HRP20041065A2 - Non-nucleoside reverse transcriptase inhibitors - Google Patents

Non-nucleoside reverse transcriptase inhibitors Download PDF

Info

Publication number: HRP20041065A2
Authority: HR; Croatia
Prior art keywords: alkyl; cooh; optionally substituted; image; mmol
Prior art date: 2002-05-16

Application number

HR20041065A

Other languages

English (en)

Croatian (hr)

Inventor

Yoakim Christiane

Thavonekham Bounkham

Simoneau Bruno

Naud Julie

O'meara Jeffrey

Malenfant Eric

R. Landry Serge

Original Assignee

Boehringer Ingelheim International Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-05-16

Filing date

2003-05-14

Publication date

2005-04-30

2003-05-14 Application filed by Boehringer Ingelheim International Gmbh filed Critical Boehringer Ingelheim International Gmbh

2005-04-30 Publication of HRP20041065A2 publication Critical patent/HRP20041065A2/hr

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Virology (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
AIDS & HIV (AREA)
Engineering & Computer Science (AREA)
Tropical Medicine & Parasitology (AREA)
Molecular Biology (AREA)
Bioinformatics & Cheminformatics (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

HR20041065A 2002-05-16 2003-05-14 Non-nucleoside reverse transcriptase inhibitors HRP20041065A2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US38088602P	2002-05-16	2002-05-16
PCT/CA2003/000718 WO2003097644A2 (en)	2002-05-16	2003-05-14	Non-nucleoside reverse transcriptase inhibitors

Publications (1)

Publication Number	Publication Date
HRP20041065A2 true HRP20041065A2 (en)	2005-04-30

Family

ID=29550032

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HR20041065A HRP20041065A2 (en)	2002-05-16	2003-05-14	Non-nucleoside reverse transcriptase inhibitors

Country Status (28)

Country	Link
US (1)	US6806265B2 (es)
EP (1)	EP1506195B1 (es)
JP (1)	JP4230448B2 (es)
KR (1)	KR20050008716A (es)
CN (1)	CN1318421C (es)
AR (1)	AR040027A1 (es)
AT (1)	ATE412653T1 (es)
AU (1)	AU2003229186A1 (es)
BR (1)	BR0310033A (es)
CA (1)	CA2485916C (es)
DE (1)	DE60324418D1 (es)
EA (1)	EA009178B1 (es)
EC (1)	ECSP045432A (es)
ES (1)	ES2315492T3 (es)
HR (1)	HRP20041065A2 (es)
IL (1)	IL163753A0 (es)
MX (1)	MXPA04010409A (es)
MY (1)	MY134646A (es)
NO (1)	NO20044104L (es)
NZ (1)	NZ536736A (es)
PE (1)	PE20040365A1 (es)
PL (1)	PL371663A1 (es)
RS (1)	RS98004A (es)
TW (1)	TW200404071A (es)
UA (1)	UA79285C2 (es)
UY (1)	UY27809A1 (es)
WO (1)	WO2003097644A2 (es)
ZA (1)	ZA200406912B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0302094D0 (en)	2003-01-29	2003-02-26	Pharmagene Lab Ltd	EP4 receptor antagonists
EP1610797A1 (en) *	2003-03-27	2006-01-04	Boehringer Ingelheim International GmbH	Antiviral combination of nevirapine and a further antiretroviral compound
KR101415503B1 (ko) *	2003-07-17	2014-07-04	플렉시콘, 인코퍼레이티드	Ｐｐａｒ 활성 화합물
US7348338B2 (en)	2003-07-17	2008-03-25	Plexxikon, Inc.	PPAR active compounds
GB0324269D0 (en)	2003-10-16	2003-11-19	Pharmagene Lab Ltd	EP4 receptor antagonists
DE102004051277A1 (de) *	2004-10-21	2006-04-27	Merck Patent Gmbh	Heterocyclische Carbonylverbindungen
US7531568B2 (en) *	2004-11-30	2009-05-12	Plexxikon, Inc.	PPAR active compounds
AU2006287528A1 (en) *	2005-09-07	2007-03-15	Plexxikon, Inc.	1 , 4 and 1 , 5-disubstituted indole derivatives for use as PPAR active compounds
AU2006287513A1 (en) *	2005-09-07	2007-03-15	Plexxikon, Inc.	1, 3-disubstituted indole derivatives for use as PPAR modulators
EP1940767A2 (en) *	2005-09-07	2008-07-09	Plexxikon, Inc.	Pparactive compounds
US8492428B2 (en)	2005-09-20	2013-07-23	Mayo Foundation For Medical Education And Research	Small-molecule botulinum toxin inhibitors
PE20090159A1 (es) *	2007-03-08	2009-02-21	Plexxikon Inc	COMPUESTOS DERIVADOS DE ACIDO INDOL-PROPIONICO COMO MODULADORES PPARs
JP2017535573A (ja)	2014-11-25	2017-11-30	バイエルファーマアクチエンゲゼルシャフト	置換されたピリドベンゾジアゼピノン誘導体およびそれの使用
CN110446708B (zh)	2017-07-21	2022-12-02	安塔比奥公司	化学化合物
MD3762368T2 (ro)	2018-03-08	2022-07-31	Incyte Corp	Compuși diol aminopirazină ca inhibitori ai PI3K-Y
US11046658B2 (en)	2018-07-02	2021-06-29	Incyte Corporation	Aminopyrazine derivatives as PI3K-γ inhibitors
JP2024534799A (ja) *	2021-08-20	2024-09-26	エナンタファーマシューティカルズインコーポレイテッド	１７－ベータ－ヒドロキシステロイドデヒドロゲナーゼ１３型阻害剤及びその使用方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5366972A (en)	1989-04-20	1994-11-22	Boehringer Ingelheim Pharmaceuticals, Inc.	5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
US5705499A (en) *	1995-10-06	1998-01-06	Boehringer Ingelheim Pharmaceuticals, Inc.	8-arylalkyl- and 8-arylheteroalkyl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-e! 1!diazepines and their use in the treatment of HIV-1 infection
TWI270547B (en)	2000-06-16	2007-01-11	Boehringer Ingelheim Ca Ltd	Non-nucleoside reverse transcriptase inhibitors
US6716836B2 (en)	2001-03-22	2004-04-06	Boehringer Ingelheim (Canada) Ltd.	Non-nucleoside reverse transcriptase inhibitors
US6673791B2 (en)	2001-07-30	2004-01-06	Boehringer Ingelheim (Canada) Ltd.	Non-nucleoside reverse transcriptase inhibitors

2003
- 2003-05-06 US US10/430,116 patent/US6806265B2/en not_active Expired - Lifetime
- 2003-05-13 MY MYPI20031796A patent/MY134646A/en unknown
- 2003-05-14 ES ES03724719T patent/ES2315492T3/es not_active Expired - Lifetime
- 2003-05-14 JP JP2004505376A patent/JP4230448B2/ja not_active Expired - Fee Related
- 2003-05-14 PE PE2003000461A patent/PE20040365A1/es not_active Application Discontinuation
- 2003-05-14 EP EP03724719A patent/EP1506195B1/en not_active Expired - Lifetime
- 2003-05-14 EA EA200401482A patent/EA009178B1/ru not_active IP Right Cessation
- 2003-05-14 DE DE60324418T patent/DE60324418D1/de not_active Expired - Lifetime
- 2003-05-14 AU AU2003229186A patent/AU2003229186A1/en not_active Abandoned
- 2003-05-14 PL PL03371663A patent/PL371663A1/xx not_active Application Discontinuation
- 2003-05-14 RS YU98004A patent/RS98004A/sr unknown
- 2003-05-14 IL IL16375303A patent/IL163753A0/xx unknown
- 2003-05-14 UA UA20041210291A patent/UA79285C2/uk unknown
- 2003-05-14 WO PCT/CA2003/000718 patent/WO2003097644A2/en not_active Ceased
- 2003-05-14 KR KR10-2004-7018428A patent/KR20050008716A/ko not_active Withdrawn
- 2003-05-14 CN CNB038111187A patent/CN1318421C/zh not_active Expired - Fee Related
- 2003-05-14 BR BR0310033-2A patent/BR0310033A/pt not_active IP Right Cessation
- 2003-05-14 MX MXPA04010409A patent/MXPA04010409A/es active IP Right Grant
- 2003-05-14 CA CA002485916A patent/CA2485916C/en not_active Expired - Fee Related
- 2003-05-14 AT AT03724719T patent/ATE412653T1/de active
- 2003-05-14 HR HR20041065A patent/HRP20041065A2/hr not_active Application Discontinuation
- 2003-05-14 NZ NZ536736A patent/NZ536736A/en unknown
- 2003-05-15 UY UY27809A patent/UY27809A1/es not_active Application Discontinuation
- 2003-05-15 TW TW092113234A patent/TW200404071A/zh unknown
- 2003-05-16 AR ARP030101708A patent/AR040027A1/es unknown
2004
- 2004-08-31 ZA ZA200406912A patent/ZA200406912B/xx unknown
- 2004-09-27 NO NO20044104A patent/NO20044104L/no unknown
- 2004-11-16 EC EC2004005432A patent/ECSP045432A/es unknown

Also Published As

Publication number	Publication date
ATE412653T1 (de)	2008-11-15
PE20040365A1 (es)	2004-07-22
ES2315492T3 (es)	2009-04-01
IL163753A0 (en)	2005-12-18
KR20050008716A (ko)	2005-01-21
US20040006071A1 (en)	2004-01-08
PL371663A1 (en)	2005-06-27
CA2485916A1 (en)	2003-11-27
MXPA04010409A (es)	2005-02-17
BR0310033A (pt)	2005-02-15
HK1080849A1 (en)	2006-05-04
WO2003097644A3 (en)	2004-02-05
WO2003097644A2 (en)	2003-11-27
EP1506195A2 (en)	2005-02-16
UA79285C2 (en)	2007-06-11
RS98004A (sr)	2006-12-15
CN1653066A (zh)	2005-08-10
AU2003229186A1 (en)	2003-12-02
EA200401482A1 (ru)	2005-06-30
US6806265B2 (en)	2004-10-19
AR040027A1 (es)	2005-03-09
EA009178B1 (ru)	2007-12-28
NZ536736A (en)	2006-11-30
MY134646A (en)	2007-12-31
CA2485916C (en)	2009-12-08
JP2005526851A (ja)	2005-09-08
TW200404071A (en)	2004-03-16
CN1318421C (zh)	2007-05-30
DE60324418D1 (de)	2008-12-11
ZA200406912B (en)	2006-06-28
UY27809A1 (es)	2003-12-31
NO20044104L (no)	2004-12-01
ECSP045432A (es)	2005-01-03
JP4230448B2 (ja)	2009-02-25
EP1506195B1 (en)	2008-10-29

Legal Events

Date	Code	Title	Description
2005-04-30	A1OB	Publication of a patent application
2005-10-26	ARAI	Request for the grant of a patent on the basis of the submitted results of a substantive examination of a patent application
2007-05-03	ODRP	Renewal fee for the maintenance of a patent	Payment date: 20070503 Year of fee payment: 5
2009-01-13	OBST	Application withdrawn

Publication	Publication Date	Title
CA2485916C (en)	2009-12-08	Non-nucleoside reverse transcriptase inhibitors
US7273861B2 (en)	2007-09-25	Non-nucleoside reverse transcriptase inhibitors
EP1554276B1 (en)	2006-06-28	Non-nucleoside reverse transcriptase inhibitors
CA2450868C (en)	2009-06-02	Non-nucleoside reverse transcriptase inhibitors
AU2001270370A1 (en)	2002-03-14	Non-nucleoside reverse transcriptase inhibitors
EP1373267B1 (en)	2005-02-02	Non-nucleoside reverse transcriptase inhibitors
EP1305313A1 (en)	2003-05-02	Fused heterocyclic derivatives as phosphodiesterase inhibitors
KR20250017244A (ko)	2025-02-04	플라비바이러스 저해제
HK1080849B (en)	2007-09-21	Non-nucleoside reverse transcriptase inhibitors
CA2479216C (en)	2009-08-18	Dipyridodiazepinones as reverse transcriptase inhibitors