ES8702923A1 - Un procedimiento para la preparacion de derivados de octa- hidro-6-azaindol-dipeptidos - Google Patents

Un procedimiento para la preparacion de derivados de octa- hidro-6-azaindol-dipeptidos

Info

Publication number
ES8702923A1
ES8702923A1 ES550149A ES550149A ES8702923A1 ES 8702923 A1 ES8702923 A1 ES 8702923A1 ES 550149 A ES550149 A ES 550149A ES 550149 A ES550149 A ES 550149A ES 8702923 A1 ES8702923 A1 ES 8702923A1
Authority
ES
Spain
Prior art keywords
derivatives
azaindol
procedure
preparation
dipeptidos
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES550149A
Other languages
English (en)
Spanish (es)
Other versions
ES550149A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB848432532A external-priority patent/GB8432532D0/en
Priority claimed from GB858514634A external-priority patent/GB8514634D0/en
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Publication of ES550149A0 publication Critical patent/ES550149A0/es
Publication of ES8702923A1 publication Critical patent/ES8702923A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
ES550149A 1984-12-21 1985-12-19 Un procedimiento para la preparacion de derivados de octa- hidro-6-azaindol-dipeptidos Expired ES8702923A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB848432532A GB8432532D0 (en) 1984-12-21 1984-12-21 Therapeutic agents
GB858514634A GB8514634D0 (en) 1985-06-10 1985-06-10 Therapeutic agents

Publications (2)

Publication Number Publication Date
ES550149A0 ES550149A0 (es) 1987-01-16
ES8702923A1 true ES8702923A1 (es) 1987-01-16

Family

ID=26288610

Family Applications (1)

Application Number Title Priority Date Filing Date
ES550149A Expired ES8702923A1 (es) 1984-12-21 1985-12-19 Un procedimiento para la preparacion de derivados de octa- hidro-6-azaindol-dipeptidos

Country Status (16)

Country Link
US (1) US4711882A (2)
EP (1) EP0186431B1 (2)
CN (1) CN85109243A (2)
AU (1) AU558427B2 (2)
CS (1) CS250699B2 (2)
DE (1) DE3561551D1 (2)
DK (1) DK595385A (2)
ES (1) ES8702923A1 (2)
FI (1) FI855112A7 (2)
GR (1) GR853117B (2)
HU (1) HUT40125A (2)
NO (1) NO855214L (2)
NZ (1) NZ214649A (2)
PL (1) PL256935A1 (2)
PT (1) PT81722B (2)
YU (1) YU199485A (2)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL58849A (en) * 1978-12-11 1983-03-31 Merck & Co Inc Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them
FR2487829A2 (fr) * 1979-12-07 1982-02-05 Science Union & Cie Nouveaux imino acides substitues, leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme
ATE20469T1 (de) * 1980-10-23 1986-07-15 Schering Corp Carboxyalkyl-dipeptide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel.
DE3302125A1 (de) * 1983-01-22 1984-07-26 Boehringer Ingelheim KG, 6507 Ingelheim Aminosaeure-derivate, verfahren zu ihrer herstellung und verwendung

Also Published As

Publication number Publication date
FI855112A0 (fi) 1985-12-20
DE3561551D1 (de) 1988-03-10
CS250699B2 (en) 1987-05-14
FI855112A7 (fi) 1986-06-22
GR853117B (2) 1986-04-22
PT81722B (en) 1987-10-19
AU558427B2 (en) 1987-01-29
DK595385A (da) 1986-06-22
NO855214L (no) 1986-06-23
ES550149A0 (es) 1987-01-16
HUT40125A (en) 1986-11-28
YU199485A (en) 1988-04-30
DK595385D0 (da) 1985-12-20
PT81722A (en) 1986-01-01
CN85109243A (zh) 1986-09-17
PL256935A1 (en) 1987-02-23
NZ214649A (en) 1988-02-12
AU5151285A (en) 1986-06-26
EP0186431B1 (en) 1988-02-03
US4711882A (en) 1987-12-08
EP0186431A1 (en) 1986-07-02

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ES8702923A1 (es) Un procedimiento para la preparacion de derivados de octa- hidro-6-azaindol-dipeptidos