 1997-06-20 1997-08-27 Celltech Therapeutics Ltd Chemical compounds
EP1085807B1 (de) * 1998-06-10 2003-05-07 Basf Aktiengesellschaft Verwendung von 2-(n-phenylamino)pyrimidinen als fungizide sowie neue 2-(n-phenylamino)pyrimidine
JP3635238B2 (ja) * 1998-11-10 2005-04-06 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Ｈｉｖの複製を阻害するピリミジン類
SK286264B6 (sk) 1998-11-17 2008-06-06 Kumiai Chemical Industry Co., Ltd. Derivát pyrimidinylbenzimidazolu alebo triazinylbenzimidazolu, medziprodukty na jeho prípravu a poľnohospodársky/záhradnícky fungicíd s jeho obsahom
JP4535350B2 (ja) * 1998-11-17 2010-09-01 クミアイ化学工業株式会社 ピリミジニルベンズイミダゾール誘導体及び農園芸用殺菌剤
GB9914258D0 (en) * 1999-06-18 1999-08-18 Celltech Therapeutics Ltd Chemical compounds
DE60025837T2 (de) 1999-09-24 2006-11-02 Janssen Pharmaceutica N.V. Antivirale feste dispersionen
GB9924862D0 (en) 1999-10-20 1999-12-22 Celltech Therapeutics Ltd Chemical compounds
AU2002312933B2 (en) * 2001-05-29 2007-12-06 Schering Ag CDK inhibiting pyrimidines, production thereof and their use as medicaments
AR038368A1 (es) * 2002-02-01 2005-01-12 Novartis Ag Compuestos n-pirimidin-2-il-aminas sustituidas como inhibidores de ige, una composicion farmaceutica y el uso de dichos compuestos para la preparacion de un medicamento
EP1871743A4 (en) * 2005-04-11 2009-12-30 Univ Murdoch PEST CONTROL COMPOUNDS

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1388825A (en) * 1971-03-19 1975-03-26 Ici Ltd Substituted amino pyrimidine compounds and pesticidal compo sitions thereof
GB1394816A (en) * 1971-03-19 1975-05-21 Ici Ltd Substituted amino diazinyl compounds and pesticidal compositions thereof
AU5319479A (en) * 1978-12-22 1980-06-26 Ici Australia Limited Pyrimidinyl amino phenoxy carboxylate derivatives
JPS5665804A (en) * 1979-11-01 1981-06-03 Ishihara Sangyo Kaisha Ltd Control agent against injurious organism
DD151404A1 (de) * 1980-06-13 1981-10-21 Friedrich Franke Fungizide mittel
DK130584A (da) * 1983-04-08 1984-10-09 Ciba Geigy Ag N-(2-nitrophenyl)-4-amino-pyrimidin-derivater samt deres fremstilling og anvendelse som mikrobicider
US4659363A (en) * 1983-07-25 1987-04-21 Ciba-Geigy Corporation N-(2-nitrophenyl)-2-aminopyrimidine derivatives, the preparation and use thereof
GR80171B (en) * 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
CH661827A5 (de) * 1983-09-05 1987-08-14 Reichle & De Massari Fa Gestell fuer den schwachstrom-anlagebau, insbesondere fuer verteiler-anlagen.

Also Published As

Publication number Publication date
ATE60591T1 (de) 1991-02-15
IL75612A0 (en) 1985-10-31
PH22765A (en) 1988-12-12
PT80683A (de) 1985-07-01
EP0172786B1 (de) 1991-01-30
DK285285D0 (da) 1985-06-24
ES544463A0 (es) 1986-02-01
DE3581570D1 (de) 1991-03-07
AU585867B2 (en) 1989-06-29
IL75612A (en) 1989-07-31
AU4398885A (en) 1986-01-02
EP0172786A2 (de) 1986-02-26
BR8503024A (pt) 1986-03-11
JPS6115877A (ja) 1986-01-23
GR851534B (es) 1985-11-25
DK285285A (da) 1985-12-26
PT80683B (de) 1987-05-08
EP0172786A3 (en) 1986-10-29
ZA854738B (en) 1986-02-26
US4694009A (en) 1987-09-15

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Legal Events

Date Code Title Description
MM4A Patent lapsed

Effective date: 19960401