HUE034802T2 - Kinurenin-3-monooxigenáz gátló, gyógyszerészeti készítmények és eljárás az elõzõek alkalmazására - Google Patents

Kinurenin-3-monooxigenáz gátló, gyógyszerészeti készítmények és eljárás az elõzõek alkalmazására Download PDF

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HUE034802T2
HUE034802T2 HUE12828501A HUE12828501A HUE034802T2 HU E034802 T2 HUE034802 T2 HU E034802T2 HU E12828501 A HUE12828501 A HU E12828501A HU E12828501 A HUE12828501 A HU E12828501A HU E034802 T2 HUE034802 T2 HU E034802T2
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Hungary
Prior art keywords
chloro
phenyl
pyrimidine
carboxylic acid
added
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HUE12828501A
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English (en)
Inventor
Stephen Martin Courtney
Michael Prime
William Mitchell
Christopher John Brown
Aguiar Pena Paula C De
Peter Johnson
Celia Dominguez
Sherman Leticia M Toledo
Ignacio Munoz
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Chdi Foundation Inc
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Publication of HUE034802T2 publication Critical patent/HUE034802T2/hu

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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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Claims (2)

  1. Süabadaiios igénypontok t4épláfei? egy kémiai isnötás a 64'3-W6r-4 e.lKk3propoxe^eai)- pifi!ytid:e,.4-ksrbonsav és gyogysxas'ésssíijsg sifepphsié ®$ mzmmmm* 2. %i^ys2eFé8Z^tobí^,;5:ám% tetainwsa as 1. igénypont szerinti legalább sgy Mmíél onMét és layaiébb agy gyógyszeiéssoliíog <s!k>g«Shaíé segédanyagot.
  2. 3. As 1. igénypont so«ríni: legalább égy kémiai snteàs klnoíeníO'Snríónö-oxigenás aktivitás áíiaí médiáit neiiiociegensratfv patológiás alapotokat fascism aiispotok és -"endeiiénesaégek kezeléséi« szolgád· oijéfé$ban vasé alksimasâsos ogy iíyan kazaléba ïboruló alanyban, amely ian.aisea.ma a.? igénylőm ssorinii iagaiabo egy kémia* anisiés terápiásán hatásos mennyiségének S2 alany sscäsoara történő adagolását. 4 As i igénypont szénné legalább egy kémiai entitás 3 igénypont sseî^Mjâriéb^JliiitîènS aíkáímazést^. ahol a neurodegenerativ patotôgsas aikspol n Humingise-kPr §. Csomapit gybipzetássttél! késxkmsnyeamoiy tariaimas .tgg4Ét^::i8fyÉ..;.^#gyMt'^!lfi!ti gyégyssefósséiS kteftw^pi»iôWtiSsÂt':8'kééÂény.silk«âmé?âsârt^Âr> szémèiykézaièsa eipéék amely kinoranin·S-moon-nxigOiPs skiiyltás Ittál msÄi állapottól vagy iandaitsftéaéégM: saanvosl* aboi ;a klnpronin^· monca ésipriázaktlvstáé ittál nis^^lt'^iipotiVigypftPPbbMbg á Huntington-AOr.
HUE12828501A 2011-08-30 2012-08-28 Kinurenin-3-monooxigenáz gátló, gyógyszerészeti készítmények és eljárás az elõzõek alkalmazására HUE034802T2 (hu)

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