ID24267A - Enansiomer-enansiomer dari 4-[[(sianoimino) [(1,2,2-trimetilpropil) amino] metil] amino] benzonitril - Google Patents

Enansiomer-enansiomer dari 4-[[(sianoimino) [(1,2,2-trimetilpropil) amino] metil] amino] benzonitril

Info

Publication number
ID24267A
ID24267A IDW20000274A ID20000274A ID24267A ID 24267 A ID24267 A ID 24267A ID W20000274 A IDW20000274 A ID W20000274A ID 20000274 A ID20000274 A ID 20000274A ID 24267 A ID24267 A ID 24267A
Authority
ID
Indonesia
Prior art keywords
amino
trimethylopopil
sianoimino
enansiomers
benzonitril
Prior art date
Application number
IDW20000274A
Other languages
English (en)
Inventor
Karnail S Atwal
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ID24267A publication Critical patent/ID24267A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/43Guanidines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00Preparations for affecting hair growth
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/28Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to cyano groups, e.g. cyanoguanidines, dicyandiamides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07Optical isomers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Dermatology (AREA)
  • Birds (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IDW20000274A 1997-08-13 1998-08-03 Enansiomer-enansiomer dari 4-[[(sianoimino) [(1,2,2-trimetilpropil) amino] metil] amino] benzonitril ID24267A (id)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5556897P 1997-08-13 1997-08-13
US7136498P 1998-01-15 1998-01-15

Publications (1)

Publication Number Publication Date
ID24267A true ID24267A (id) 2000-07-13

Family

ID=26734360

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW20000274A ID24267A (id) 1997-08-13 1998-08-03 Enansiomer-enansiomer dari 4-[[(sianoimino) [(1,2,2-trimetilpropil) amino] metil] amino] benzonitril

Country Status (20)

Country Link
US (3) US6013668A (id)
EP (1) EP1003502A4 (id)
JP (1) JP2001515034A (id)
KR (1) KR20010022672A (id)
CN (1) CN1265589A (id)
AR (1) AR015149A1 (id)
AU (1) AU736687B2 (id)
BR (1) BR9811485A (id)
CA (1) CA2300414A1 (id)
CO (1) CO4750804A1 (id)
HU (1) HUP0003417A3 (id)
ID (1) ID24267A (id)
IL (1) IL133826A0 (id)
NO (1) NO20000686L (id)
NZ (1) NZ502125A (id)
PE (1) PE109199A1 (id)
PL (1) PL338668A1 (id)
TR (1) TR200000343T2 (id)
UY (1) UY25129A1 (id)
WO (1) WO1999008673A1 (id)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6458835B2 (en) * 1997-08-13 2002-10-01 Bristol-Myers Squibb Company Method of inhibiting or treating chemotherapy-induced hair loss
AU2005214167B2 (en) * 2004-02-13 2008-08-07 Warner-Lambert Company Llc Androgen receptor modulators
CN100475781C (zh) * 2004-02-13 2009-04-08 沃尼尔·朗伯有限责任公司 雄激素受体调节剂
CA2563291A1 (en) 2004-04-13 2005-10-27 Warner-Lambert Company Llc 4-cyano-phenoxy-alkyl carboxyl derivatives as androgen modulators
BRPI0509980A (pt) 2004-04-22 2007-10-16 Warner Lambert Co moduladores de androgênio
BRPI0513020A (pt) 2004-07-08 2008-04-22 Warner Lambert Co moduladores de andrÈgenio, seus usos, composição farmacêutica, formulação farmacêutica tópica e artigo de fabricação
TW200724139A (en) 2005-05-05 2007-07-01 Warner Lambert Co Androgen modulators
CN108440307B (zh) * 2018-04-16 2020-11-17 浙江工业大学 一种手性胺类化合物的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1489879A (en) * 1974-12-20 1977-10-26 Leo Pharm Prod Ltd N'-cyano-n'-3-pyridylguanidines
US4596812A (en) * 1976-05-24 1986-06-24 The Upjohn Company Methods and solutions for treating male pattern alopecia
US4139619A (en) * 1976-05-24 1979-02-13 The Upjohn Company 6-Amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidine, topical compositions and process for hair growth
US5244664A (en) * 1988-01-21 1993-09-14 Leo Pharmaceutical Products Ltd. Topical preparation for treatment of alopecia
US5011837A (en) * 1988-08-09 1991-04-30 E. R. Squibb & Sons, Inc. Aryl cyanoguanidines: potassium channel activators and method of making same
GB8908063D0 (en) * 1989-04-11 1989-05-24 Beecham Group Plc Novel compounds
JP3004718B2 (ja) * 1990-08-10 2000-01-31 ファルマシア・アンド・アップジョン・カンパニー カリウムチャネルオープナーおよび5α―レダクターゼ抑制剤を用いる育毛刺激
WO1992009259A1 (en) * 1990-11-29 1992-06-11 The Upjohn Company Stimulation of hair growth with potassium channel openers and an androgen receptor blocker
USH1480H (en) * 1993-12-09 1995-09-05 The Procter & Gamble Company Methods of using dyphylline for the promotion of hair growth
FR2740331B1 (fr) * 1995-10-25 1997-12-19 Sederma Sa Nouvelles compositions cosmetiques pour le traitement des cheveux et du cuir chevelu

Also Published As

Publication number Publication date
JP2001515034A (ja) 2001-09-18
EP1003502A1 (en) 2000-05-31
PE109199A1 (es) 2000-01-30
NO20000686L (no) 2000-03-31
US6262122B1 (en) 2001-07-17
PL338668A1 (en) 2000-11-20
BR9811485A (pt) 2000-09-19
HUP0003417A2 (hu) 2001-02-28
KR20010022672A (ko) 2001-03-26
IL133826A0 (en) 2001-04-30
NZ502125A (en) 2001-08-31
AU736687B2 (en) 2001-08-02
NO20000686D0 (no) 2000-02-11
US6013668A (en) 2000-01-11
CO4750804A1 (es) 1999-03-31
AR015149A1 (es) 2001-04-18
TR200000343T2 (tr) 2000-08-21
EP1003502A4 (en) 2000-06-07
CA2300414A1 (en) 1999-02-25
AU8680898A (en) 1999-03-08
CN1265589A (zh) 2000-09-06
HUP0003417A3 (en) 2002-11-28
WO1999008673A1 (en) 1999-02-25
UY25129A1 (es) 2000-12-29
US6472427B1 (en) 2002-10-29

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