HK7497A - 6-arylpyrimidines and herbicidal use thereof - Google Patents

6-arylpyrimidines and herbicidal use thereof

Info

Publication number
HK7497A
HK7497A HK7497A HK7497A HK7497A HK 7497 A HK7497 A HK 7497A HK 7497 A HK7497 A HK 7497A HK 7497 A HK7497 A HK 7497A HK 7497 A HK7497 A HK 7497A
Authority
HK
Hong Kong
Prior art keywords
alkyl
phenyl
alkenyl
halo
alkynyl
Prior art date
Application number
HK7497A
Other languages
German (de)
English (en)
Inventor
Michael Tice Colin
Original Assignee
Rohm And Haas Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rohm And Haas Company filed Critical Rohm And Haas Company
Publication of HK7497A publication Critical patent/HK7497A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/74—Quinazolines; Hydrogenated quinazolines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to ring carbon atoms of the hetero ring
    • C07D239/76—N-oxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Claims (11)

  1. Composé de formule : dans laquelle :
    (a) R2 est de l'hydrogène ou un groupe alkyle en (C1-C6) à chaîne droite, alkyle en (C3-C8) à chaîne ramifiée, alcényle en (C2-C6), alcynyle en (C2-C6), haloalkyle en (C1-C6), polyhaloalkyle en- (C1-C6), haloalcényle en (C2-C6), polyhaloalcényle en (C2-C6), haloalcynyle en (C2-C6), polyhaloalcynyle en (C2-C6), alcoxy en (C1-C4) alkyle en (C1-C4), alkyle en (C1-C6) thio, alcoxy en (C1-C6), alcoxy en (C1-C3) carbonyle, alcoxy en (C1-C3) carbonylalkyle en (C1-C3), arylalkyle en (C1-C4), cycloalkyle en (C3-C7), alkyl en (C1-C3) amino, dialkyl en (C1-C3) amino, dialkyl en (C1-C3) aminocarbonyle, halo ou cyano; et
    (b) R3 est un groupe alkyle en (C1-C4), alcényle en (C3-C6), alcynyle en (C3-C6), halo- ou polyhaloalkyle en (C1-C6);    ou facultativement R2 et R3 sont fusionnés en un radical de liaison à deux à cinq chaînons, chacun desdits éléments de liaison étant indépendamment du carbone, de l'oxygène ou du soufre;
    (c) R5 est un groupe alcynyle en (C2-C6) qui est facultativement substitué par jusqu'à cinq atomes d'halogène; et
    (d) R6 est un groupe phényle qui est facultativement substitué par jusqu'à trois substituants indépendamment choisis parmi les groupes bromo; chloro; fluoro; alkyle en (C1-C12), cycloalkyle en (C3-C8), alcényle en (C2-C12), cycloalcényle en (C3-C8), alcynyle en (C2-C12), haloalkyle en (C1-C12), polyhaloalkyle en (C1-C12), haloalcényle en (C2-C12), polyhaloalcényle en (C2-C12), haloalcynyle en (C2-C6), polyhaloalcynyle en (C2-C6); alcoxy en (C1-C12), alkyle en (C1-C12) thio, alkyle en (C1-C12) sulfonyle; alkyle en (C1-C12) sulfinyle; phényle; phénylalkyle en (C1-C12); phénylalcényle en (C2-C12); phénylalcynyle en (C2-C12); cyano; haloalcoxy en (C1-C6), alcoxy en (C1-C6) carbonyle ou nitro, et
    (e) X est de l'oxygène ou du soufre.
  2. Composé selon la revendication 1, dans lequel R2 est un groupe méthyle, éthyle, n-propyle, n-butyle, n-hexyle, i-propyle, i-butyle, t-butyle, méthoxy, éthoxy, éthoxycarbonyle, but-2-ynyle, but-3-ynyle, prop-2-ynyle, fluoro, bromo, chloro, trifluorométhyle, pentafluoroéthyle, méthylthio, méthoxyméthyle, benzyle, cyclopropyle, cyclobutyle, diméthylamino, diméthylaminocarbonyle ou allyle.
  3. Composé selon la revendication 1 ou 2, dans lequel R3 est le groupe méthyle, éthyle, prop-2-ynyle, allyle ou trifluorométhyle.
  4. Composé selon la revendication 1, dans lequel :
    (a) ladite liaison R2-R3 est choisie parmi -(CH2)2-5- et -SCH2CH2-;
    (b) R5 est un groupe propargyl; et
    (c) R6 est un groupe phényle.
  5. Composé selon l'une quelconque des revendications précédentes, dans lequel le groupe R5 est un groupe prop-2-ynyle ou but-2-ynyle.
  6. Composé selon l'une quelconque des revendications précédentes, dans lequel R6 est un groupe phényle, 2-fluorophényle, 3-fluorophényle, 4-fluorophényle, 3-chlorophényle ou 3,5-difluorophényle.
  7. Composé selon l'une quelconque des revendications précédentes, dans lequel X est de l'oxygène.
  8. Composé selon l'une quelconque des revendications précédentes, qui est l'un des composés suivants :
    2,3-diméthyl-6-phényl-5-propargyl-4(3 H)-pyrimidinone;
    3-méthyl-6-phényl-5-propargyl-2-propyl-4(3H) pyrimidinone;
    2,3-diéthyl-6-phényl-5-propargyl-4(3H)-pyrimidinone;
    3-éthyl-6-phényl-5-propargyl-2-trifluorométhyl-4(3H)-pyrimidinone; et
    3-éthyl-2-isopropyl-6-phényl-5-propargyl-4(3 H)-pyrimidinone.
  9. Composition comprenant une quantité herbicide efficace d'un composé selon l'une quelconque des revendications précédentes et un véhicule acceptable d'un point de vue agronomique.
  10. Procédé de contrôle d'une plante consistant à appliquer à ladite plante ou audit site ou audit milieu de croissance une quantité herbicide efficace d'un composé ou d'une composition tel(le) que défini(e) dans l'une quelconque des revendications précédentes.
  11. Utilisation d'un composé ou d'une composition tel(le) que défini(e) dans l'une quelconque des revendications 1 à 9, à titre d'herbicide.
HK7497A 1992-07-17 1997-01-16 6-arylpyrimidines and herbicidal use thereof HK7497A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/916,315 US5298481A (en) 1992-07-17 1992-07-17 6-arylpyrimidines and herbicidal use

Publications (1)

Publication Number Publication Date
HK7497A true HK7497A (en) 1997-01-24

Family

ID=25437051

Family Applications (1)

Application Number Title Priority Date Filing Date
HK7497A HK7497A (en) 1992-07-17 1997-01-16 6-arylpyrimidines and herbicidal use thereof

Country Status (19)

Country Link
US (2) US5298481A (fr)
EP (1) EP0579425B1 (fr)
JP (1) JPH06100544A (fr)
KR (1) KR940005589A (fr)
CN (1) CN1081439A (fr)
AT (1) ATE143951T1 (fr)
AU (1) AU672408B2 (fr)
BR (1) BR9302830A (fr)
CA (1) CA2099923A1 (fr)
DE (1) DE69305265T2 (fr)
DK (1) DK0579425T3 (fr)
ES (1) ES2092768T3 (fr)
HK (1) HK7497A (fr)
HU (1) HUT65123A (fr)
IL (1) IL106231A0 (fr)
MX (1) MX9304218A (fr)
NZ (1) NZ248089A (fr)
TW (1) TW239063B (fr)
ZA (1) ZA935032B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5270317A (en) * 1990-03-20 1993-12-14 Elf Sanofi N-substituted heterocyclic derivatives, their preparation and the pharmaceutical compositions in which they are present
JPH0687835A (ja) * 1992-07-17 1994-03-29 Rohm & Haas Co 除草性２−アリール−５，６−縮合環−ピリミジン
ATE144500T1 (de) * 1992-07-17 1996-11-15 Rohm & Haas 2-substituierte pyrimidine und ihre verwendung als herbizide
US5391541A (en) * 1993-08-11 1995-02-21 Fmc Corporation Herbicidal 3-(substituted-benzyl)-1-methyl-6-trifluoromethyluracils
WO1995011235A1 (fr) * 1993-10-20 1995-04-27 The Upjohn Company Pyrimidinones utilisees comme antiarthritiques et anti-inflammatoires
US6410729B1 (en) 1996-12-05 2002-06-25 Amgen Inc. Substituted pyrimidine compounds and methods of use
US6096753A (en) 1996-12-05 2000-08-01 Amgen Inc. Substituted pyrimidinone and pyridone compounds and methods of use
US20070129282A1 (en) * 1998-11-24 2007-06-07 Ahlem Clarence N Pharmaceutical treatments and compositions
KR100356738B1 (ko) * 2000-09-07 2002-10-18 주식회사 삼양제넥스 염기성 단백질로부터 엔도톡신을 제거하는 방법
US6513603B2 (en) * 2001-03-29 2003-02-04 Planet Air Turf Products, Llc Soil aeration tine
JP2008515902A (ja) * 2004-10-06 2008-05-15 エヌピーエス ファーマシューティカルズ インコーポレイテッド カルシウム拮抗化合物としての相補ピリミジノン化合物
US10441588B2 (en) 2012-05-02 2019-10-15 Curators Of The University Of Missouri Methods and compositions for treating bacterial infection
US9814719B2 (en) 2012-05-02 2017-11-14 Curators Of The University Of Missouri Methods and compositions for treating bacterial infection
US9504688B2 (en) 2012-05-02 2016-11-29 The Regents Of The University Of Michigan Methods and compositions for treating bacterial infection

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1003802A (en) * 1963-06-04 1965-09-08 Searle & Co Pyrimidinone derivatives
US3214430A (en) * 1963-06-04 1965-10-26 Kurt J Rorig 3, 5-dialkylated-2-amino-6-aryl-4(3h)-pyrimidinones
IT1153066B (it) * 1982-11-18 1987-01-14 Mentedison S P A Derivati del pirimidin-4-one ad attivita' erbicida
US4725600A (en) * 1984-07-13 1988-02-16 Fujisawa Pharmaceutical Co., Ltd. Pyrimidine compounds having activity as a cardiotonic anti-hypertensive cerebrovascular vasodilator and anti-platelet aggregation agent
ATE144500T1 (de) * 1992-07-17 1996-11-15 Rohm & Haas 2-substituierte pyrimidine und ihre verwendung als herbizide

Also Published As

Publication number Publication date
DK0579425T3 (da) 1996-11-18
BR9302830A (pt) 1994-02-16
ZA935032B (en) 1994-01-17
KR940005589A (ko) 1994-03-21
US5397767A (en) 1995-03-14
US5298481A (en) 1994-03-29
EP0579425A1 (fr) 1994-01-19
ES2092768T3 (es) 1996-12-01
AU672408B2 (en) 1996-10-03
CN1081439A (zh) 1994-02-02
EP0579425B1 (fr) 1996-10-09
AU4175293A (en) 1994-01-20
JPH06100544A (ja) 1994-04-12
ATE143951T1 (de) 1996-10-15
NZ248089A (en) 1996-01-26
DE69305265D1 (de) 1996-11-14
HU9302054D0 (en) 1993-11-29
CA2099923A1 (fr) 1994-01-18
IL106231A0 (en) 1993-11-15
HUT65123A (en) 1994-04-28
TW239063B (fr) 1995-01-21
DE69305265T2 (de) 1997-05-07
MX9304218A (es) 1994-02-28

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)