HRP20090578T1 - Postupak za pripravu dorzolamida - Google Patents

Postupak za pripravu dorzolamida Download PDF

Info

Publication number
HRP20090578T1
HRP20090578T1 HR20090578T HRP20090578T HRP20090578T1 HR P20090578 T1 HRP20090578 T1 HR P20090578T1 HR 20090578 T HR20090578 T HR 20090578T HR P20090578 T HRP20090578 T HR P20090578T HR P20090578 T1 HRP20090578 T1 HR P20090578T1
Authority
HR
Croatia
Prior art keywords
dorzolamide
formula
racemate
image
camphorsulfonic acid
Prior art date
Application number
HR20090578T
Other languages
English (en)
Croatian (hr)
Inventor
Maragni Paolo
Michieletto Ivan
Cotarca Livius
Original Assignee
Zach System S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zach System S.P.A. filed Critical Zach System S.P.A.
Publication of HRP20090578T1 publication Critical patent/HRP20090578T1/hr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Catalysts (AREA)
  • Dental Preparations (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
HR20090578T 2006-04-21 2007-04-16 Postupak za pripravu dorzolamida HRP20090578T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06112883 2006-04-21
PCT/EP2007/053691 WO2007122130A1 (en) 2006-04-21 2007-04-16 Process for preparing dorzolamide

Publications (1)

Publication Number Publication Date
HRP20090578T1 true HRP20090578T1 (hr) 2009-11-30

Family

ID=38137401

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20090578T HRP20090578T1 (hr) 2006-04-21 2007-04-16 Postupak za pripravu dorzolamida

Country Status (14)

Country Link
US (1) US8183391B2 (de)
EP (1) EP2010544B1 (de)
JP (1) JP5097770B2 (de)
CN (1) CN101426795B (de)
AT (1) ATE438649T1 (de)
CA (1) CA2646133A1 (de)
CY (1) CY1110510T1 (de)
DE (1) DE602007001885D1 (de)
DK (1) DK2010544T3 (de)
ES (1) ES2331162T3 (de)
HR (1) HRP20090578T1 (de)
PT (1) PT2010544E (de)
SI (1) SI2010544T1 (de)
WO (1) WO2007122130A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20121165A1 (it) 2012-07-03 2014-01-04 Zach System Spa Processo di riduzione asimmetrica
CN103497202B (zh) * 2013-10-23 2015-12-02 武汉武药科技有限公司 盐酸多佐胺中间体的合成方法
US20160332962A1 (en) * 2015-05-13 2016-11-17 Janssen Pharmaceutica Nv (s)-csa salt of s-ketamine, (r)-csa salt of s-ketamine and processes for the preparation of s-ketamine
CN108822127B (zh) * 2018-05-30 2020-05-15 沈阳药科大学 4-羟亚胺基噻吩并[2,3-b]噻喃-2-甲酰胺类化合物及其用途
CN108822126B (zh) * 2018-05-30 2020-05-15 沈阳药科大学 噻吩并噻喃甲酰基哌嗪类化合物及其医药用途
CN108586485B (zh) * 2018-05-30 2020-05-15 沈阳药科大学 1-(4-羟亚胺基噻吩并[2,3-b]噻喃甲酰基)哌嗪类化合物及其应用
CN110903299A (zh) * 2018-09-17 2020-03-24 武汉武药科技有限公司 一种盐酸多佐胺的精制方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3810899A (en) * 1972-03-10 1974-05-14 Hoffmann La Roche 2-hydroxy-n-substituted-morphinan derivatives
DD150456A5 (de) * 1979-03-01 1981-09-02 Ciba Geigy Ag Verfahren zur herstellung von derivaten des 3-amino-1,2-propandiols
US4863922A (en) * 1984-12-12 1989-09-05 Merck & Co., Inc. Substituted aromatic sulfonamides as antiglaucoma agents, compositions and use
JP4218310B2 (ja) * 2002-11-06 2009-02-04 住友化学株式会社 光学活性2−アミノ−2−フェニルエタノール類の製造方法およびその中間体
US20050059696A1 (en) 2003-05-08 2005-03-17 Dr. Reddy's Laboratories Limited Process for the recovery of S -(+)-methyl- (2-chlorophenyl)- (6,7-dihydro- 4H-thieno [3,2-c] pyrid-5-yl) acetate hydrogen sulfate (clopidogrel bisulfate) from its (R) and mixture of (R) and (S)- isomers
CN1293041C (zh) * 2003-05-30 2007-01-03 上海实业化工有限公司 D-(-)-1-苯甘氨酸的制备方法
DE10336185A1 (de) * 2003-08-07 2005-02-24 Bayer Chemicals Ag Enantiomerenangereicherte 1-Phenylethylamine
US8198316B2 (en) * 2004-07-09 2012-06-12 Fdc Ltd Process for the preparation of 5,6 -dihydro -4H-4(S)-ethylamino-6(S)-methylthieno[2,3-b] thiopyran-2-sulfonamide- 7,7 -dioxide and its salt

Also Published As

Publication number Publication date
CN101426795A (zh) 2009-05-06
JP2009534349A (ja) 2009-09-24
SI2010544T1 (sl) 2009-12-31
CN101426795B (zh) 2011-01-12
US20090275759A1 (en) 2009-11-05
EP2010544B1 (de) 2009-08-05
WO2007122130A1 (en) 2007-11-01
DE602007001885D1 (de) 2009-09-17
PT2010544E (pt) 2009-11-03
US8183391B2 (en) 2012-05-22
CA2646133A1 (en) 2007-11-01
DK2010544T3 (da) 2009-11-30
ATE438649T1 (de) 2009-08-15
EP2010544A1 (de) 2009-01-07
CY1110510T1 (el) 2015-04-29
JP5097770B2 (ja) 2012-12-12
ES2331162T3 (es) 2009-12-22

Similar Documents

Publication Publication Date Title
CN103980275B (zh) 磷酸二酯酶5抑制剂他达拉非的制备方法
WO2009101634A3 (en) A novel process for the preparation of eszopiclone
JP5097770B2 (ja) ドルゾラミドの調製方法
WO2013020388A1 (zh) 一种(s)-奥拉西坦的纯化方法
EP2683724B1 (de) Asymetrisches reduktionsverfahren
WO2007094006A1 (en) Process for preparation of clopidogrel bisulfate form 1
CN102320986A (zh) 一种氯吡格雷中间体的制备方法
CN110642765A (zh) 一种d-对甲砜基苯丝氨酸乙酯的合成方法
CN104151313A (zh) 一种纯化他达拉非中间体的方法
NO20084217L (no) Fremgangsmate for fremstilling av polymorf form I av (S)-(+)-metyl-α-(2-klorfenyl)-6,7-dihydrotieno-[3,2-c]pyridin-5(4H)-acetathydrogensulfat
CN112574197B (zh) 一种化合物c的手性纯化方法
CN102603594A (zh) (s)-奥拉西坦的制备方法
EP2264016A3 (de) Verfahren zur Herstellung einer reinen Form von 2-Methyl-4-(4-Methyl-1-Piperazinyl)-10H-thieno[2,3-B][1,5]-Benzodiazepin
CA2589146A1 (en) Process for producing muscarine receptor antagonist and intermediate therefor
JP2023521100A (ja) 4,5-ジヒドロ-1h-ピラゾール及び中間体を製造する方法
WO2012143801A1 (en) Manufacturing process for tadalafil from racemic or l-tryptophan
TW200611901A (en) Method for producing 1, 3-dioxolan-4, 6-dione compound
CN102336766A (zh) 一锅法制备消旋氯吡格雷的方法
CN106749569B (zh) 一种pf1022a的分离纯化方法
CN103012264A (zh) 3-取代氨基-六氢-1h-氮杂环庚烷的拆分方法
WO2016028016A1 (ko) D-아르기닌의 제조 방법
WO2009008303A1 (ja) 光学活性ミルタザピンの製造方法
CN103435617B (zh) 一种6,7-二氢-5H-吡咯并[1,2-a]咪唑-2-甲醛的合成方法
CN103131747A (zh) 利用生物酶手性拆分合成(s)-3-(4-羟基苯基)-3-甲氨基丙酸的方法
EP1765828B1 (de) VERBESSERTES VERFAHREN ZUR HERSTELLUNG VON 5,6 -DIHYDRO -4H-4(S)-ETHYLAMIN-6(S)-METHYLTHIENO[2,3-b] THIOPYRAN-2-SULFONAMID- 7,7 -DIOXID UND SEINEN SALZEN