IL87421A - Pharmaceutical compositions containing 5-amino (or substituted amino) - 1,2,3-triazoles - Google Patents

Pharmaceutical compositions containing 5-amino (or substituted amino) - 1,2,3-triazoles

Info

Publication number: IL87421A
Authority: IL; Israel
Prior art keywords: amino; triazoles; pharmaceutical compositions; compositions containing; substituted amino
Prior art date: 1987-08-20

Application number

IL87421A

Other languages

English (en)

Other versions

IL87421A0 (en

Original Assignee

Merck & Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-08-20

Filing date

1988-08-11

Publication date

1992-12-01

1988-08-11 Application filed by Merck & Co Inc filed Critical Merck & Co Inc

1989-01-31 Publication of IL87421A0 publication Critical patent/IL87421A0/xx

1992-12-01 Publication of IL87421A publication Critical patent/IL87421A/xx

Links

239000008194 pharmaceutical composition Substances 0.000 title 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 title 1
JSIAIROWMJGMQZ-UHFFFAOYSA-N 2h-triazol-4-amine Chemical class NC1=CNN=N1 JSIAIROWMJGMQZ-UHFFFAOYSA-N 0.000 abstract 1
206010028980 Neoplasm Diseases 0.000 abstract 1
201000004681 Psoriasis Diseases 0.000 abstract 1
230000001028 anti-proliverative effect Effects 0.000 abstract 1
201000011510 cancer Diseases 0.000 abstract 1
230000002757 inflammatory effect Effects 0.000 abstract 1
208000011580 syndromic disease Diseases 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

Landscapes

Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

IL87421A 1987-08-20 1988-08-11 Pharmaceutical compositions containing 5-amino (or substituted amino) - 1,2,3-triazoles IL87421A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/087,494 US4847257A (en)	1987-08-20	1987-08-20	5-Amino or substituted amino 1,2,3,-triazoles useful as antiproliferative agents

Publications (2)

Publication Number	Publication Date
IL87421A0 IL87421A0 (en)	1989-01-31
IL87421A true IL87421A (en)	1992-12-01

Family

ID=22205528

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL87421A IL87421A (en)	1987-08-20	1988-08-11	Pharmaceutical compositions containing 5-amino (or substituted amino) - 1,2,3-triazoles

Country Status (16)

Country	Link
US (2)	US4847257A (de)
EP (1)	EP0304221B1 (de)
JP (1)	JP2572115B2 (de)
KR (1)	KR960014871B1 (de)
AT (1)	ATE101513T1 (de)
AU (1)	AU612172B2 (de)
CA (1)	CA1325977C (de)
CY (1)	CY1954A (de)
DE (1)	DE3887793T2 (de)
DK (1)	DK175915B1 (de)
HK (1)	HK107596A (de)
IE (1)	IE61719B1 (de)
IL (1)	IL87421A (de)
NZ (1)	NZ225770A (de)
PT (1)	PT88275B (de)
ZA (1)	ZA886125B (de)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5359078A (en) *	1989-05-19	1994-10-25	The United States Of America As Represented By The Department Of Health And Human Services	Signal transduction inhibitor compounds
US5880129A (en) *	1989-05-19	1999-03-09	The United States Of America As Represented By The Department Of Health And Human Services	Methods of inhibiting invasion and metastasis of malignant solid tumors
US5498620A (en) *	1989-05-19	1996-03-12	The United States Of America As Represented By The Department Of Health And Human Services	Signal transduction inhibitor 1,2,3-triazolo compounds
US5132315A (en) *	1989-05-19	1992-07-21	The United States Of America As Represented By The Department Of Health And Human Services	Therapeutic application of an anti-invasive compound
WO1992012144A1 (en) *	1990-12-28	1992-07-23	Teijin Limited	Condensed benzoxa ring compound, production thereof, and pharmaceutical composition containing the same
US5744492A (en) *	1993-09-17	1998-04-28	United States Of America	Method for inhibiting angiogenesis
US5602156A (en) *	1993-09-17	1997-02-11	The United States Of America As Represented By The Department Of Health And Human Services	Method for inhibiting metalloproteinase expression
US5728707A (en) *	1995-07-21	1998-03-17	Constantia Gruppe	Treatment and prevention of primary and metastatic neoplasms with salts of aminoimidazole carboxamide
ATE278399T1 (de) *	1995-07-21	2004-10-15	Savvipharm Inc	Orotatsalze von 5-amino- oder substituierten amino-1,2,3-triazolen zur behandlung von neoplasmen
US8198334B2 (en) *	1997-10-27	2012-06-12	Pathologica Llc	Methods for modulating macrophage proliferation in ocular disease using polyamine analogs
US7087648B1 (en) *	1997-10-27	2006-08-08	The Regents Of The University Of California	Methods for modulating macrophage proliferation using polyamine analogs
US5886038A (en) *	1998-03-24	1999-03-23	Panda Pharmaceuticals, L.L.C.	Composition and method for treatment of psoriasis
US5990100A (en) *	1998-03-24	1999-11-23	Panda Pharmaceuticals, L.L.C.	Composition and method for treatment of psoriasis
US6702801B2 (en) *	1998-05-07	2004-03-09	Kimberly-Clark Worldwide, Inc.	Absorbent garment with an extensible backsheet
AU2005294514A1 (en) *	2004-10-04	2006-04-20	Cellgate, Inc.	Polyamine analogs as therapeutic agents for ocular diseases
US7531560B2 (en) *	2004-11-10	2009-05-12	Boehringer Ingelheim Pharmaceuticals, Inc.	Anti-cytokine heterocyclic compounds
CN101164538B (zh) *	2006-10-16	2011-12-14	中国医学科学院基础医学研究所	羧胺三唑类化合物及其盐在制备治疗疼痛性疾病和/或炎症性疾病的药物中的应用
CA2772075C (en) *	2009-09-04	2017-02-28	Rashida A. Karmali	Novel compositions and processes for preparing 5-amino or substituted amino 1,2,3-triazoles and triazole orotate formulations
CN112358451B (zh) *	2021-01-11	2021-04-13	广东银珠医药科技有限公司	羧胺三唑的合成方法
CN113620892B (zh) *	2021-10-12	2022-02-22	广东银珠医药科技有限公司	羧胺三唑单晶、制备方法及其组合物和用途

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4590201A (en) *	1984-02-02	1986-05-20	Merck & Co., Inc.	5-amino or substituted amino 1,2,3-triazoles

1987
- 1987-08-20 US US07/087,494 patent/US4847257A/en not_active Expired - Lifetime
1988
- 1988-08-10 NZ NZ225770A patent/NZ225770A/xx unknown
- 1988-08-11 IL IL87421A patent/IL87421A/xx not_active IP Right Cessation
- 1988-08-11 EP EP88307418A patent/EP0304221B1/de not_active Expired - Lifetime
- 1988-08-11 AT AT88307418T patent/ATE101513T1/de not_active IP Right Cessation
- 1988-08-11 DE DE3887793T patent/DE3887793T2/de not_active Expired - Lifetime
- 1988-08-15 CA CA000574763A patent/CA1325977C/en not_active Expired - Fee Related
- 1988-08-16 PT PT88275A patent/PT88275B/pt not_active IP Right Cessation
- 1988-08-18 ZA ZA886125A patent/ZA886125B/xx unknown
- 1988-08-19 KR KR1019880010519A patent/KR960014871B1/ko not_active Expired - Fee Related
- 1988-08-19 DK DK198804654A patent/DK175915B1/da not_active IP Right Cessation
- 1988-08-19 AU AU21159/88A patent/AU612172B2/en not_active Expired
- 1988-08-19 IE IE255188A patent/IE61719B1/en not_active IP Right Cessation
- 1988-08-20 JP JP63205715A patent/JP2572115B2/ja not_active Expired - Fee Related
1989
- 1989-05-08 US US07/348,823 patent/US5045543A/en not_active Expired - Lifetime
1996
- 1996-06-19 HK HK107596A patent/HK107596A/en not_active IP Right Cessation
1997
- 1997-05-16 CY CY195497A patent/CY1954A/xx unknown

Also Published As

Publication number	Publication date
KR960014871B1 (ko)	1996-10-21
DE3887793D1 (de)	1994-03-24
US4847257A (en)	1989-07-11
HK107596A (en)	1996-06-28
EP0304221A2 (de)	1989-02-22
DK465488D0 (da)	1988-08-19
IE61719B1 (en)	1994-11-30
DK465488A (da)	1989-03-15
EP0304221A3 (en)	1990-09-05
ZA886125B (en)	1989-04-26
EP0304221B1 (de)	1994-02-16
JP2572115B2 (ja)	1997-01-16
IE882551L (en)	1989-02-20
ATE101513T1 (de)	1994-03-15
KR890003385A (ko)	1989-04-14
JPS6468321A (en)	1989-03-14
AU612172B2 (en)	1991-07-04
IL87421A0 (en)	1989-01-31
CY1954A (en)	1997-05-16
CA1325977C (en)	1994-01-11
PT88275A (pt)	1989-06-30
DE3887793T2 (de)	1994-07-28
NZ225770A (en)	1991-11-26
AU2115988A (en)	1989-03-16
PT88275B (pt)	1995-03-01
US5045543A (en)	1991-09-03
DK175915B1 (da)	2005-06-27

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Legal Events

Date	Code	Title
1998-12-27	KB	Patent renewed
2002-09-12	KB	Patent renewed
2006-10-04	KB	Patent renewed
2009-02-11	EXP	Patent expired
2010-04-14	EXP	Patent expired