ID23971A - PROSTAGLANDIN TETRAHIDRO SUBSTITUTEDIC C <16> -C <20> AROMATICS USING AS FP AGONISTS - Google Patents

PROSTAGLANDIN TETRAHIDRO SUBSTITUTEDIC C <16> -C <20> AROMATICS USING AS FP AGONISTS

Info

Publication number
ID23971A
ID23971A IDW20000639A ID20000639A ID23971A ID 23971 A ID23971 A ID 23971A ID W20000639 A IDW20000639 A ID W20000639A ID 20000639 A ID20000639 A ID 20000639A ID 23971 A ID23971 A ID 23971A
Authority
ID
Indonesia
Prior art keywords
substitutedic
tetrahidro
prostaglandin
aromatics
agonists
Prior art date
Application number
IDW20000639A
Other languages
Indonesian (id)
Inventor
John August Wos
Mitchell Anthony Delong
Jack S Amburgey Jr
Biswanath De
Haiyan George Dai
Yili Wang
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of ID23971A publication Critical patent/ID23971A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Rheumatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IDW20000639A 1997-09-09 1998-09-04 PROSTAGLANDIN TETRAHIDRO SUBSTITUTEDIC C <16> -C <20> AROMATICS USING AS FP AGONISTS ID23971A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5821797P 1997-09-09 1997-09-09

Publications (1)

Publication Number Publication Date
ID23971A true ID23971A (en) 2000-06-14

Family

ID=22015427

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW20000639A ID23971A (en) 1997-09-09 1998-09-04 PROSTAGLANDIN TETRAHIDRO SUBSTITUTEDIC C <16> -C <20> AROMATICS USING AS FP AGONISTS

Country Status (24)

Country Link
US (1) US5977173A (en)
EP (1) EP1012136B1 (en)
JP (1) JP2001515882A (en)
KR (1) KR20010023839A (en)
CN (1) CN1269786A (en)
AR (1) AR013477A1 (en)
AT (1) ATE270660T1 (en)
AU (1) AU731153B2 (en)
BR (1) BR9811774A (en)
CA (1) CA2303764C (en)
CO (1) CO4970731A1 (en)
DE (1) DE69824966T2 (en)
ES (1) ES2223141T3 (en)
HU (1) HUP0100638A3 (en)
ID (1) ID23971A (en)
IL (1) IL134839A0 (en)
NO (1) NO20001141L (en)
NZ (1) NZ503735A (en)
PE (1) PE115499A1 (en)
PL (1) PL339212A1 (en)
SK (1) SK3372000A3 (en)
TR (1) TR200000671T2 (en)
WO (1) WO1999012895A1 (en)
ZA (1) ZA988230B (en)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4834224B2 (en) * 1999-03-05 2011-12-14 デューク ユニバーシティ C16 unsaturated FP-selective prostaglandin analogs
US6894175B1 (en) 1999-08-04 2005-05-17 The Procter & Gamble Company 2-Decarboxy-2-phosphinico prostaglandin derivatives and methods for their preparation and use
ES2202156T3 (en) 1999-08-04 2004-04-01 Procter & Gamble NEW ANALOGS OF 2-DESCARBOXI-2-PHOSPHINIC PROSTAGLANDINA F.
US20020013294A1 (en) * 2000-03-31 2002-01-31 Delong Mitchell Anthony Cosmetic and pharmaceutical compositions and methods using 2-decarboxy-2-phosphinico derivatives
US20020172693A1 (en) * 2000-03-31 2002-11-21 Delong Michell Anthony Compositions and methods for treating hair loss using non-naturally occurring prostaglandins
US20020037914A1 (en) * 2000-03-31 2002-03-28 Delong Mitchell Anthony Compositions and methods for treating hair loss using C16-C20 aromatic tetrahydro prostaglandins
KR100437873B1 (en) * 2001-05-08 2004-06-26 연성정밀화학(주) Process for preparing prostaglandin derivatives and stereospecific starting material thereof
US8758733B2 (en) 2002-02-04 2014-06-24 Allergan, Inc. Topical treatment for chemotherapy induced eyelash loss or hypotrichosis using prostamide F2 alpha agonists
US7351404B2 (en) 2002-02-04 2008-04-01 Allergan, Inc. Method of enhancing hair growth
US9216183B2 (en) 2002-02-04 2015-12-22 Allergan, Inc. Topical treatment for chemotherapy induced eyelash loss or hypotrichosis using prostamide F2 alpha agonists
WO2006047466A2 (en) * 2004-10-21 2006-05-04 Duke University Ophthamological drugs
US20070254920A1 (en) * 2006-04-26 2007-11-01 Aerie Pharmaceuticals, Inc. Prodrug derivatives of acids using alcohols with homotopic hydroxy groups and methods for their preparation and use
US8455513B2 (en) 2007-01-10 2013-06-04 Aerie Pharmaceuticals, Inc. 6-aminoisoquinoline compounds
EP2214482A4 (en) 2007-10-31 2011-08-24 Pamela Lipkin Prostaglandin analog compositions and methods to treat epithelial-related conditions
US20100074857A1 (en) * 2008-09-23 2010-03-25 Pamela Lipkin Compositions and methods to treat epithelial-related conditions
US8450344B2 (en) 2008-07-25 2013-05-28 Aerie Pharmaceuticals, Inc. Beta- and gamma-amino-isoquinoline amide compounds and substituted benzamide compounds
US8623918B2 (en) 2008-10-29 2014-01-07 Novaer Holdings, Inc. Amino acid salts of prostaglandins
US8722739B2 (en) 2008-10-29 2014-05-13 Novaer Holdings, Inc. Amino acid salts of prostaglandins
WO2010096123A2 (en) 2008-10-29 2010-08-26 Aerie Pharmaceuticals, Inc. Amino acid salts of prostaglandins
US8637558B2 (en) 2008-12-30 2014-01-28 Industry-Academic Cooperation Foundation, Chosun University Thiazolidinedione derivative and use thereof
US20110293549A1 (en) 2009-02-03 2011-12-01 Athena Cosmetics, Inc. Composition, method and kit for enhancing hair
EP3053913B1 (en) 2009-05-01 2018-03-07 Aerie Pharmaceuticals, Inc. Dual mechanism inhibitors for the treatment of disease
US9149484B2 (en) 2009-11-09 2015-10-06 Allergan, Inc. Compositions and methods for stimulating hair growth
PH12012500928A1 (en) 2009-11-09 2012-11-26 Allergan Inc Compositions and methods for stimulating hair growth
US8859616B2 (en) 2011-01-21 2014-10-14 Allergan, Inc. Compounds and methods for enhancing hair growth
DK3811943T3 (en) 2013-03-15 2023-04-03 Aerie Pharmaceuticals Inc Compound for use in the treatment of eye disorders
US9643927B1 (en) 2015-11-17 2017-05-09 Aerie Pharmaceuticals, Inc. Process for the preparation of kinase inhibitors and intermediates thereof
KR102568079B1 (en) 2016-08-31 2023-08-17 에어리 파마슈티컬즈, 인코포레이티드 Ophthalmic compositions
KR20190135027A (en) 2017-03-31 2019-12-05 에어리 파마슈티컬즈, 인코포레이티드 Aryl Cyclopropyl-amino-isoquinolinyl Amide Compound
AU2019337703B2 (en) 2018-09-14 2023-02-02 Aerie Pharmaceuticals, Inc. Aryl cyclopropyl-amino-isoquinolinyl amide compounds

Family Cites Families (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3776938A (en) * 1958-05-28 1973-12-04 S Bergstrom Dihydro-pge1
US4011262A (en) * 1972-07-13 1977-03-08 Pfizer Inc. 13,14-Dihydro-15-substituted-ω-pentanorprostaglandins of the two series
US4024179A (en) * 1972-11-08 1977-05-17 Pfizer Inc. Substituted ω-pentanorprostaglandins
IL43571A (en) * 1972-11-08 1977-08-31 Pfizer Omega-pentanorprostaglandins and their preparation
JPS5720305B2 (en) * 1973-02-28 1982-04-27
DE2365101A1 (en) * 1973-12-21 1975-07-10 Schering Ag NEW PROSTANIC ACID DERIVATIVES AND METHOD FOR THEIR PRODUCTION
DE2460990A1 (en) * 1974-12-21 1976-07-01 Hoechst Ag NEW PROSTAGLANDIN ANALOGS AND PROCEDURES FOR THEIR PRODUCTION
GB1507211A (en) * 1975-02-14 1978-04-12 Ono Pharmaceutical Co Prostaglandin analogues
GB1506816A (en) * 1975-03-31 1978-04-12 Upjohn Co Prostaglandins
DE2517771A1 (en) * 1975-04-18 1976-10-28 Schering Ag NEW PROSTAGLANDIN ACETYLENE ANALOGS AND METHOD FOR THEIR PRODUCTION
US4051238A (en) * 1976-06-03 1977-09-27 The Upjohn Company Treatment of genital tract diseases of domestic animals with prostaglandins
DE2737808A1 (en) * 1976-08-27 1978-03-16 Pfizer 2-SUBSTITUTED ARYL HETEROCYCLIC OMEGA PENTANOR PROSTAGLANDIN
US4206151A (en) * 1978-12-21 1980-06-03 American Cyanamid Company 15-Deoxy-16-hydroxy-16-vinyl or cyclopropyl prostan-1-ols of the E, A and F series
US4621100A (en) * 1981-09-25 1986-11-04 The Upjohn Company Treatment of osteoporosis with prostaglandins
US5166178B1 (en) * 1987-09-18 1998-07-21 R Tech Ueno Ltd Ocular hypotensive agents
DE1300150T1 (en) * 1988-09-06 2003-09-18 Pharmacia Ab, Stockholm Prostaglandin derivatives used to treat glaucoma or hypertension
US5321128A (en) * 1988-09-06 1994-06-14 Kabi Pharmacia Ab Prostaglandin derivatives for the treatment of glaucoma or ocular hypertension
US5296504A (en) * 1988-09-06 1994-03-22 Kabi Pharmacia Prostaglandin derivatives for the treatment of glaucoma or ocular hypertension
CA2030345C (en) * 1989-11-22 1998-12-08 Ryuji Ueno Use of 15-keto-prostaglandin compound for improvement of encephalic function
TW224942B (en) * 1990-04-04 1994-06-11 Adka Ueno Kk
US5302617A (en) * 1990-04-27 1994-04-12 Kabushikikaisha Ueno Seiyaku Oyo Kenkyuio Biochemical treatment with 15-dehydroxy-16-oxoprostaglandin compounds
DE4024347A1 (en) * 1990-07-27 1992-01-30 Schering Ag CYCLOPENTANE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THEIR PHARMACEUTICAL USE
US5409911A (en) * 1992-09-11 1995-04-25 Merck & Co., Inc. Prostaglandin analog for treating osteoporosis
US5688819A (en) * 1992-09-21 1997-11-18 Allergan Cyclopentane heptanoic acid, 2-cycloalkyl or arylalkyl derivatives as therapeutic agents
US5834498A (en) * 1992-09-21 1998-11-10 Allergan Cyclopentane heptan(ene)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
US5332730A (en) * 1992-10-16 1994-07-26 Allergan, Inc. Azido derivatives of cyclopentane heptanoic or heptenoic acid
US5510383A (en) * 1993-08-03 1996-04-23 Alcon Laboratories, Inc. Use of cloprostenol, fluprostenol and their salts and esters to treat glaucoma and ocular hypertension
US5545665A (en) * 1993-12-28 1996-08-13 Allergan Cyclopentane(ene) heptenoic or heptanoic acids and derivatives thereof useful as therapeutic agents
AU7672096A (en) * 1995-06-07 1998-06-03 Alcon Laboratories, Inc. Conformationally rigid aryl- or heteroaryl prostaglandins for use in glaucoma therapy
AU7680096A (en) * 1995-12-22 1997-07-17 Alcon Laboratories, Inc. Combinations of dp and fp type prostaglandins for lowering iop
US5703108A (en) * 1996-02-28 1997-12-30 Pfizer Inc. Bone deposition by certain prostaglandin agonists
US5741810A (en) * 1996-02-29 1998-04-21 Allergan Cyclopentane heptan(ene)oic acid, 2- heteroarylalkenyl derivatives as therapeutic agents
WO1997047595A1 (en) * 1996-06-10 1997-12-18 R-Tech Ueno, Ltd. Endothelin antagonist
ATE221048T1 (en) * 1996-09-17 2002-08-15 Asahi Glass Co Ltd FLUORINATED PROSTAGLAND DERIVATIVES AND MEDICATIONS
WO1998020881A1 (en) * 1996-11-12 1998-05-22 Alcon Laboratories, Inc 15-ketal prostaglandins for the treatment of glaucoma or ocular hypertension
US6353000B1 (en) * 1996-11-12 2002-03-05 Alcon Laboratories, Inc. 11-halo prostaglandins for the treatment of glaucoma or ocular hypertension
WO1998050024A1 (en) * 1997-05-09 1998-11-12 The Mount Sinai School Of Medicine Of The City University Of New York 8-iso-prostaglandins for glaucoma therapy

Also Published As

Publication number Publication date
AR013477A1 (en) 2000-12-27
WO1999012895A1 (en) 1999-03-18
TR200000671T2 (en) 2000-07-21
DE69824966D1 (en) 2004-08-12
NO20001141L (en) 2000-05-04
NO20001141D0 (en) 2000-03-06
US5977173A (en) 1999-11-02
DE69824966T2 (en) 2005-04-07
CA2303764C (en) 2005-02-15
AU731153B2 (en) 2001-03-22
HUP0100638A3 (en) 2002-12-28
ZA988230B (en) 1999-03-09
KR20010023839A (en) 2001-03-26
ES2223141T3 (en) 2005-02-16
IL134839A0 (en) 2001-05-20
NZ503735A (en) 2001-05-25
CO4970731A1 (en) 2000-11-07
EP1012136A1 (en) 2000-06-28
PL339212A1 (en) 2000-12-04
JP2001515882A (en) 2001-09-25
EP1012136B1 (en) 2004-07-07
BR9811774A (en) 2000-08-29
ATE270660T1 (en) 2004-07-15
SK3372000A3 (en) 2000-10-09
HUP0100638A2 (en) 2001-07-30
AU9219398A (en) 1999-03-29
CA2303764A1 (en) 1999-03-18
CN1269786A (en) 2000-10-11
PE115499A1 (en) 2000-02-03

Similar Documents

Publication Publication Date Title
ID23971A (en) PROSTAGLANDIN TETRAHIDRO SUBSTITUTEDIC C &lt;16&gt; -C &lt;20&gt; AROMATICS USING AS FP AGONISTS
ID24836A (en) PROSTAGLANDIN AGONIST
NO20010603D0 (en) 2-substituted-1-piperidylbenzimidazole compounds as ORL 1 receptor agonists
ID24845A (en) AROMATIC C16-C20 SUBSTITUTED PROSTAGLANDIN PROSTAGLANDIN USED AS A FP AGONIST
IS5430A (en) New composition
ID19802A (en) MICROSCOPIC STRUCTURAL COMPOSITIONS
ID16926A (en) ANTIJAMUR COMPOSITIONS WITH BETTER BIOLOGICAL AVAILABILITY
DE69807760D1 (en) Positive working photoresist composition
DK0945132T3 (en) Ibuprofen composition
DK0922386T3 (en) Controlled release compositions
DE69516018D1 (en) THICKENED PERSONIC COMPOSITION
PT946100E (en) HERBICIDAL COMPOSITIONS CONTAINING N-¬ (4,6-DIMETOXYPYRIMIDIN-2-YL) AMINOCARBONYL-5-METHYLSULFONAMIDOMETHYL-2-ALCOXYCARBONYLENZENESULFONAMIDES
ID25508A (en) DEMATOLOGICAL COMPOSITION
NO992470D0 (en) 2-amidazolinyl-amino-indole compounds useful as &lt;alpha&gt; -2-adrenoceptor agonists
NO20001142D0 (en) Aromatic C16-C20 substituted tetrahydro-prostaglandins useful as FP agonists
ID16298A (en) 1,2,3,4-TETRAHIDRONAFTALENA SUBSTITUTED SUBSIDERS
ID21009A (en) COMPOSITION FOR SUPOSITORY
NO990164L (en) Illudin analogs useful as anti-tumor agents
DE69700310D1 (en) Anti-rust composition
DE69825133D1 (en) Fixed fuel composition
ID23250A (en) PAROXSETIN COMPOSITION
ID22060A (en) COMPOUNDS OF 2-IMIDAZOLINYLAMINOBENZOKSAZOL USE AS ADRENOSEPTOR AGONISTS
ID21906A (en) ADESIVE COMPOSITION
ID16154A (en) STABILIZED MONOMER COMPOSITION
ID23429A (en) SOLID SERTRALINA COMPOSITIONS