IL50938A - 2-(9-substituted alkyl-6-purin-yl-amino)-and 2-(1-substituted alkyl-pyrazolo (3,4-d)pyrimidin-4-yl-amino)benzoic acid derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

2-(9-substituted alkyl-6-purin-yl-amino)-and 2-(1-substituted alkyl-pyrazolo (3,4-d)pyrimidin-4-yl-amino)benzoic acid derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number: IL50938A
Authority: IL; Israel
Prior art keywords: amino; substituted alkyl; purin; pyrazolo; pyrimidin
Prior art date: 1975-11-19

Application number

IL50938A

Other languages

English (en)

Original Assignee

Medicale Rech France

Science Union & Cie

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1975-11-19

Filing date

1976-11-18

Publication date

1980-06-30

1976-11-18 Application filed by Medicale Rech France, Science Union & Cie filed Critical Medicale Rech France

1980-06-30 Publication of IL50938A publication Critical patent/IL50938A/xx

Links

150000001558 benzoic acid derivatives Chemical class 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heat Sensitive Colour Forming Recording (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

IL50938A 1975-11-19 1976-11-18 2-(9-substituted alkyl-6-purin-yl-amino)-and 2-(1-substituted alkyl-pyrazolo (3,4-d)pyrimidin-4-yl-amino)benzoic acid derivatives,their preparation and pharmaceutical compositions containing them IL50938A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB47618/75A GB1544419A (en)	1975-11-19	1975-11-19	Purines and pyrazolo-pyrimidines a process for their preparation and pharmaceutical compositions containing them

Publications (1)

Publication Number	Publication Date
IL50938A true IL50938A (en)	1980-06-30

Family

ID=10445643

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL50938A IL50938A (en)	1975-11-19	1976-11-18	2-(9-substituted alkyl-6-purin-yl-amino)-and 2-(1-substituted alkyl-pyrazolo (3,4-d)pyrimidin-4-yl-amino)benzoic acid derivatives,their preparation and pharmaceutical compositions containing them

Country Status (21)

Country	Link
US (1)	US4100286A (fr)
JP (1)	JPS5265296A (fr)
AR (1)	AR214186A1 (fr)
AU (1)	AU508926B2 (fr)
BE (1)	BE848505A (fr)
CA (1)	CA1083148A (fr)
CH (1)	CH596210A5 (fr)
DE (1)	DE2651789C2 (fr)
ES (1)	ES453460A1 (fr)
FR (1)	FR2332020A1 (fr)
GB (1)	GB1544419A (fr)
GR (1)	GR61601B (fr)
IE (1)	IE44078B1 (fr)
IL (1)	IL50938A (fr)
MX (1)	MX3904E (fr)
NL (1)	NL7612894A (fr)
NZ (1)	NZ182681A (fr)
OA (1)	OA05485A (fr)
PH (1)	PH11898A (fr)
PT (1)	PT65859B (fr)
ZA (1)	ZA766923B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3131365A1 (de) *	1981-08-07	1983-02-24	Henkel KGaA, 4000 Düsseldorf	Neue diglycidyl-substituierte heterocyclische verbindungen, verfahren zu ihrer herstellung und ihre verwendung in arzneimittelzubereitungen mit cytostatischer wirksamkeit
US6057305A (en)	1992-08-05	2000-05-02	Institute Of Organic Chemistry And Biochemistry Of The Academy Of Sciences Of The Czech Republic	Antiretroviral enantiomeric nucleotide analogs
FR2699176B1 (fr) *	1992-12-11	1995-03-03	Adir	Nouveaux composés bicycliques de pyrimidine, leur procédé de préparation et les compositions pharmaceutiques les renfermant.
US6110923A (en) *	1994-06-22	2000-08-29	Biochem Pharma Inc.	Method for treating cancer using novel substituted purinyl derivatives with immunomodulating activity
FR2741881B1 (fr) *	1995-12-01	1999-07-30	Centre Nat Rech Scient	Nouveaux derives de purine possedant notamment des prorietes anti-proliferatives et leurs applications biologiques
US6107300A (en) *	1996-03-27	2000-08-22	Dupont Pharmaceuticals	Arylamino fused pyrimidines
TW200400034A (en) *	2002-05-20	2004-01-01	Bristol Myers Squibb Co	Pyrazolo-pyrimidine aniline compounds useful as kinase inhibitors
TWI638814B (zh) *	2012-10-31	2018-10-21	富山化學工業股份有限公司	新穎之胺衍生物或其鹽

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3551428A (en) *	1956-02-10	1970-12-29	Ciba Geigy Corp	New 1- (or 2-) substituted 4-mercapto-pyrazolo(3,4-d)pyrimidines

1975
- 1975-11-19 GB GB47618/75A patent/GB1544419A/en not_active Expired
1976
- 1976-11-12 IE IE2499/76A patent/IE44078B1/en unknown
- 1976-11-12 DE DE2651789A patent/DE2651789C2/de not_active Expired
- 1976-11-15 US US05/741,740 patent/US4100286A/en not_active Expired - Lifetime
- 1976-11-17 GR GR52204A patent/GR61601B/el unknown
- 1976-11-17 FR FR7634552A patent/FR2332020A1/fr active Granted
- 1976-11-18 AR AR265520A patent/AR214186A1/es active
- 1976-11-18 JP JP51139012A patent/JPS5265296A/ja active Granted
- 1976-11-18 ES ES453460A patent/ES453460A1/es not_active Expired
- 1976-11-18 BE BE172495A patent/BE848505A/fr unknown
- 1976-11-18 PT PT65859A patent/PT65859B/pt unknown
- 1976-11-18 AU AU19757/76A patent/AU508926B2/en not_active Expired
- 1976-11-18 IL IL50938A patent/IL50938A/xx unknown
- 1976-11-18 CA CA265,988A patent/CA1083148A/fr not_active Expired
- 1976-11-18 ZA ZA766923A patent/ZA766923B/xx unknown
- 1976-11-19 NL NL7612894A patent/NL7612894A/xx not_active Application Discontinuation
- 1976-11-19 PH PH19147A patent/PH11898A/en unknown
- 1976-11-19 OA OA55987A patent/OA05485A/fr unknown
- 1976-11-19 CH CH1458776A patent/CH596210A5/xx not_active IP Right Cessation
- 1976-11-19 MX MX765141U patent/MX3904E/es unknown
- 1976-11-22 NZ NZ182681A patent/NZ182681A/xx unknown

Also Published As

Publication number	Publication date
ES453460A1 (es)	1977-11-16
PH11898A (en)	1978-08-29
IE44078L (en)	1977-05-19
CH596210A5 (fr)	1978-03-15
AU1975776A (en)	1978-05-25
US4100286A (en)	1978-07-11
ZA766923B (en)	1977-10-26
FR2332020B1 (fr)	1980-10-10
DE2651789C2 (de)	1984-09-13
JPS5439396B2 (fr)	1979-11-27
AU508926B2 (en)	1980-04-17
BE848505A (fr)	1977-05-18
NZ182681A (en)	1978-07-10
AR214186A1 (es)	1979-05-15
GB1544419A (en)	1979-04-19
NL7612894A (nl)	1977-05-23
PT65859B (en)	1978-05-17
DE2651789A1 (de)	1977-06-02
JPS5265296A (en)	1977-05-30
MX3904E (es)	1981-09-11
CA1083148A (fr)	1980-08-05
PT65859A (en)	1976-12-01
IE44078B1 (en)	1981-08-12
OA05485A (fr)	1981-03-31
GR61601B (en)	1978-12-02
FR2332020A1 (fr)	1977-06-17

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