IL165355A0 - Synthesis of diaryl pyrazoles - Google Patents

Synthesis of diaryl pyrazoles

Info

Publication number
IL165355A0
IL165355A0 IL16535503A IL16535503A IL165355A0 IL 165355 A0 IL165355 A0 IL 165355A0 IL 16535503 A IL16535503 A IL 16535503A IL 16535503 A IL16535503 A IL 16535503A IL 165355 A0 IL165355 A0 IL 165355A0
Authority
IL
Israel
Prior art keywords
synthesis
diaryl pyrazoles
pyrazoles
diaryl
Prior art date
Application number
IL16535503A
Other languages
English (en)
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of IL165355A0 publication Critical patent/IL165355A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IL16535503A 2002-05-24 2003-05-23 Synthesis of diaryl pyrazoles IL165355A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38300702P 2002-05-24 2002-05-24
PCT/US2003/016404 WO2003099794A1 (fr) 2002-05-24 2003-05-23 Synthese de diarylpyrazoles

Publications (1)

Publication Number Publication Date
IL165355A0 true IL165355A0 (en) 2006-01-15

Family

ID=29584488

Family Applications (2)

Application Number Title Priority Date Filing Date
IL16535503A IL165355A0 (en) 2002-05-24 2003-05-23 Synthesis of diaryl pyrazoles
IL165355A IL165355A (en) 2002-05-24 2004-11-23 Synthesis of diaryl pyrazoles

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL165355A IL165355A (en) 2002-05-24 2004-11-23 Synthesis of diaryl pyrazoles

Country Status (14)

Country Link
US (2) US7141678B2 (fr)
EP (1) EP1507766A4 (fr)
JP (1) JP2005532333A (fr)
KR (1) KR20050013553A (fr)
CN (1) CN100348586C (fr)
AU (1) AU2003241603B2 (fr)
BR (1) BR0311267A (fr)
CA (1) CA2487401A1 (fr)
IL (2) IL165355A0 (fr)
MX (1) MXPA04011654A (fr)
PL (1) PL373807A1 (fr)
RU (1) RU2319695C2 (fr)
WO (1) WO2003099794A1 (fr)
ZA (1) ZA200409434B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA04011654A (es) * 2002-05-24 2005-03-07 Pharmacia Corp Sintesis de diarilpirazoles.
CN1279789C (zh) 2004-08-05 2006-10-11 华为技术有限公司 在一个物理移动交换中心覆盖的多子网间实现通信的方法
US7919633B2 (en) * 2007-03-19 2011-04-05 Dr. Reddy's Laboratories Limited Process for preparation of celecoxib
KR101005834B1 (ko) * 2008-08-04 2011-01-05 이화여자대학교 산학협력단 피라졸의 제조방법
WO2010095024A2 (fr) 2009-02-20 2010-08-26 Aurobindo Pharma Limited Procédé amélioré de préparation de célécoxib
CN102746231A (zh) * 2011-04-20 2012-10-24 天津药物研究院 塞来昔布制备工艺
CN102558057B (zh) * 2012-01-16 2014-04-02 兰州大学 多取代吡唑制备方法
CN103242233B (zh) * 2012-02-08 2014-07-30 北京博爱汇康医药科技有限责任公司 制备塞来昔布的新方法
CN102617473A (zh) * 2012-03-13 2012-08-01 扬州天和药业有限公司 马氟考昔的一种制备方法
CN103044329B (zh) * 2013-01-10 2015-03-25 齐河诚汇精细化工有限公司 一种高收率高纯度塞来昔布的制备方法
CN103923011A (zh) * 2014-05-04 2014-07-16 苏州天马精细化学品股份有限公司 一种塞来西布的合成方法
CN103951549B (zh) * 2014-05-20 2016-04-27 河北科技大学 一种cox-2酶抑制剂塞来昔布中间体的合成方法
CN104177294A (zh) * 2014-08-27 2014-12-03 齐鲁天和惠世制药有限公司 一种塞来昔布的制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH27357A (en) 1989-09-22 1993-06-21 Fujisawa Pharmaceutical Co Pyrazole derivatives and pharmaceutical compositions comprising the same
IL104311A (en) 1992-02-05 1997-07-13 Fujisawa Pharmaceutical Co Pyrazole derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
US5466823A (en) * 1993-11-30 1995-11-14 G.D. Searle & Co. Substituted pyrazolyl benzenesulfonamides
DE69422306T4 (de) * 1993-11-30 2000-09-07 G.D. Searle & Co., Chicago Substituierte pyrazolyl-benzolsulfonamide zur behandlung von entzündungen
EP0828717B1 (fr) * 1995-05-25 2002-09-04 G.D. SEARLE & CO. Procede de preparation de 3-haloalkyl-1h-pyrazoles
US5643933A (en) * 1995-06-02 1997-07-01 G. D. Searle & Co. Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors
JP2002534509A (ja) * 1999-01-14 2002-10-15 メルク フロスト カナダ アンド カンパニー ４−［（５−置換または未置換フェニル）−３−置換−１ｈ−ピラゾール−１−イル］ベンゼンスルホンアミド類の合成
AU4308300A (en) * 1999-05-03 2000-11-17 Dr. Reddy's Research Foundation Pyrazoles having antiinflammatory activity
CA2326970C (fr) * 1999-12-03 2004-11-23 Pfizer Products Inc. Derives d'acetylene en tant qu'agents anti-inflammatoires et analgesiques
TR200001872A3 (tr) * 2000-06-26 2002-01-21 Fako Ilaclari A.S 4-[5-(4-Metilfenil-3-(triflorometil)-1H-pirazol-1-il] benzensulfonamit' in yeni kristal biçimi "Biçim I" ve bu ürünün üretilmesine iliskin yöntem.
MXPA04011654A (es) * 2002-05-24 2005-03-07 Pharmacia Corp Sintesis de diarilpirazoles.

Also Published As

Publication number Publication date
BR0311267A (pt) 2005-05-10
AU2003241603A1 (en) 2003-12-12
CN100348586C (zh) 2007-11-14
AU2003241603B2 (en) 2008-05-15
CA2487401A1 (fr) 2003-12-04
RU2004137819A (ru) 2005-07-20
WO2003099794A1 (fr) 2003-12-04
US7759497B2 (en) 2010-07-20
RU2319695C2 (ru) 2008-03-20
IL165355A (en) 2009-07-20
US20070004924A1 (en) 2007-01-04
ZA200409434B (en) 2006-10-25
EP1507766A1 (fr) 2005-02-23
MXPA04011654A (es) 2005-03-07
HK1079197A1 (en) 2006-03-31
US7141678B2 (en) 2006-11-28
CN1671669A (zh) 2005-09-21
PL373807A1 (en) 2005-09-19
EP1507766A4 (fr) 2006-06-14
US20040024225A1 (en) 2004-02-05
KR20050013553A (ko) 2005-02-04
JP2005532333A (ja) 2005-10-27

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