IL83792A - 5- and/or 23-o-acylated milbemycin analogs and pesticidal compositions containing them - Google Patents

5- and/or 23-o-acylated milbemycin analogs and pesticidal compositions containing them

Info

Publication number: IL83792A
Authority: IL; Israel
Prior art keywords: compounds; acyl; compositions containing; acylated; pesticidal compositions
Prior art date: 1986-09-12

Application number

IL83792A

Other languages

English (en)

Original Assignee

American Cyanamid Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-09-12

Filing date

1987-09-06

Publication date

1993-02-21

1987-09-06 Application filed by American Cyanamid Co filed Critical American Cyanamid Co

1993-02-21 Publication of IL83792A publication Critical patent/IL83792A/xx

Links

239000000203 mixture Substances 0.000 title abstract 2
FXWHFKOXMBTCMP-WMEDONTMSA-N milbemycin Natural products COC1C2OCC3=C/C=C/C(C)CC(=CCC4CC(CC5(O4)OC(C)C(C)C(OC(=O)C(C)CC(C)C)C5O)OC(=O)C(C=C1C)C23O)C FXWHFKOXMBTCMP-WMEDONTMSA-N 0.000 title 1
230000000361 pesticidal effect Effects 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 5
VHYFNPMBLIVWCW-UHFFFAOYSA-N 4-Dimethylaminopyridine Chemical compound CN(C)C1=CC=NC=C1 VHYFNPMBLIVWCW-UHFFFAOYSA-N 0.000 abstract 2
230000010933 acylation Effects 0.000 abstract 2
238000005917 acylation reaction Methods 0.000 abstract 2
241000970253 Streptomyces cyaneogriseus Species 0.000 abstract 1
230000000895 acaricidal effect Effects 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
150000008064 anhydrides Chemical class 0.000 abstract 1
230000000507 anthelmentic effect Effects 0.000 abstract 1
150000001805 chlorine compounds Chemical class 0.000 abstract 1
230000001984 ectoparasiticidal effect Effects 0.000 abstract 1
230000004151 fermentation Effects 0.000 abstract 1
238000000855 fermentation Methods 0.000 abstract 1
230000000749 insecticidal effect Effects 0.000 abstract 1
230000001069 nematicidal effect Effects 0.000 abstract 1
230000003389 potentiating effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N49/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds containing the group, wherein m+n>=1, both X together may also mean —Y— or a direct carbon-to-carbon bond, and the carbon atoms marked with an asterisk are not part of any ring system other than that which may be formed by the atoms X, the carbon atoms in square brackets being part of any acyclic or cyclic structure, or the group, wherein A means a carbon atom or Y, n>=0, and not more than one of these carbon atoms being a member of the same ring system, e.g. juvenile insect hormones or mimics thereof
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/195—Antibiotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents

Landscapes

Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Zoology (AREA)
Polymers & Plastics (AREA)
Agronomy & Crop Science (AREA)
Environmental Sciences (AREA)
Wood Science & Technology (AREA)
Dentistry (AREA)
Plant Pathology (AREA)
Pest Control & Pesticides (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Insects & Arthropods (AREA)
Food Science & Technology (AREA)
Animal Husbandry (AREA)
Genetics & Genomics (AREA)
Veterinary Medicine (AREA)
Biotechnology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Tropical Medicine & Parasitology (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Photoreceptors In Electrophotography (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

IL83792A 1986-09-12 1987-09-06 5- and/or 23-o-acylated milbemycin analogs and pesticidal compositions containing them IL83792A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/907,281 US5149832A (en)	1986-09-12	1986-09-12	Mono and diacyl derivatives of ll-f28249 compounds

Publications (1)

Publication Number	Publication Date
IL83792A true IL83792A (en)	1993-02-21

Family

ID=25423825

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL83792A IL83792A (en)	1986-09-12	1987-09-06	5- and/or 23-o-acylated milbemycin analogs and pesticidal compositions containing them

Country Status (17)

Country	Link
US (1)	US5149832A (de)
EP (1)	EP0259686B1 (de)
JP (1)	JPS63132890A (de)
KR (1)	KR880003948A (de)
AT (1)	ATE96440T1 (de)
AU (1)	AU593682B2 (de)
BR (1)	BR8704737A (de)
CA (1)	CA1317936C (de)
DE (1)	DE3787942T2 (de)
DK (1)	DK475487A (de)
ES (1)	ES2059333T3 (de)
HU (1)	HU199145B (de)
IE (1)	IE62248B1 (de)
IL (1)	IL83792A (de)
NZ (1)	NZ221692A (de)
PT (1)	PT85673B (de)
ZA (1)	ZA876834B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4806527A (en) *	1987-03-16	1989-02-21	Merck & Co., Inc.	Avermectin derivatives
GB8721378D0 (en) *	1987-09-11	1987-10-21	Glaxo Group Ltd	Chemical process
JP2629047B2 (ja) *	1988-05-10	1997-07-09	アメリカン・サイアナミツド・カンパニー	マクロライド化合物
WO1999017760A2 (en)	1997-10-02	1999-04-15	Microcide Pharmaceuticals, Inc.	Fungal or mammalian cell efflux pump inhibitors for enhancing susceptibility of the cell to a drug
FR2948261B1 (fr) *	2009-07-22	2015-10-30	Sarl Herbarom Laboratoire	Procede insecticide et/ou repulsif
CN104860961B (zh) *	2015-04-10	2017-08-04	新宇药业股份有限公司	一种制备5‑氧（对‑硝基苯甲酰）‑尼莫克汀的方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4201861A (en) *	1977-10-03	1980-05-06	Merck & Co., Inc.	Acyl derivatives of C-076 compounds
IL56149A (en) *	1977-12-19	1989-09-28	Merck & Co Inc	13-halo and 13-deoxy derivatives of c-076 compounds,their preparation and method for the treatment of parasitic infections in animals therewith
USRE32034E (en) *	1977-12-19	1985-11-19	Merck & Co., Inc.	13-Halo and 13-deoxy derivatives of C-076 compounds
JPS57120589A (en) *	1981-01-20	1982-07-27	Sankyo Co Ltd	5-methoxy and 5-lower alkanoyloxy derivative, its preparation and acaricide and parasiticide
DK165119C (da) *	1984-06-05	1993-03-01	American Cyanamid Co	Antibiotiske forbindelser betegnet ll-f28249alfa, beta, gamma, delta, epsilon, zeta, eta, theta, iota, kappa, my og ny og pharmaceutisk or pharmakologisk acceptable salte deraf samt fremgangsmaade til deres fremstilling
DE3532794A1 (de) *	1984-09-14	1986-04-17	Glaxo Group Ltd., London	Antibiotika, verfahren zu deren herstellung und diese verbindungen enthaltende mittel
ES8802229A1 (es) *	1985-04-30	1988-04-16	Glaxo Group Ltd	Un procedimiento para preparar nuevos derivados lactonicos macrociclicos.
ES8800986A1 (es) *	1985-07-27	1987-12-01	Pfizer	Un procedimiento para la produccion de un nuevo derivado de avermectina
IE67373B1 (en) *	1985-09-13	1996-03-20	American Cyanamid Co	Macrolide antibiotics and their preparation

1986
- 1986-09-12 US US06/907,281 patent/US5149832A/en not_active Expired - Fee Related
1987
- 1987-08-25 AT AT87112277T patent/ATE96440T1/de not_active IP Right Cessation
- 1987-08-25 EP EP87112277A patent/EP0259686B1/de not_active Expired - Lifetime
- 1987-08-25 DE DE87112277T patent/DE3787942T2/de not_active Expired - Fee Related
- 1987-08-25 ES ES87112277T patent/ES2059333T3/es not_active Expired - Lifetime
- 1987-09-06 IL IL83792A patent/IL83792A/xx not_active IP Right Cessation
- 1987-09-07 NZ NZ221692A patent/NZ221692A/xx unknown
- 1987-09-10 PT PT85673A patent/PT85673B/pt not_active IP Right Cessation
- 1987-09-10 CA CA000546558A patent/CA1317936C/en not_active Expired - Fee Related
- 1987-09-11 IE IE243387A patent/IE62248B1/en not_active IP Right Cessation
- 1987-09-11 ZA ZA876834A patent/ZA876834B/xx unknown
- 1987-09-11 BR BR8704737A patent/BR8704737A/pt not_active IP Right Cessation
- 1987-09-11 HU HU874051A patent/HU199145B/hu not_active IP Right Cessation
- 1987-09-11 AU AU78279/87A patent/AU593682B2/en not_active Ceased
- 1987-09-11 KR KR870010119A patent/KR880003948A/ko not_active Withdrawn
- 1987-09-11 JP JP62226735A patent/JPS63132890A/ja active Pending
- 1987-09-11 DK DK475487A patent/DK475487A/da not_active Application Discontinuation

Also Published As

Publication number	Publication date
ZA876834B (en)	1988-03-15
PT85673A (en)	1987-10-01
US5149832A (en)	1992-09-22
NZ221692A (en)	1990-09-26
KR880003948A (ko)	1988-05-31
JPS63132890A (ja)	1988-06-04
ES2059333T3 (es)	1994-11-16
DE3787942T2 (de)	1994-05-11
CA1317936C (en)	1993-05-18
DE3787942D1 (de)	1993-12-02
BR8704737A (pt)	1988-05-03
AU593682B2 (en)	1990-02-15
HUT45535A (en)	1988-07-28
DK475487D0 (da)	1987-09-11
IE62248B1 (en)	1995-01-11
DK475487A (da)	1988-03-13
IE872433L (en)	1988-03-12
EP0259686A1 (de)	1988-03-16
ATE96440T1 (de)	1993-11-15
PT85673B (pt)	1990-05-31
AU7827987A (en)	1988-03-17
EP0259686B1 (de)	1993-10-27
HU199145B (en)	1990-01-29

Legal Events

Date	Code	Title	Description
1998-09-24	RH	Patent void

Publication	Publication Date	Title
IE872438L (en)	1988-03-12	23-oxo(keto) and 23-imino derivatives of ll-f28249 compounds
ZA876833B (en)	1988-03-15	Novel 23-imino derivatives of 23-keto compounds
AU7827987A (en)	1988-03-17	Spiro derivatives
IE872440L (en)	1988-03-12	13-deoxy-23-oxo (keto) and 23-imino derivatives of 13-deoxy¹c-076-aglycone compounds
NZ221691A (en)	1990-09-26	Milbemycin (ll-f28249) derivatives and parasiticidal compositions
IE880622L (en)	1988-09-06	Mono- and diepoxide derivatives of delta 22-LL-F28249¹compounds
NZ221693A (en)	1989-11-28	Delta-23-milbemycin derivatives and parasiticidal compositions
IE880621L (en)	1988-09-06	Mono- and diepoxide derivatives of 23-deoxy-LL-F28249¹compounds