IL161444A0 - A process for the preparation of the 14beta-hydroxy-baccatin iii-1,14-carbonate - Google Patents

A process for the preparation of the 14beta-hydroxy-baccatin iii-1,14-carbonate

Info

Publication number: IL161444A0
Authority: IL; Israel
Prior art keywords: preparation; 14beta; hydroxy; carbonate; baccatin iii
Prior art date: 2001-10-19

Application number

IL16144402A

Other languages

English (en)

Original Assignee

Indena Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-10-19

Filing date

2002-07-18

Publication date

2004-09-27

2002-07-18 Application filed by Indena Spa filed Critical Indena Spa

2004-09-27 Publication of IL161444A0 publication Critical patent/IL161444A0/xx

Links

238000000034 method Methods 0.000 title abstract 2
230000000259 anti-tumor effect Effects 0.000 abstract 1
DKPFODGZWDEEBT-QFIAKTPHSA-N taxane Chemical class C([C@]1(C)CCC[C@@H](C)[C@H]1C1)C[C@H]2[C@H](C)CC[C@@H]1C2(C)C DKPFODGZWDEEBT-QFIAKTPHSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/08—Bridged systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Epoxy Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Peptides Or Proteins (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

IL16144402A 2001-10-19 2002-07-18 A process for the preparation of the 14beta-hydroxy-baccatin iii-1,14-carbonate IL161444A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IT2001MI002185A ITMI20012185A1 (it)	2001-10-19	2001-10-19	Procedimento per la preparazione della 14beta-idrossi-baccatina iii-1,14-carbonato
PCT/EP2002/008007 WO2003035634A1 (fr)	2001-10-19	2002-07-18	Procede de preparation de 14beta-hydroxy-baccatin iii-1,14-carbonate

Publications (1)

Publication Number	Publication Date
IL161444A0 true IL161444A0 (en)	2004-09-27

Family

ID=11448528

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
IL16144402A IL161444A0 (en)	2001-10-19	2002-07-18	A process for the preparation of the 14beta-hydroxy-baccatin iii-1,14-carbonate
IL161444A IL161444A (en)	2001-10-19	2004-04-15	Process for the preparation of the 14 beta-hydroxy-baccatin iii-1, 14-carbonate
IL185921A IL185921A (en)	2001-10-19	2007-09-11	Intermediate compound for the preparation of the 14 beta-hydroxy-baccatin iii -1,14-carbonate
IL185920A IL185920A (en)	2001-10-19	2007-09-11	14 beta-hydroxy-7- boc-13- keto- baccatin iii- 1, 14-carbonate

Family Applications After (3)

Application Number	Title	Priority Date	Filing Date
IL161444A IL161444A (en)	2001-10-19	2004-04-15	Process for the preparation of the 14 beta-hydroxy-baccatin iii-1, 14-carbonate
IL185921A IL185921A (en)	2001-10-19	2007-09-11	Intermediate compound for the preparation of the 14 beta-hydroxy-baccatin iii -1,14-carbonate
IL185920A IL185920A (en)	2001-10-19	2007-09-11	14 beta-hydroxy-7- boc-13- keto- baccatin iii- 1, 14-carbonate

Country Status (22)

Country	Link
US (1)	US7317113B2 (fr)
EP (1)	EP1436278B1 (fr)
JP (2)	JP4467976B2 (fr)
KR (1)	KR100896543B1 (fr)
CN (1)	CN100338049C (fr)
AT (1)	ATE466847T1 (fr)
AU (1)	AU2002363080B2 (fr)
BR (1)	BR0213329A (fr)
CA (1)	CA2464336C (fr)
DE (1)	DE60236303D1 (fr)
DK (1)	DK1436278T3 (fr)
ES (1)	ES2341611T3 (fr)
HU (1)	HU229256B1 (fr)
IL (4)	IL161444A0 (fr)
IT (1)	ITMI20012185A1 (fr)
MX (1)	MXPA04003517A (fr)
NO (1)	NO328534B1 (fr)
PL (1)	PL207878B1 (fr)
PT (1)	PT1436278E (fr)
RU (1)	RU2285000C2 (fr)
SI (1)	SI1436278T1 (fr)
WO (1)	WO2003035634A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ITMI20012185A1 (it) *	2001-10-19	2003-04-19	Indena Spa	Procedimento per la preparazione della 14beta-idrossi-baccatina iii-1,14-carbonato
ITMI20012186A1 (it) *	2001-10-19	2003-04-19	Indena Spa	Procedimento per la preparazione della 14-beta-idrossi-baccatina iii-1,14-carbonato
WO2004025826A1 (fr) *	2002-09-16	2004-03-25	Nokia Corporation	Recepteur a conversion directe et procede de reception
ES2389518T3 (es)	2008-01-18	2012-10-26	Indena S.P.A.	Formas sólidas de ortataxel

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH0620877A (ja) *	1992-03-02	1994-01-28	Du Pont Japan Ltd	タンタル固体電解コンデンサ
IT1254517B (it)	1992-03-06	1995-09-25	Indena Spa	14-beta idrossi-10-deacetil-baccatina iii, suoi derivati, loro prepazione ed impiego terapeutico
US5475011A (en) *	1993-03-26	1995-12-12	The Research Foundation Of State University Of New York	Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment
FR2718137B1 (fr) *	1994-04-05	1996-04-26	Rhone Poulenc Rorer Sa	Procédé de préparation de trialcoylsilyl-7 baccatine III.
IT1275936B1 (it) *	1995-03-17	1997-10-24	Indena Spa	Derivati della 10-deacetilbaccatina iii e della 10-deacetil-14b- idrossibaccatina iii loro metodo di preparazione e formulazioni
FR2732341A1 (fr)	1995-03-27	1996-10-04	Rhone Poulenc Rorer Sa	Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
IT1275435B (it)	1995-05-19	1997-08-07	Indena Spa	Derivati della 10-desacetil-14beta-idrossibaccatina iii,loro metodo di preparazione e formulazioni che li contengono
IT1283633B1 (it) *	1996-05-10	1998-04-23	Indena Spa	Derivati tassanici loro sintesi e formulazioni che li contengono
US5811452A (en) *	1997-01-08	1998-09-22	The Research Foundation Of State University Of New York	Taxoid reversal agents for drug-resistance in cancer chemotherapy and pharmaceutical compositions thereof
US5917062A (en) *	1997-11-21	1999-06-29	Indena S.P.A	Intermediates and methods useful in the semisynthesis of paclitaxel and analogs
IT1318678B1 (it) *	2000-08-10	2003-08-27	Indena Spa	Procedimento per la preparazione di derivati della baccatina iii.
IT1320107B1 (it) *	2000-11-28	2003-11-18	Indena Spa	Procedimento per la preparazione di derivati tassanici.
IT1319682B1 (it) *	2000-12-06	2003-10-23	Indena Spa	Procedimento di sintesi del paclitaxel.
ITMI20012186A1 (it) *	2001-10-19	2003-04-19	Indena Spa	Procedimento per la preparazione della 14-beta-idrossi-baccatina iii-1,14-carbonato
ITMI20012185A1 (it) *	2001-10-19	2003-04-19	Indena Spa	Procedimento per la preparazione della 14beta-idrossi-baccatina iii-1,14-carbonato
ITMI20021921A1 (it) *	2002-09-10	2004-03-11	Indena Spa	Funzionalizzazione della posizione 14 dei nuclei tassanici e sintesi di nuovi derivati antitumorali.

2001
- 2001-10-19 IT IT2001MI002185A patent/ITMI20012185A1/it unknown
2002
- 2002-07-15 US US10/492,589 patent/US7317113B2/en not_active Expired - Lifetime
- 2002-07-18 EP EP02801856A patent/EP1436278B1/fr not_active Expired - Lifetime
- 2002-07-18 AU AU2002363080A patent/AU2002363080B2/en not_active Ceased
- 2002-07-18 PT PT02801856T patent/PT1436278E/pt unknown
- 2002-07-18 JP JP2003538150A patent/JP4467976B2/ja not_active Expired - Fee Related
- 2002-07-18 RU RU2004111670/04A patent/RU2285000C2/ru active
- 2002-07-18 PL PL367981A patent/PL207878B1/pl unknown
- 2002-07-18 SI SI200230907T patent/SI1436278T1/sl unknown
- 2002-07-18 CN CNB028205235A patent/CN100338049C/zh not_active Expired - Fee Related
- 2002-07-18 DE DE60236303T patent/DE60236303D1/de not_active Expired - Lifetime
- 2002-07-18 HU HU0402020A patent/HU229256B1/hu not_active IP Right Cessation
- 2002-07-18 BR BR0213329-6A patent/BR0213329A/pt not_active IP Right Cessation
- 2002-07-18 WO PCT/EP2002/008007 patent/WO2003035634A1/fr not_active Ceased
- 2002-07-18 ES ES02801856T patent/ES2341611T3/es not_active Expired - Lifetime
- 2002-07-18 CA CA002464336A patent/CA2464336C/fr not_active Expired - Lifetime
- 2002-07-18 DK DK02801856.2T patent/DK1436278T3/da active
- 2002-07-18 MX MXPA04003517A patent/MXPA04003517A/es active IP Right Grant
- 2002-07-18 IL IL16144402A patent/IL161444A0/xx unknown
- 2002-07-18 AT AT02801856T patent/ATE466847T1/de active
- 2002-07-18 KR KR1020047004622A patent/KR100896543B1/ko not_active Expired - Fee Related
2004
- 2004-04-15 NO NO20041542A patent/NO328534B1/no not_active IP Right Cessation
- 2004-04-15 IL IL161444A patent/IL161444A/en active IP Right Grant
2007
- 2007-09-11 IL IL185921A patent/IL185921A/en active IP Right Grant
- 2007-09-11 IL IL185920A patent/IL185920A/en active IP Right Grant
2009
- 2009-10-23 JP JP2009244284A patent/JP2010047600A/ja active Pending

Also Published As

Publication number	Publication date
ES2341611T3 (es)	2010-06-23
NO20041542L (no)	2004-04-15
SI1436278T1 (sl)	2010-08-31
NO328534B1 (no)	2010-03-15
JP2010047600A (ja)	2010-03-04
IL185920A0 (en)	2008-01-06
BR0213329A (pt)	2004-10-13
HK1080475A1 (en)	2006-04-28
IL185921A0 (en)	2008-01-06
IL185921A (en)	2011-06-30
HU229256B1 (hu)	2013-10-28
KR100896543B1 (ko)	2009-05-07
US20050020669A1 (en)	2005-01-27
EP1436278B1 (fr)	2010-05-05
US7317113B2 (en)	2008-01-08
CA2464336A1 (fr)	2003-05-01
CN100338049C (zh)	2007-09-19
PT1436278E (pt)	2010-05-31
ITMI20012185A1 (it)	2003-04-19
AU2002363080B2 (en)	2007-11-29
PL367981A1 (en)	2005-03-21
IL161444A (en)	2008-12-29
IL185920A (en)	2011-02-28
WO2003035634A1 (fr)	2003-05-01
WO2003035634A8 (fr)	2004-05-21
JP2005509638A (ja)	2005-04-14
DK1436278T3 (da)	2010-08-02
RU2004111670A (ru)	2005-04-20
CA2464336C (fr)	2009-12-22
DE60236303D1 (de)	2010-06-17
ATE466847T1 (de)	2010-05-15
KR20040045024A (ko)	2004-05-31
MXPA04003517A (es)	2004-07-23
PL207878B1 (pl)	2011-02-28
HUP0402020A2 (hu)	2005-01-28
CN1688563A (zh)	2005-10-26
JP4467976B2 (ja)	2010-05-26
HUP0402020A3 (en)	2007-05-29
RU2285000C2 (ru)	2006-10-10
EP1436278A1 (fr)	2004-07-14

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