IL238461A0 - 1 hindole-3-carboxamide derivatives and their use as p2y12 inhibitors - Google Patents

1 hindole-3-carboxamide derivatives and their use as p2y12 inhibitors

Info

Publication number
IL238461A0
IL238461A0 IL238461A IL23846115A IL238461A0 IL 238461 A0 IL238461 A0 IL 238461A0 IL 238461 A IL238461 A IL 238461A IL 23846115 A IL23846115 A IL 23846115A IL 238461 A0 IL238461 A0 IL 238461A0
Authority
IL
Israel
Prior art keywords
indole
antagonists
carboxamide derivatives
carboxamide
derivatives
Prior art date
Application number
IL238461A
Other languages
English (en)
Hebrew (he)
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of IL238461A0 publication Critical patent/IL238461A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epidemiology (AREA)
  • Indole Compounds (AREA)
IL238461A 2012-10-26 2015-04-26 1 hindole-3-carboxamide derivatives and their use as p2y12 inhibitors IL238461A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12306334.9A EP2725025A1 (de) 2012-10-26 2012-10-26 Derivate von 1H-Indol-3-Carboxamid und ihre Verwendung als P2Y12 Antogonisten.
PCT/EP2013/072322 WO2014064219A1 (fr) 2012-10-26 2013-10-24 Derives de 1 h-indole-3-carboxamide et leurs utilisation comme antagonistes du p2y12

Publications (1)

Publication Number Publication Date
IL238461A0 true IL238461A0 (en) 2015-06-30

Family

ID=47146304

Family Applications (1)

Application Number Title Priority Date Filing Date
IL238461A IL238461A0 (en) 2012-10-26 2015-04-26 1 hindole-3-carboxamide derivatives and their use as p2y12 inhibitors

Country Status (14)

Country Link
US (1) US20150274703A1 (de)
EP (2) EP2725025A1 (de)
JP (1) JP6235029B2 (de)
KR (1) KR20150074131A (de)
CN (1) CN104936950B (de)
AU (1) AU2013336628A1 (de)
BR (1) BR112015009136A2 (de)
CA (1) CA2889538A1 (de)
ES (1) ES2608787T3 (de)
IL (1) IL238461A0 (de)
MX (1) MX2015005312A (de)
RU (1) RU2015119642A (de)
SG (1) SG11201503221PA (de)
WO (1) WO2014064219A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10167257B2 (en) 2014-04-04 2019-01-01 Iomet Pharma Ltd. Indole derivatives for use in medicine
US10858319B2 (en) 2016-10-03 2020-12-08 Iomet Pharma Ltd. Indole derivatives for use in medicine
MY202326A (en) 2017-09-14 2024-04-24 Daiichi Sankyo Co Ltd Compound having cyclic structure

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7470712B2 (en) * 2004-01-21 2008-12-30 Bristol-Myers Squibb Company Amino-benzazoles as P2Y1 receptor inhibitors
DE602006017694D1 (de) * 2005-06-27 2010-12-02 Bristol Myers Squibb Co C-verknüpfte zyklische antagonisten des p2y1-rezeptors mit eignung bei der behandlung thrombotischer leiden
MX2009011089A (es) * 2007-04-23 2009-10-30 Sanofi Aventis Derivados de quinolina-carboxamida en calidad de antagonistas de p2y12.
EP2238127B1 (de) * 2007-12-26 2012-08-15 Sanofi Pyrazolcarboxamid-derivate als p2y12-antagonisten
FR2974576B1 (fr) * 2011-04-29 2013-07-19 Sanofi Aventis Derives de n-[(1h-pyrazol-1-yl)aryl]-1h-indole ou 1h- indazole-3-carboxamide, leur preparation et leurs applications en therapeutique

Also Published As

Publication number Publication date
WO2014064219A1 (fr) 2014-05-01
RU2015119642A (ru) 2016-12-20
CN104936950B (zh) 2017-08-08
AU2013336628A1 (en) 2015-05-21
MX2015005312A (es) 2015-11-16
EP2917204B1 (de) 2016-09-28
ES2608787T3 (es) 2017-04-17
KR20150074131A (ko) 2015-07-01
CA2889538A1 (en) 2014-05-01
JP2015535230A (ja) 2015-12-10
JP6235029B2 (ja) 2017-11-22
SG11201503221PA (en) 2015-06-29
EP2725025A1 (de) 2014-04-30
EP2917204A1 (de) 2015-09-16
CN104936950A (zh) 2015-09-23
BR112015009136A2 (pt) 2017-07-04
US20150274703A1 (en) 2015-10-01

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