HRP20090078A2 - Novel pyridazine compound and use thereof - Google Patents

Novel pyridazine compound and use thereof

Info

Publication number
HRP20090078A2
HRP20090078A2 HR20090078A HRP20090078A HRP20090078A2 HR P20090078 A2 HRP20090078 A2 HR P20090078A2 HR 20090078 A HR20090078 A HR 20090078A HR P20090078 A HRP20090078 A HR P20090078A HR P20090078 A2 HRP20090078 A2 HR P20090078A2
Authority
HR
Croatia
Prior art keywords
pyridazine compound
novel pyridazine
compound
novel
solvates
Prior art date
Application number
HR20090078A
Other languages
English (en)
Croatian (hr)
Inventor
S. Bondy Steven
C. Dahl Terrence
A. Oare David
Oliyai Reza
C. Tse Winston
Zia Vahid
Original Assignee
Gilead Sciences
K.U. Leuven Research & Development
Gerhard Puerstinger
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences, K.U. Leuven Research & Development, Gerhard Puerstinger filed Critical Gilead Sciences
Publication of HRP20090078A2 publication Critical patent/HRP20090078A2/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HR20090078A 2006-07-07 2007-07-06 Novel pyridazine compound and use thereof HRP20090078A2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US81928906P 2006-07-07 2006-07-07
US83240306P 2006-07-21 2006-07-21
US83276906P 2006-07-24 2006-07-24
PCT/US2007/015553 WO2008005519A2 (en) 2006-07-07 2007-07-06 Novel pyridazine compound and use thereof

Publications (1)

Publication Number Publication Date
HRP20090078A2 true HRP20090078A2 (en) 2009-06-30

Family

ID=38814329

Family Applications (2)

Application Number Title Priority Date Filing Date
HR20090078A HRP20090078A2 (en) 2006-07-07 2007-07-06 Novel pyridazine compound and use thereof
HR20100180T HRP20100180T1 (hr) 2006-07-07 2007-07-06 Novi spoj piridazina i njegova primjena

Family Applications After (1)

Application Number Title Priority Date Filing Date
HR20100180T HRP20100180T1 (hr) 2006-07-07 2007-07-06 Novi spoj piridazina i njegova primjena

Country Status (27)

Country Link
US (3) US8569487B2 (sr)
EP (1) EP2038275B1 (sr)
JP (1) JP4958974B2 (sr)
KR (1) KR101143596B1 (sr)
CN (1) CN102617571B (sr)
AP (1) AP3430A (sr)
AR (1) AR061969A1 (sr)
AT (1) ATE454384T1 (sr)
AU (1) AU2007269614B2 (sr)
CA (1) CA2656415C (sr)
CY (1) CY1112107T1 (sr)
DE (1) DE602007004220D1 (sr)
DK (1) DK2038275T3 (sr)
EA (1) EA019452B1 (sr)
ES (1) ES2339298T3 (sr)
HR (2) HRP20090078A2 (sr)
IL (1) IL195528A (sr)
MX (1) MX2009000235A (sr)
NO (1) NO20090595L (sr)
NZ (1) NZ574312A (sr)
PL (1) PL2038275T3 (sr)
PT (1) PT2038275E (sr)
RS (1) RS51336B (sr)
SG (1) SG175604A1 (sr)
SI (1) SI2038275T1 (sr)
TW (1) TWI360549B (sr)
WO (1) WO2008005519A2 (sr)

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AR077125A1 (es) 2009-06-23 2011-08-03 Gilead Sciences Inc Combinaciones farmaceuticas utiles para tratar el vhc
EA201200650A1 (ru) 2009-10-30 2012-12-28 Бёрингер Ингельхайм Интернациональ Гмбх Курсы комбинированного лечения вируса гепатита с, включающие bi201335, интерферон-альфа и рибавирин
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EP2571882A1 (en) 2010-05-21 2013-03-27 Gilead Sciences, Inc. Heterocyclic flaviviridae virus inhibitors
WO2011156757A1 (en) * 2010-06-10 2011-12-15 Gilead Sciences, Inc. Combination of anti-hcv compounds with ribavirin for the treatment of hcv
US20130273005A1 (en) * 2010-12-20 2013-10-17 Gilead Sciences, Inc. Methods for treating hcv
DK2701720T3 (en) 2011-04-28 2017-10-09 Oncopeptides Ab Lyophilized preparation with cytotoxic dipeptides
EP2709613B2 (en) 2011-09-16 2020-08-12 Gilead Pharmasset LLC Methods for treating hcv
SMT202000058T1 (it) 2012-10-26 2020-03-13 Oncopeptides Ab Preparazioni liofilizzate di melfalan flufenammide
EP2950786B1 (en) 2013-01-31 2019-11-27 Gilead Pharmasset LLC Combination formulation of two antiviral compounds
JP7381190B2 (ja) 2014-12-26 2023-11-15 エモリー・ユニバーシテイ Ｎ４－ヒドロキシシチジン及び誘導体並びにそれに関連する抗ウイルス用途
PT3706762T (pt) 2017-12-07 2024-12-05 Univ Emory N4-hidroxicitidina e derivados e utilizações antivirais relacionadas com os mesmos

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Also Published As

Publication number Publication date
IL195528A (en) 2014-07-31
US7956184B2 (en) 2011-06-07
CA2656415C (en) 2012-05-22
NO20090595L (no) 2009-04-07
AP3430A (en) 2015-09-30
US7754720B2 (en) 2010-07-13
JP2009542692A (ja) 2009-12-03
CY1112107T1 (el) 2015-11-04
AU2007269614A1 (en) 2008-01-10
EP2038275B1 (en) 2010-01-06
PT2038275E (pt) 2010-04-08
KR101143596B1 (ko) 2012-05-11
PL2038275T3 (pl) 2010-08-31
DK2038275T3 (da) 2010-05-10
HRP20100180T1 (hr) 2010-06-30
ES2339298T3 (es) 2010-05-18
AU2007269614B2 (en) 2011-09-08
TW200811180A (en) 2008-03-01
EP2038275A2 (en) 2009-03-25
CA2656415A1 (en) 2008-01-10
NZ574312A (en) 2012-02-24
US20080199427A1 (en) 2008-08-21
US20100152444A1 (en) 2010-06-17
HK1123803A1 (en) 2009-06-26
KR20090028813A (ko) 2009-03-19
US20100063059A1 (en) 2010-03-11
ATE454384T1 (de) 2010-01-15
WO2008005519A2 (en) 2008-01-10
WO2008005519A3 (en) 2008-04-24
SI2038275T1 (sl) 2010-06-30
AP2008004717A0 (en) 2008-12-31
TWI360549B (en) 2012-03-21
AR061969A1 (es) 2008-08-10
EA200900156A1 (ru) 2009-06-30
CN102617571B (zh) 2015-06-10
EA019452B1 (ru) 2014-03-31
JP4958974B2 (ja) 2012-06-20
IL195528A0 (en) 2009-09-01
SG175604A1 (en) 2011-11-28
MX2009000235A (es) 2009-01-23
DE602007004220D1 (de) 2010-02-25
CN102617571A (zh) 2012-08-01
RS51336B (sr) 2011-02-28
US8569487B2 (en) 2013-10-29

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