FR2235687A2 - 1-Trimethoxy phenyl-3-carboxamido indoles - anti-inflammatories, sedatives, vasodilators, hypotensives, analgesics, anticholinergics, anti-ulcer agents etc. - Google Patents

1-Trimethoxy phenyl-3-carboxamido indoles - anti-inflammatories, sedatives, vasodilators, hypotensives, analgesics, anticholinergics, anti-ulcer agents etc.

Info

Publication number
FR2235687A2
FR2235687A2 FR7324387A FR7324387A FR2235687A2 FR 2235687 A2 FR2235687 A2 FR 2235687A2 FR 7324387 A FR7324387 A FR 7324387A FR 7324387 A FR7324387 A FR 7324387A FR 2235687 A2 FR2235687 A2 FR 2235687A2
Authority
FR
France
Prior art keywords
carboxamido
indoles
hypotensives
anticholinergics
inflammatories
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7324387A
Other languages
French (fr)
Other versions
FR2235687B2 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Delalande SA filed Critical Delalande SA
Priority to FR7324387A priority Critical patent/FR2235687A2/en
Publication of FR2235687A2 publication Critical patent/FR2235687A2/en
Application granted granted Critical
Publication of FR2235687B2 publication Critical patent/FR2235687B2/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Carboxamido indoles of formula (I): (where R is straight or branched 1-4C alkylamino, pyrrolidino, piperidino, morpholino, hexamethyleneimino or piperazino substd. in the 4-posn. by a pyrrolidino carbonylmethyl, isopropylamino carbonylmethyl, morpholino carbonylmethyl or ethoxycarbonylmethyl gp.). have antiulcerous, antibroncho-constrictive, anticholinergic, analgesic, anti-inflammatory, sedative, diuretic, vasodilative and hypotensive activity.
FR7324387A 1973-07-03 1973-07-03 1-Trimethoxy phenyl-3-carboxamido indoles - anti-inflammatories, sedatives, vasodilators, hypotensives, analgesics, anticholinergics, anti-ulcer agents etc. Granted FR2235687A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7324387A FR2235687A2 (en) 1973-07-03 1973-07-03 1-Trimethoxy phenyl-3-carboxamido indoles - anti-inflammatories, sedatives, vasodilators, hypotensives, analgesics, anticholinergics, anti-ulcer agents etc.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7324387A FR2235687A2 (en) 1973-07-03 1973-07-03 1-Trimethoxy phenyl-3-carboxamido indoles - anti-inflammatories, sedatives, vasodilators, hypotensives, analgesics, anticholinergics, anti-ulcer agents etc.

Publications (2)

Publication Number Publication Date
FR2235687A2 true FR2235687A2 (en) 1975-01-31
FR2235687B2 FR2235687B2 (en) 1977-08-19

Family

ID=9121983

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7324387A Granted FR2235687A2 (en) 1973-07-03 1973-07-03 1-Trimethoxy phenyl-3-carboxamido indoles - anti-inflammatories, sedatives, vasodilators, hypotensives, analgesics, anticholinergics, anti-ulcer agents etc.

Country Status (1)

Country Link
FR (1) FR2235687A2 (en)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3466287A (en) * 1966-10-07 1969-09-09 Sterling Drug Inc 1-((3-indolyl)-lower-alkyl)-4-substituted piperazines
GB1273563A (en) * 1968-07-24 1972-05-10 Wyeth John & Brother Ltd Indoles

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3466287A (en) * 1966-10-07 1969-09-09 Sterling Drug Inc 1-((3-indolyl)-lower-alkyl)-4-substituted piperazines
GB1273563A (en) * 1968-07-24 1972-05-10 Wyeth John & Brother Ltd Indoles

Also Published As

Publication number Publication date
FR2235687B2 (en) 1977-08-19

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