IL140904A0 - Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors - Google Patents

Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors

Info

Publication number
IL140904A0
IL140904A0 IL14090401A IL14090401A IL140904A0 IL 140904 A0 IL140904 A0 IL 140904A0 IL 14090401 A IL14090401 A IL 14090401A IL 14090401 A IL14090401 A IL 14090401A IL 140904 A0 IL140904 A0 IL 140904A0
Authority
IL
Israel
Prior art keywords
methods
glycogen phosphorylase
treating diabetic
phosphorylase inhibitors
diabetic cardiomyopathy
Prior art date
Application number
IL14090401A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of IL140904A0 publication Critical patent/IL140904A0/xx

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL14090401A 2000-01-24 2001-01-15 Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors IL140904A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17777000P 2000-01-24 2000-01-24

Publications (1)

Publication Number Publication Date
IL140904A0 true IL140904A0 (en) 2002-02-10

Family

ID=22649922

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14090401A IL140904A0 (en) 2000-01-24 2001-01-15 Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors

Country Status (12)

Country Link
US (1) US6867184B2 (de)
EP (1) EP1125580A3 (de)
JP (1) JP2001206856A (de)
KR (1) KR20010083148A (de)
AU (1) AU1639901A (de)
CA (1) CA2331847A1 (de)
CO (1) CO5271699A1 (de)
HU (1) HUP0100321A3 (de)
IL (1) IL140904A0 (de)
NZ (1) NZ509481A (de)
PE (1) PE20011053A1 (de)
ZA (1) ZA200100607B (de)

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GB0205166D0 (en) 2002-03-06 2002-04-17 Astrazeneca Ab Chemical compounds
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GB0309154D0 (en) 2003-01-14 2003-05-28 Aventis Pharma Inc Use of insulin glargine to reduce or prevent cardiovascular events in patients being treated for dysglycemia
AU2004212004B2 (en) * 2003-02-13 2008-01-10 Albert Einstein College Of Medicine Of Yeshiva University Regulation of food intake and glucose production by modulation of long-chain fatty acyl-coa levels in the hypothalamus
WO2006041922A2 (en) * 2004-10-08 2006-04-20 Dara Biosciences, Inc. Agents and methods for administration to the central nervous system
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US7214704B2 (en) * 2004-11-15 2007-05-08 Bristol-Myers Squibb Company 2-Amino-1-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
US7226942B2 (en) 2004-11-15 2007-06-05 Bristol-Myers Squibb Company 2-amino-4-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
US7365061B2 (en) * 2004-11-15 2008-04-29 Bristol-Myers Squibb Company 2-Amino-3-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
WO2006088798A2 (en) * 2005-02-14 2006-08-24 Albert Einstein College Of Medicine Of Yeshiva University Modulation of hypothalamic atp-sensitive potassium channels
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
EP2069289B1 (de) * 2006-09-13 2013-10-02 Sanofi ISOSERINDERIVATE ALS INHIBITOREN DES KOAGULATIONSFAKTORS IXa
KR101481041B1 (ko) * 2007-11-30 2015-01-12 (주)아모레퍼시픽 글루코오스-6-인산 탈수소효소의 활성 억제제 및 이를포함하는 지방세포 분화 억제용 조성물
MX363056B (es) 2012-08-21 2019-03-06 Ardelyx Inc Compuestos y metodos para inhibir al antipuerto mediado por nhe en el tratamiento de trastornos asociados con la retencion de fluidos o la sobrecarga de sal y trastornos del tracto gastrointestinal.
KR102687458B1 (ko) * 2016-06-16 2024-07-24 호유 가부시키가이샤 생선 알레르기의 항원
IL275273B2 (en) 2017-12-15 2024-09-01 Medizinische Hochschule Hannover Improved compound for treatment of heart failure
CN113304149A (zh) * 2021-06-23 2021-08-27 广州医科大学 一种化合物在制备治疗2型糖尿病心肌病的药物中的应用
CN121591637B (zh) * 2025-11-28 2026-07-17 广州医科大学 5-(苄基氨基甲酰基)-吲哚类化合物及其在制备防治糖尿病心肌病药物中的应用

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JP2001206856A (ja) 2001-07-31
AU1639901A (en) 2001-07-26
PE20011053A1 (es) 2001-10-17
KR20010083148A (ko) 2001-08-31
HUP0100321A3 (en) 2004-03-01
ZA200100607B (en) 2002-07-22
HUP0100321A2 (en) 2002-10-28
CO5271699A1 (es) 2003-04-30
CA2331847A1 (en) 2001-07-24
US20010046958A1 (en) 2001-11-29
US6867184B2 (en) 2005-03-15
HU0100321D0 (en) 2001-03-28
EP1125580A2 (de) 2001-08-22

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