IL157243A0 - Preparation of n-methylparoxetine and related intermediate compounds - Google Patents
Preparation of n-methylparoxetine and related intermediate compoundsInfo
- Publication number
- IL157243A0 IL157243A0 IL15724302A IL15724302A IL157243A0 IL 157243 A0 IL157243 A0 IL 157243A0 IL 15724302 A IL15724302 A IL 15724302A IL 15724302 A IL15724302 A IL 15724302A IL 157243 A0 IL157243 A0 IL 157243A0
- Authority
- IL
- Israel
- Prior art keywords
- methylparoxetine
- preparation
- intermediate compounds
- related intermediate
- compounds
- Prior art date
Links
- MOJZPKOBKCXNKG-YJBOKZPZSA-N N-methylparoxetine Chemical compound C1([C@@H]2CCN(C[C@H]2COC=2C=C3OCOC3=CC=2)C)=CC=C(F)C=C1 MOJZPKOBKCXNKG-YJBOKZPZSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
- C07D317/64—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26649801P | 2001-02-05 | 2001-02-05 | |
| US27758701P | 2001-03-21 | 2001-03-21 | |
| PCT/US2002/003223 WO2002062790A1 (en) | 2001-02-05 | 2002-02-04 | Preparation of n-methylparoxetine and related intermediate compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL157243A0 true IL157243A0 (en) | 2004-02-19 |
Family
ID=26951885
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL15724302A IL157243A0 (en) | 2001-02-05 | 2002-02-04 | Preparation of n-methylparoxetine and related intermediate compounds |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US6777554B2 (cs) |
| EP (1) | EP1366041A4 (cs) |
| KR (1) | KR20040014452A (cs) |
| CA (1) | CA2437392A1 (cs) |
| CZ (1) | CZ20032354A3 (cs) |
| HR (1) | HRP20030690A2 (cs) |
| HU (1) | HUP0303153A2 (cs) |
| IL (1) | IL157243A0 (cs) |
| SK (1) | SK10992003A3 (cs) |
| WO (1) | WO2002062790A1 (cs) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002006275A1 (en) * | 2000-07-17 | 2002-01-24 | Smithkline Beecham P.L.C. | Novel processes for the preparation of 4-phenylpiperidine derivatives |
| US20080029575A1 (en) * | 2006-08-02 | 2008-02-07 | Shelton Frederick E | Surgical cutting and fastening instrument with distally mounted pneumatically powered rotary drive member |
| US9138430B2 (en) * | 2007-12-27 | 2015-09-22 | Mylan Specialty L.P. | Formulation and method for the release of paroxetine in the large intestine |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1422263A (en) | 1973-01-30 | 1976-01-21 | Ferrosan As | 4-phenyl-piperidine compounds |
| US4585777A (en) | 1984-02-07 | 1986-04-29 | A/S Ferrosan | (-)-Trans-4-(4-fluorophenyl)-3-(4-methoxyphenoxy)methylpiperidine for potentiating 5-HT |
| DE3680184D1 (de) | 1985-08-10 | 1991-08-14 | Beecham Group Plc | Verfahren zur herstellung von arylpiperidincarbinol. |
| IE66332B1 (en) | 1986-11-03 | 1995-12-27 | Novo Nordisk As | Piperidine compounds and their preparation and use |
| GB8714707D0 (en) | 1987-06-23 | 1987-07-29 | Beecham Group Plc | Chemical process |
| FR2634207B1 (fr) | 1988-07-12 | 1990-09-07 | Synthelabo | Derives de ((piperidinyl-4)methyl) benzazepines, leur preparation et leur application en therapeutique |
| EP0351283A1 (fr) | 1988-07-12 | 1990-01-17 | Synthelabo | Dérivés de [(pipéridinyl-4) méthyl]-2 dihydro-2,3 1H-isoindole et tétrahydro-2,3,4,5 1H-benzazépines, leur préparation et leur application en thérapeutique |
| FR2659323B1 (fr) | 1990-03-07 | 1992-06-12 | Synthelabo | Derives de 4-(aminomethyl) piperidine, leur preparation et leur application en therapeutique. |
| US5258517A (en) | 1992-08-06 | 1993-11-02 | Sepracor, Inc. | Method of preparing optically pure precursors of paroxetine |
| US6004990A (en) | 1994-06-03 | 1999-12-21 | Zebra Pharmaceuticals | Meta substituted arylalkylamines and therapeutic and diagnostic uses therefor |
| GB9526645D0 (en) | 1995-12-28 | 1996-02-28 | Chiroscience Ltd | Stereoselective synthesis |
| JP3882224B2 (ja) | 1996-05-31 | 2007-02-14 | 旭硝子株式会社 | パロキセチンの製造方法 |
| EP0812827B1 (en) | 1996-06-13 | 2009-09-02 | Sumitomo Chemical Company, Limited | Piperidine derivative as intermediates for the preparation of paroxetine and process for their preparation |
| HU221921B1 (hu) | 1996-07-08 | 2003-02-28 | Richter Gedeon Vegyészeti Gyár Rt. | N-benzil-piperidin- és tetrahidropiridinszármazékok és eljárás azok előállítására |
| GB9710004D0 (en) | 1997-05-17 | 1997-07-09 | Knoll Ag | Chemical process |
| WO2002006275A1 (en) | 2000-07-17 | 2002-01-24 | Smithkline Beecham P.L.C. | Novel processes for the preparation of 4-phenylpiperidine derivatives |
| IL159280A0 (en) * | 2001-06-14 | 2004-06-01 | Teva Pharma | A process for preparing paroxetine hcl which limits formation of pink colored compounds |
| CN1336363A (zh) * | 2001-07-25 | 2002-02-20 | 张元宾 | 乙酰磺胺酸钾的合成制备方法 |
| NZ532432A (en) | 2001-10-22 | 2005-02-25 | Synthon Bv | N-formyl paroxetine compounds and their use in a synthetic route for obtaining paroxetine |
-
2002
- 2002-02-02 US US10/067,160 patent/US6777554B2/en not_active Expired - Fee Related
- 2002-02-04 CZ CZ20032354A patent/CZ20032354A3/cs unknown
- 2002-02-04 CA CA002437392A patent/CA2437392A1/en not_active Abandoned
- 2002-02-04 IL IL15724302A patent/IL157243A0/xx unknown
- 2002-02-04 HR HR20030690A patent/HRP20030690A2/hr not_active Application Discontinuation
- 2002-02-04 SK SK1099-2003A patent/SK10992003A3/sk unknown
- 2002-02-04 EP EP02702143A patent/EP1366041A4/en not_active Withdrawn
- 2002-02-04 KR KR10-2003-7010266A patent/KR20040014452A/ko not_active Abandoned
- 2002-02-04 HU HU0303153A patent/HUP0303153A2/hu unknown
- 2002-02-04 WO PCT/US2002/003223 patent/WO2002062790A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| CA2437392A1 (en) | 2002-08-15 |
| CZ20032354A3 (cs) | 2004-08-18 |
| EP1366041A1 (en) | 2003-12-03 |
| SK10992003A3 (sk) | 2004-03-02 |
| KR20040014452A (ko) | 2004-02-14 |
| HRP20030690A2 (en) | 2005-04-30 |
| WO2002062790A1 (en) | 2002-08-15 |
| US6777554B2 (en) | 2004-08-17 |
| EP1366041A4 (en) | 2004-12-22 |
| US20020151567A1 (en) | 2002-10-17 |
| HUP0303153A2 (hu) | 2004-03-01 |
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