IE43841L - Triazolylbenzophenones - Google Patents
TriazolylbenzophenonesInfo
- Publication number
- IE43841L IE43841L IE762215A IE221576A IE43841L IE 43841 L IE43841 L IE 43841L IE 762215 A IE762215 A IE 762215A IE 221576 A IE221576 A IE 221576A IE 43841 L IE43841 L IE 43841L
- Authority
- IE
- Ireland
- Prior art keywords
- formula
- compounds
- triazolylbenzophenones
- gb1531980a
- spasmolytics
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000000935 antidepressant agent Substances 0.000 abstract 1
- 229940005513 antidepressants Drugs 0.000 abstract 1
- 239000002249 anxiolytic agent Substances 0.000 abstract 1
- 230000000949 anxiolytic effect Effects 0.000 abstract 1
- 229940005530 anxiolytics Drugs 0.000 abstract 1
- 238000006698 hydrazinolysis reaction Methods 0.000 abstract 1
- 239000003326 hypnotic agent Substances 0.000 abstract 1
- 230000000147 hypnotic effect Effects 0.000 abstract 1
- 229940035363 muscle relaxants Drugs 0.000 abstract 1
- 239000003158 myorelaxant agent Substances 0.000 abstract 1
- 125000001557 phthalyl group Chemical group C(=O)(O)C1=C(C(=O)*)C=CC=C1 0.000 abstract 1
- 239000000932 sedative agent Substances 0.000 abstract 1
- 229940125723 sedative agent Drugs 0.000 abstract 1
- 230000002048 spasmolytic effect Effects 0.000 abstract 1
- -1 spasmolytics Substances 0.000 abstract 1
- 239000007858 starting material Substances 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/92—Oxygen atoms with hetero atoms directly attached to nitrogen atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Anesthesiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
The compounds of the formula Ia in which the substituents have the meaning stated in Claim 1 are obtained by hydrazinolysis of phthalyl derivatives of the formula IV. The resulting products can be used as anxiolytics, sedatives, hypnotics, spasmolytics, muscle relaxants, antidepressants and can furthermore be employed as starting materials for the preparation of pharmacologically active compounds. <IMAGE>
[GB1531980A]
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB53224/75A GB1531980A (en) | 1975-12-30 | 1975-12-30 | Triazolylbenzophenone derivatives and preparation thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE43841L true IE43841L (en) | 1977-06-30 |
| IE43841B1 IE43841B1 (en) | 1981-06-03 |
Family
ID=10467048
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE2215/76A IE43841B1 (en) | 1975-12-30 | 1976-10-07 | Triazolylbenzophenone derivatives and preparation thereof |
Country Status (19)
| Country | Link |
|---|---|
| JP (1) | JPS5283469A (en) |
| AR (2) | AR218613A1 (en) |
| AT (1) | AT350052B (en) |
| AU (1) | AU498113B2 (en) |
| BE (1) | BE846410A (en) |
| CA (1) | CA1126274A (en) |
| CH (1) | CH623315A5 (en) |
| DE (1) | DE2641164A1 (en) |
| DK (1) | DK393576A (en) |
| ES (3) | ES451896A1 (en) |
| FR (1) | FR2336930A1 (en) |
| GB (1) | GB1531980A (en) |
| HU (1) | HU172539B (en) |
| IE (1) | IE43841B1 (en) |
| IL (1) | IL50664A (en) |
| NL (1) | NL7610799A (en) |
| NZ (1) | NZ181958A (en) |
| SE (1) | SE7609813L (en) |
| ZA (1) | ZA765851B (en) |
-
1975
- 1975-12-30 GB GB53224/75A patent/GB1531980A/en not_active Expired
-
1976
- 1976-08-31 DK DK393576A patent/DK393576A/en not_active Application Discontinuation
- 1976-09-02 CA CA260,438A patent/CA1126274A/en not_active Expired
- 1976-09-06 SE SE7609813A patent/SE7609813L/en not_active Application Discontinuation
- 1976-09-06 AU AU17498/76A patent/AU498113B2/en not_active Expired
- 1976-09-07 NZ NZ181958A patent/NZ181958A/en unknown
- 1976-09-08 HU HU76SI00001538A patent/HU172539B/en unknown
- 1976-09-13 DE DE19762641164 patent/DE2641164A1/en not_active Withdrawn
- 1976-09-15 AT AT684276A patent/AT350052B/en not_active IP Right Cessation
- 1976-09-17 AR AR264755A patent/AR218613A1/en active
- 1976-09-21 CH CH1193976A patent/CH623315A5/en not_active IP Right Cessation
- 1976-09-21 BE BE170796A patent/BE846410A/en unknown
- 1976-09-27 ES ES451896A patent/ES451896A1/en not_active Expired
- 1976-09-29 ZA ZA765851A patent/ZA765851B/en unknown
- 1976-09-29 NL NL7610799A patent/NL7610799A/en not_active Application Discontinuation
- 1976-10-06 FR FR7630125A patent/FR2336930A1/en active Granted
- 1976-10-06 JP JP12081576A patent/JPS5283469A/en active Pending
- 1976-10-07 IE IE2215/76A patent/IE43841B1/en unknown
- 1976-10-11 IL IL50664A patent/IL50664A/en unknown
-
1977
- 1977-06-30 AR AR268275A patent/AR220519A1/en active
- 1977-09-09 ES ES462244A patent/ES462244A1/en not_active Expired
- 1977-09-09 ES ES462243A patent/ES462243A1/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES462243A1 (en) | 1978-06-01 |
| JPS5283469A (en) | 1977-07-12 |
| DE2641164A1 (en) | 1977-07-14 |
| HU172539B (en) | 1978-09-28 |
| IE43841B1 (en) | 1981-06-03 |
| NZ181958A (en) | 1979-03-28 |
| AU498113B2 (en) | 1979-02-08 |
| IL50664A (en) | 1983-09-30 |
| NL7610799A (en) | 1977-07-04 |
| AU1749876A (en) | 1978-03-16 |
| SE7609813L (en) | 1977-07-01 |
| DK393576A (en) | 1977-07-01 |
| IL50664A0 (en) | 1976-12-31 |
| ZA765851B (en) | 1977-09-28 |
| CA1126274A (en) | 1982-06-22 |
| BE846410A (en) | 1977-01-17 |
| FR2336930A1 (en) | 1977-07-29 |
| AT350052B (en) | 1979-05-10 |
| ES462244A1 (en) | 1978-06-01 |
| FR2336930B1 (en) | 1978-12-22 |
| GB1531980A (en) | 1978-11-15 |
| ATA684276A (en) | 1978-10-15 |
| AR220519A1 (en) | 1980-11-14 |
| CH623315A5 (en) | 1981-05-29 |
| ES451896A1 (en) | 1978-01-16 |
| AR218613A1 (en) | 1980-06-30 |
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