GT200200093A - CRYSTALLINE FORMS OF AZITHROMYCIN - Google Patents
CRYSTALLINE FORMS OF AZITHROMYCINInfo
- Publication number
- GT200200093A GT200200093A GT200200093A GT200200093A GT200200093A GT 200200093 A GT200200093 A GT 200200093A GT 200200093 A GT200200093 A GT 200200093A GT 200200093 A GT200200093 A GT 200200093A GT 200200093 A GT200200093 A GT 200200093A
- Authority
- GT
- Guatemala
- Prior art keywords
- azithromycin
- forms
- crystalline forms
- document
- refers
- Prior art date
Links
- MQTOSJVFKKJCRP-BICOPXKESA-N azithromycin Chemical compound O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 MQTOSJVFKKJCRP-BICOPXKESA-N 0.000 title abstract 2
- 229960004099 azithromycin Drugs 0.000 title abstract 2
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000013078 crystal Substances 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
- 230000002458 infectious effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A FORMAS CRISTALINAS DE AZITROMICINA Y COMO SE USA EN ESTE DOCUMENTO, LA EXPRESION "FORMAS CRISTALINAS", A MENOS QUE SE INDIQUE OTRA COSA, SE REFIERE EN PARTICULAR A LAS FORMAS C,D,E,F,G,H,J,M,N,O,P,Q Y R SIENDO DICHAS FORMAS COMO SE DEFINEN EN EL DOCUMENTO. ESTOS COMPUESTOS POR SU NATURALEZA ANTIBIOTICA SON UTILES EN ESTADOS INFECCIOSOS.THE PRESENT INVENTION REFERS TO CRYSTALLINE FORMS OF AZITHROMYCIN AND AS USED IN THIS DOCUMENT, THE EXPRESSION "CRYSTAL FORMS", UNLESS OTHERWISE INDICATED, REFERS IN PARTICULAR TO FORMS C, D, E, F, G, H, J, M, N, O, P, QYR BEING SUCH FORMS AS DEFINED IN THE DOCUMENT. THESE COMPOUNDS FOR THEIR ANTIBIOTIC NATURE ARE USEFUL IN INFECTIOUS STATES.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29256501P | 2001-05-22 | 2001-05-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT200200093A true GT200200093A (en) | 2003-05-23 |
Family
ID=34115151
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT200200093A GT200200093A (en) | 2001-05-22 | 2002-05-21 | CRYSTALLINE FORMS OF AZITHROMYCIN |
Country Status (6)
| Country | Link |
|---|---|
| CN (1) | CN100354294C (en) |
| EC (1) | ECSP034861A (en) |
| GT (1) | GT200200093A (en) |
| PY (1) | PY0211797A (en) |
| UA (1) | UA74887C2 (en) |
| ZA (1) | ZA200308341B (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102911219A (en) * | 2011-08-03 | 2013-02-06 | 山东方明药业集团股份有限公司 | Method for directly crystallizing azithromycin in aqueous phase |
| CN105030704B (en) * | 2015-06-29 | 2018-09-07 | 石药集团欧意药业有限公司 | Azithromycin and preparation method thereof |
| CN105061528B (en) * | 2015-08-05 | 2017-10-17 | 浙江维康药业股份有限公司 | A kind of azithromycin compound and the Azithromycin soft capsules containing the compound |
| CN106188177A (en) * | 2016-07-12 | 2016-12-07 | 浙江亚太药业股份有限公司 | The preparation method of a kind of azithromycin compound and pharmaceutical preparation thereof |
| CN111170959A (en) * | 2019-12-30 | 2020-05-19 | 南开大学 | Crystal form of macrolide compound, preparation method and application thereof |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1093370A (en) * | 1993-12-10 | 1994-10-12 | 北京市集才药物研究所 | A kind of new azido erythromycin crystal and preparation method thereof |
-
2002
- 2002-01-05 UA UA20031110541A patent/UA74887C2/en unknown
- 2002-05-01 CN CNB028104935A patent/CN100354294C/en not_active Expired - Fee Related
- 2002-05-21 GT GT200200093A patent/GT200200093A/en unknown
- 2002-05-21 PY PY200200211797A patent/PY0211797A/en unknown
-
2003
- 2003-10-27 ZA ZA200308341A patent/ZA200308341B/en unknown
- 2003-11-21 EC ECSP034861 patent/ECSP034861A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| UA74887C2 (en) | 2006-02-15 |
| ECSP034861A (en) | 2004-01-28 |
| PY0211797A (en) | 2004-07-01 |
| CN1780847A (en) | 2006-05-31 |
| ZA200308341B (en) | 2004-10-27 |
| CN100354294C (en) | 2007-12-12 |
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