FR2361914A1 - Nouvelles formulations de medicaments a danger d'emploi abusif reduit - Google Patents

Nouvelles formulations de medicaments a danger d'emploi abusif reduit

Info

Publication number
FR2361914A1
FR2361914A1 FR7621071A FR7621071A FR2361914A1 FR 2361914 A1 FR2361914 A1 FR 2361914A1 FR 7621071 A FR7621071 A FR 7621071A FR 7621071 A FR7621071 A FR 7621071A FR 2361914 A1 FR2361914 A1 FR 2361914A1
Authority
FR
France
Prior art keywords
drugs
new formulations
reduced danger
abusive use
danger
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7621071A
Other languages
English (en)
Other versions
FR2361914B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of FR2361914A1 publication Critical patent/FR2361914A1/fr
Application granted granted Critical
Publication of FR2361914B1 publication Critical patent/FR2361914B1/fr
Granted legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/60—Salicylic acid; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

L'invention concerne un procédé pour réduire le danger d'emploi abusif de préparations pharmaceutiques à usage entéral renfermant des analgésiques d'activité moyenne à forte. Le procédé consiste à ajouter des substances gonflantes déterminées, notamment des dérivés méthylcellulosiques qui s'opposent à l'extraction des substances actives. Une solution injectable de la substance active ne peut plus être obtenue à partir de comprimés et de dragées conformes à l'invention.
FR7621071A 1975-07-09 1976-07-09 Nouvelles formulations de medicaments a danger d'emploi abusif reduit Granted FR2361914A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2530563A DE2530563C2 (de) 1975-07-09 1975-07-09 Analgetische Arzneimittel mit vermindertem Mißbrauchspotential

Publications (2)

Publication Number Publication Date
FR2361914A1 true FR2361914A1 (fr) 1978-03-17
FR2361914B1 FR2361914B1 (fr) 1978-12-15

Family

ID=5951020

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7621071A Granted FR2361914A1 (fr) 1975-07-09 1976-07-09 Nouvelles formulations de medicaments a danger d'emploi abusif reduit

Country Status (7)

Country Link
US (1) US4070494A (fr)
JP (1) JPS5210415A (fr)
BE (1) BE843865A (fr)
CA (1) CA1064397A (fr)
DE (1) DE2530563C2 (fr)
FR (1) FR2361914A1 (fr)
GB (1) GB1517480A (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011154414A1 (fr) 2010-06-07 2011-12-15 Ethypharm Microgranules et microcomprimes resistants au detournement

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BE663600A (fr) * 1964-05-09 1965-11-08
GB1171691A (en) * 1967-02-24 1969-11-26 Forest Laboratories Lond-Acting Oral Carrier

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011154414A1 (fr) 2010-06-07 2011-12-15 Ethypharm Microgranules et microcomprimes resistants au detournement

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FR2361914B1 (fr) 1978-12-15
DE2530563C2 (de) 1986-07-24
CA1064397A (fr) 1979-10-16
BE843865A (fr) 1977-01-07
US4070494A (en) 1978-01-24
JPS5210415A (en) 1977-01-26
GB1517480A (en) 1978-07-12
DE2530563A1 (de) 1977-01-27

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