IE34278L - Alpha-carboxy arylmethyl penicillins - Google Patents
Alpha-carboxy arylmethyl penicillinsInfo
- Publication number
- IE34278L IE34278L IE691239A IE123969A IE34278L IE 34278 L IE34278 L IE 34278L IE 691239 A IE691239 A IE 691239A IE 123969 A IE123969 A IE 123969A IE 34278 L IE34278 L IE 34278L
- Authority
- IE
- Ireland
- Prior art keywords
- penicillins
- alpha
- arylmethyl
- carboxy
- carboxyarylmethyl
- Prior art date
Links
- 229930182555 Penicillin Natural products 0.000 title 1
- NGHVIOIJCVXTGV-ALEPSDHESA-N 6-aminopenicillanic acid Chemical compound [O-]C(=O)[C@H]1C(C)(C)S[C@@H]2[C@H]([NH3+])C(=O)N21 NGHVIOIJCVXTGV-ALEPSDHESA-N 0.000 abstract 1
- NGHVIOIJCVXTGV-UHFFFAOYSA-N 6beta-amino-penicillanic acid Natural products OC(=O)C1C(C)(C)SC2C(N)C(=O)N21 NGHVIOIJCVXTGV-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 239000012442 inert solvent Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Abstract
Orally active alpha-carboxyarylmethyl-penicillins. N3A. Are prepared by treating 6-aminopenicillanic acid or a salt in an inert solvent with an arylmalonic acid ester. The reaction is carried out at temperatures between 0 and 50 degrees C at a pH 5 to 8.
[FR2017293A1]
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US75708768A | 1968-09-03 | 1968-09-03 | |
| US83051769A | 1969-06-04 | 1969-06-04 | |
| US83051669A | 1969-06-04 | 1969-06-04 | |
| US83051869A | 1969-06-04 | 1969-06-04 | |
| US83048169A | 1969-06-04 | 1969-06-04 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE34278L true IE34278L (en) | 1970-03-03 |
| IE34278B1 IE34278B1 (en) | 1975-04-02 |
Family
ID=27542173
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE1239/69A IE34278B1 (en) | 1968-09-03 | 1969-09-03 | Novel esters of alpha-carboxy arylmethylpenicillins and process therefor |
Country Status (5)
| Country | Link |
|---|---|
| BE (1) | BE738353A (en) |
| FR (1) | FR2017293A1 (en) |
| IE (1) | IE34278B1 (en) |
| IL (1) | IL32927A (en) |
| PH (1) | PH9984A (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE754141A (en) * | 1969-08-04 | 1971-02-01 | Pfizer | ALPHA-CARBOXYARYLMETHYL PENICILLINS ESTERS |
-
1969
- 1969-09-01 IL IL32927A patent/IL32927A/en unknown
- 1969-09-03 FR FR6929991A patent/FR2017293A1/en active Granted
- 1969-09-03 BE BE738353D patent/BE738353A/xx not_active IP Right Cessation
- 1969-09-03 PH PH10692A patent/PH9984A/en unknown
- 1969-09-03 IE IE1239/69A patent/IE34278B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BE738353A (en) | 1970-03-03 |
| IE34278B1 (en) | 1975-04-02 |
| DE1944379B2 (en) | 1977-02-24 |
| PH9984A (en) | 1976-07-13 |
| IL32927A0 (en) | 1969-11-30 |
| FR2017293A1 (en) | 1970-05-22 |
| IL32927A (en) | 1974-03-14 |
| FR2017293B1 (en) | 1974-08-09 |
| DE1944379A1 (en) | 1970-03-12 |
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