IL73853A - Substituted 1-aryl-2-fluoro-2-azolyl-alkanones,-alkanols,esters and ethers,their preparation and their use as microbicides - Google Patents

Substituted 1-aryl-2-fluoro-2-azolyl-alkanones,-alkanols,esters and ethers,their preparation and their use as microbicides

Info

Publication number: IL73853A
Authority: IL; Israel
Prior art keywords: halogen; c6alkyl; cyano; nitro; substituted
Prior art date: 1983-12-20

Application number

IL73853A

Other languages

English (en)

Other versions

IL73853A0 (en

Original Assignee

Ciba Geigy

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-12-20

Filing date

1984-12-18

Publication date

1988-07-31

1984-12-18 Application filed by Ciba Geigy filed Critical Ciba Geigy

1985-03-31 Publication of IL73853A0 publication Critical patent/IL73853A0/xx

1988-07-31 Publication of IL73853A publication Critical patent/IL73853A/xx

Links

150000002148 esters Chemical class 0.000 title abstract 2
150000002170 ethers Chemical class 0.000 title abstract 2
230000003641 microbiacidal effect Effects 0.000 title abstract 2
229940124561 microbicide Drugs 0.000 title 1
229910052736 halogen Inorganic materials 0.000 abstract 6
150000002367 halogens Chemical group 0.000 abstract 6
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 5
125000004093 cyano group Chemical group *C#N 0.000 abstract 5
229910052739 hydrogen Inorganic materials 0.000 abstract 5
239000001257 hydrogen Substances 0.000 abstract 5
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 5
150000002431 hydrogen Chemical group 0.000 abstract 4
125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 3
125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 3
RAXXELZNTBOGNW-UHFFFAOYSA-N 1H-imidazole Chemical compound C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 abstract 3
-1 2-tetrahydrofuryl Chemical group 0.000 abstract 3
125000006677 (C1-C3) haloalkoxy group Chemical group 0.000 abstract 2
NSPMIYGKQJPBQR-UHFFFAOYSA-N 4H-1,2,4-triazole Chemical compound C=1N=CNN=1 NSPMIYGKQJPBQR-UHFFFAOYSA-N 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 1
125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 1
125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
125000002941 2-furyl group Chemical group O1C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
240000007594 Oryza sativa Species 0.000 abstract 1
235000007164 Oryza sativa Nutrition 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
201000010099 disease Diseases 0.000 abstract 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
239000002184 metal Chemical class 0.000 abstract 1
229910052760 oxygen Inorganic materials 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
235000009566 rice Nutrition 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
229910052717 sulfur Inorganic materials 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
- A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
- C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Zoology (AREA)
Pest Control & Pesticides (AREA)
Plant Pathology (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Dentistry (AREA)
Environmental Sciences (AREA)
Wood Science & Technology (AREA)
Agronomy & Crop Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Carbon And Carbon Compounds (AREA)
Micromachines (AREA)

IL73853A 1983-12-20 1984-12-18 Substituted 1-aryl-2-fluoro-2-azolyl-alkanones,-alkanols,esters and ethers,their preparation and their use as microbicides IL73853A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CH675783		1983-12-20
CH273184		1984-06-05

Publications (2)

Publication Number	Publication Date
IL73853A0 IL73853A0 (en)	1985-03-31
IL73853A true IL73853A (en)	1988-07-31

Family

ID=25691269

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL73853A IL73853A (en)	1983-12-20	1984-12-18	Substituted 1-aryl-2-fluoro-2-azolyl-alkanones,-alkanols,esters and ethers,their preparation and their use as microbicides

Country Status (14)

Country	Link
US (1)	US4690942A (fr)
EP (1)	EP0149426B1 (fr)
JP (1)	JPS60222464A (fr)
KR (1)	KR920005825B1 (fr)
AT (1)	ATE33982T1 (fr)
AU (1)	AU579338B2 (fr)
BR (1)	BR8406579A (fr)
DE (1)	DE3470881D1 (fr)
ES (3)	ES8607250A1 (fr)
GB (1)	GB2152045B (fr)
HK (1)	HK31989A (fr)
IL (1)	IL73853A (fr)
MY (1)	MY100384A (fr)
PH (1)	PH23094A (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR880001813B1 (ko) *	1983-01-10	1988-09-19	시바-가이기 코오포레이숀	플루오로아졸릴 프로판 유도체의 제조방법
GB8305377D0 (en) *	1983-02-25	1983-03-30	Pfizer Ltd	Antifungal agents
EP0228995A1 (fr) *	1985-12-20	1987-07-15	Ciba-Geigy Ag	Microbicides
IT1204773B (it) *	1986-01-23	1989-03-10	Montedison Spa	Azolilderivati fungicidi
US4851423A (en) *	1986-12-10	1989-07-25	Schering Corporation	Pharmaceutically active compounds
TW432733B (en) *	1997-10-02	2001-05-01	Basf Ag	Esters as solvents in electrolyte systems for Li-ion storage cells
US6297239B1 (en) *	1997-10-08	2001-10-02	Merck & Co., Inc.	Inhibitors of prenyl-protein transferase
US8212053B2 (en) *	2005-12-28	2012-07-03	Daikin Industries, Ltd.	Process for preparing heteroaromatic ring compound having N-Rf group
CN100382801C (zh) *	2006-03-14	2008-04-23	北京大学	α-(2,4-二氯苯基)-1H-咪唑-1-乙醇在制备治疗肝炎的药物中的用途
KR20140040235A (ko)	2011-06-19	2014-04-02	비아멧 파마슈티컬즈, 인코포레이티드	금속효소 억제제 화합물
WO2012177635A1 (fr) *	2011-06-19	2012-12-27	Viamet Pharmaceuticals, Inc.	Composés inhibiteurs de métalloenzymes
EP2746262A1 (fr)	2012-12-19	2014-06-25	Basf Se	Composés de [1,2,4]triazole et d'imidazole substitués pour combattre les champignons phytopathogènes
EP2746263A1 (fr)	2012-12-19	2014-06-25	Basf Se	Triazoles à substitution alpha et imidazoles
CA2986041C (fr)	2015-05-18	2021-06-29	Viamet Pharmaceuticals, Inc.	Composes de 4-((6-(2-(2,4-difluorophenyle)1,1-difluoro-2-hydroxy-3(1h-1,2,4-triazol-1-yl)propyle)pyridine-3-yl)oxy)benzonitrile et de 4-((6-(2-(2,4-difluorophenyle)1,1-difluoro-2-hydroxy-3(5-thioxo-4,5-dihydro-1h-1,2,4-triazol-1-yl)propyle)pyridine-3-yl)oxy)benzonitrite comme

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2431407C2 (de) *	1974-06-29	1982-12-02	Bayer Ag, 5090 Leverkusen	1,2,4-Triazol-1-yl-alkanone und -alkanole, Verfahren zu ihrer Herstellung sowie ihre Verwendung als Fungizide
US4389409A (en) *	1977-03-18	1983-06-21	Rohm And Haas Company	1-(α-n-Butylthio-2,4-dichlorophenethyl)imidazol-3-yl and fungicidal use thereof
GB2010813B (en) *	1977-10-19	1982-07-28	Wellcome Found	Imidazole derivatives and salts thereof their synthesis and intermediates and pharmaceutical formulations
EP0003732B1 (fr) *	1978-02-01	1983-10-19	The Wellcome Foundation Limited	Dérivés d'imidazole et leurs sels, leur préparation et leurs formulations pharmaceutiques
DE2833194A1 (de) *	1978-07-28	1980-02-14	Basf Ag	Triazolderivate
DE2926280A1 (de) *	1979-06-29	1981-01-08	Basf Ag	Fungizide alpha -triazolylglykolderivate, ihre herstellung und verwendung
DE2937595A1 (de) *	1979-09-18	1981-04-02	Bayer Ag, 5090 Leverkusen	Verfahren zur herstellung von 1-azolyl-1-phenoxy-alkan-2-onen
GB2078719B (en) *	1980-06-02	1984-04-26	Ici Ltd	Heterocyclic compounds
DE3021551A1 (de) *	1980-06-07	1981-12-24	Bayer Ag, 5090 Leverkusen	4-substituierte 1-azolyl-1-phenoxy-3,3-dimethyl-butan-2-one und -ole, verfahren zu ihrer herstellung und ihre verwendung als fungizide
DE3169611D1 (en) *	1980-12-12	1985-05-02	Sankyo Co	Diazole and triazole derivatives, processes for their preparation and anti-microbial compositions containing them
DE3267642D1 (en) *	1981-03-10	1986-01-09	Ciba Geigy Ag	Process for the preparation of phenylethyl triazoles
DE3126478A1 (de) *	1981-07-04	1983-01-20	Basf Ag, 6700 Ludwigshafen	Azolderivate, verfahren zu ihrer herstellung und diese enthaltende fungizide
DE3132335A1 (de) *	1981-08-17	1983-03-03	Bayer Ag, 5090 Leverkusen	Substituierte azolyl-phenoxy-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
DE3140276A1 (de) *	1981-10-10	1983-04-28	Bayer Ag, 5090 Leverkusen	Phenoxyphenyl-azolylmethyl-ketone und -carbinole, verfahren zu ihrer herstellung und ihre verwendung als fungizide und als zwischenprodukte
JPS6055072B2 (ja) *	1982-07-12	1985-12-03	四国化成工業株式会社	新規イミダゾ−ル化合物及びその製造方法
KR880001813B1 (ko) *	1983-01-10	1988-09-19	시바-가이기 코오포레이숀	플루오로아졸릴 프로판 유도체의 제조방법
GB8305377D0 (en) *	1983-02-25	1983-03-30	Pfizer Ltd	Antifungal agents
US4539325A (en) *	1983-11-07	1985-09-03	Janssen Pharmaceutica N.V.	1-(2-Aryl-2-halo-1-ethenyl)-1H-azoles, and anticonvulsant use thereof
US4577032A (en) *	1984-06-15	1986-03-18	Takayuki Fujita	1-Benzoyldibromomethyl-2-methylimidazole as a fungicidal agent

1984
- 1984-12-14 DE DE8484810619T patent/DE3470881D1/de not_active Expired
- 1984-12-14 AT AT84810619T patent/ATE33982T1/de active
- 1984-12-14 US US06/681,989 patent/US4690942A/en not_active Expired - Fee Related
- 1984-12-14 EP EP84810619A patent/EP0149426B1/fr not_active Expired
- 1984-12-18 GB GB08431974A patent/GB2152045B/en not_active Expired
- 1984-12-18 IL IL73853A patent/IL73853A/xx not_active IP Right Cessation
- 1984-12-19 BR BR8406579A patent/BR8406579A/pt not_active IP Right Cessation
- 1984-12-19 AU AU36957/84A patent/AU579338B2/en not_active Ceased
- 1984-12-19 ES ES538851A patent/ES8607250A1/es not_active Expired
- 1984-12-19 PH PH31609A patent/PH23094A/en unknown
- 1984-12-20 JP JP59267599A patent/JPS60222464A/ja active Granted
- 1984-12-20 KR KR1019840008158A patent/KR920005825B1/ko not_active Expired
1986
- 1986-01-02 ES ES551189A patent/ES8703850A1/es not_active Expired
- 1986-01-02 ES ES551190A patent/ES8802361A1/es not_active Expired
1987
- 1987-05-18 MY MYPI87000675A patent/MY100384A/en unknown
1989
- 1989-04-13 HK HK319/89A patent/HK31989A/xx unknown

Also Published As

Publication number	Publication date
KR850004469A (ko)	1985-07-15
ES8607250A1 (es)	1986-06-01
JPH0582387B2 (fr)	1993-11-18
US4690942A (en)	1987-09-01
EP0149426B1 (fr)	1988-05-04
MY100384A (en)	1990-09-17
ES551189A0 (es)	1987-03-01
PH23094A (en)	1989-04-10
ES538851A0 (es)	1986-06-01
BR8406579A (pt)	1985-10-15
EP0149426A1 (fr)	1985-07-24
AU3695784A (en)	1985-07-04
AU579338B2 (en)	1988-11-24
GB2152045B (en)	1988-04-27
KR920005825B1 (ko)	1992-07-20
GB8431974D0 (en)	1985-01-30
ATE33982T1 (de)	1988-05-15
ES8703850A1 (es)	1987-03-01
ES8802361A1 (es)	1988-05-16
IL73853A0 (en)	1985-03-31
JPS60222464A (ja)	1985-11-07
HK31989A (en)	1989-04-21
DE3470881D1 (de)	1988-06-09
ES551190A0 (es)	1988-05-16
GB2152045A (en)	1985-07-31

Legal Events

Date	Code	Title	Description
1998-02-08	HC	Change of name of proprietor(s)
1999-12-22	RH	Patent void

Publication	Publication Date	Title
AU579338B2 (en)	1988-11-24	1-Aryl-2-fluoro-2-azolylalkanones and derivatives thereof
DE69522947D1 (en)	2001-10-31	Phenylxanthin-derivate
ES8207169A1 (es)	1982-09-01	Un procedimiento para la preparacion de nuevos derivados de piperazinilquinazolina y de homopiperazinilquinazolina hi- pertensora con acticidad.
IL112074A0 (en)	1995-03-15	Branched-amino-substituted thiazoles, their preparation and pharmaceutical compositions containing them
GR880300169T1 (en)	1989-01-31	N-hydroxypropylisopropyl ether derivatives of chitosan, and cosmetic compositions containing them
NO932992D0 (no)	1993-08-23	Nye polyjoderte forbindelser, fremgangsmaate for deres fremstilling og kontrastmidler inneholdende dem
IL108856A0 (en)	1994-06-24	Hydroxymethyl-furazancarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
IL89716A0 (en)	1989-09-28	Substituted isonicotinic acid esters,their preparation and their use for protecting plants against diseases
PL313037A1 (en)	1996-05-27	Phenoxphenylocyclopententenylohydroxyureas
ES8203350A1 (es)	1982-04-01	Procedimiento para la fabricacion de derivados del pirazol
AU563810B2 (en)	1987-07-23	Plant growth regulators
EP0337413A3 (fr)	1990-11-22	Dérivés de naphtopyranes et leur usage
IL95608A0 (en)	1991-06-30	1-methoxypyrimidinyl-n-nitro-phenyl-1h,1,2,4-triazole-3-sulphonamide derivatives and herbicidal compositions containing the same
ES8105307A1 (es)	1981-06-01	Procedimiento para la preparacion de 4-oxa-6-aza-6(fenil-es-piro)(2.4)heptan-5,7-dionas
ES8605467A1 (es)	1986-03-16	Procedimiento para la preparacion de derivados de 1-(amino- fenil)-2-amino-etanona
IL67272A (en)	1986-04-29	Alkylcycloalkyl imidazolylmethyl ketones and their preparation
GR3024709T3 (en)	1997-12-31	Novel cytarabine derivatives, their production and use