IN2012DN00539A - - Google Patents

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Publication number
IN2012DN00539A
IN2012DN00539A IN539DEN2012A IN2012DN00539A IN 2012DN00539 A IN2012DN00539 A IN 2012DN00539A IN 539DEN2012 A IN539DEN2012 A IN 539DEN2012A IN 2012DN00539 A IN2012DN00539 A IN 2012DN00539A
Authority
IN
India
Prior art keywords
fluoropyrimidinones
fungicides
acyl
derivatives
compounds
Prior art date
Application number
Inventor
Boebel Timothy
Bryan Kristy
Lorsbach Beth
Martin Timothy
Owen W
Pobanz Mark
Thornburgh Scott
Webster Jeffery
Yao Chenglin
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2012DN00539(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of IN2012DN00539A publication Critical patent/IN2012DN00539A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

This present disclosure is related to filed of N1-acyl-5- fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides.
IN539DEN2012 2009-08-07 2010-08-05 IN2012DN00539A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
IN2012DN00539A true IN2012DN00539A (en) 2015-06-12

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
IN539DEN2012 IN2012DN00539A (en) 2009-08-07 2010-08-05

Country Status (33)

Country Link
US (1) US8470839B2 (en)
EP (1) EP2519512B1 (en)
JP (1) JP5748754B2 (en)
KR (1) KR101792285B1 (en)
CN (1) CN102548981B (en)
AU (1) AU2010279402B2 (en)
BR (1) BR112012002810B1 (en)
CA (1) CA2768510C (en)
CL (1) CL2012000316A1 (en)
CO (1) CO6491117A2 (en)
CR (1) CR20120030A (en)
CY (1) CY1122115T1 (en)
DK (1) DK2519512T3 (en)
EA (1) EA023411B1 (en)
EC (1) ECSP12011653A (en)
ES (1) ES2728966T3 (en)
HN (1) HN2012000269A (en)
HR (1) HRP20190919T1 (en)
HU (1) HUE045290T2 (en)
IL (1) IL217952A (en)
IN (1) IN2012DN00539A (en)
LT (1) LT2519512T (en)
MX (1) MX2012001620A (en)
NI (1) NI201200022A (en)
NZ (1) NZ597570A (en)
PE (1) PE20120688A1 (en)
PL (1) PL2519512T3 (en)
PT (1) PT2519512T (en)
SI (1) SI2519512T1 (en)
TR (1) TR201908180T4 (en)
UA (1) UA106889C2 (en)
WO (1) WO2011017538A1 (en)
ZA (1) ZA201200819B (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010279411B2 (en) * 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives
HUE035248T2 (en) * 2011-08-17 2018-05-02 Adama Makhteshim Ltd 1-substituted-5-fluoro-3,6-dihydro-6-imino-2(1H)-pyrimidinone derivatives as fungicidal agents for use in plant protection
HUE047711T2 (en) 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
UA117123C2 (en) * 2012-12-28 2018-06-25 Адама Махтешім Лтд. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
RU2015131149A (en) 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N- (SUBSTITUTED) -5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydro-pyrimidine-1 (2H) -carboxamide derivatives
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
EP3097096A4 (en) 2013-12-31 2017-10-11 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
EA030030B1 (en) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Synergistic fungicidal mixtures and synergistic fungicidal compositions for fungal control
CN107001397B (en) 2014-09-26 2020-10-13 科慕埃弗西有限公司 Isocyanate-Derived Organosilanes
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CR20210270A (en) 2018-11-05 2021-07-20 Adama Makhteshim Ltd MIXTURES AND COMPOSITIONS INCLUDING 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ONA, AND METHODS OF USE OF THE SAME
TWI808347B (en) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 Process for preparing 5-fluoro-4-imino-3-methyl-1-tosyl-3,4 dihydropyrimidine-2(1h)-one and derivatives of the compound
MX2022011088A (en) 2020-03-09 2022-09-29 Adama Makhteshim Ltd Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulf onyl)-3,4-dihydro-1h-pyrimidin-2-one.

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (en) * 1962-05-01 1966-10-15 Hoffmann La Roche Process for the production of a cytosine derivative
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (en) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (en) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie NOVEL DERIVATIVES OF 2,3,6,7-TETRAHYDRO 5H-THIAZOLO (3,2-A) PYRIMIDINE, THEIR PREPARATION AND THEIR USE AS HERBICIDES
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (en) 1988-03-09 1994-10-16 Ciba Geigy Ag AGENT FOR THE PROTECTION OF PLANTS AGAINST DISEASES.
DE3821711A1 (en) 1988-06-28 1990-02-08 Bayer Ag THIAZOLOPYRIMIDINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A SCHAEDLINGSBEKAEMPFUNGSMITTEL
JP3217191B2 (en) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト Heteroaromatic compounds and plant protective agents containing the same
MX9800136A (en) 1995-07-05 1998-03-29 Du Pont Fungicidal pyrimidinones.
IL125589A0 (en) 1996-03-11 1999-03-12 Novartis Ag Pyrimidin-4-one derivatives as pesticides
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (en) 1998-11-06 2001-04-18 NOVEDOSA PIRIMIDIN-4-ENAMINE AS A FUNGICIDE.
US7914799B2 (en) 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
JPWO2005095419A1 (en) 2004-04-01 2008-02-21 武田薬品工業株式会社 Thiazolopyrimidine derivatives
US20080004253A1 (en) 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
AR070228A1 (en) 2008-01-22 2010-03-25 Dow Agrosciences Llc DERIVATIVES OF 5-FLUORO PIRIMIDINA
WO2010047866A2 (en) 2008-08-01 2010-04-29 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide
ME02254B (en) 2009-01-23 2015-12-31 Euro Celtique Sa Hydroxamic acid derivatives
AU2010279411B2 (en) 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
CY1122115T1 (en) 2020-11-25
CA2768510C (en) 2018-05-15
CO6491117A2 (en) 2012-07-31
LT2519512T (en) 2019-07-25
CN102548981A (en) 2012-07-04
CL2012000316A1 (en) 2014-06-27
UA106889C2 (en) 2014-10-27
ZA201200819B (en) 2013-05-29
IL217952A (en) 2017-11-30
NI201200022A (en) 2012-05-22
CR20120030A (en) 2012-03-28
JP2013501723A (en) 2013-01-17
AU2010279402B2 (en) 2015-04-16
TR201908180T4 (en) 2019-06-21
EA023411B1 (en) 2016-06-30
EP2519512A1 (en) 2012-11-07
AU2010279402A1 (en) 2012-02-02
BR112012002810A2 (en) 2015-09-15
HN2012000269A (en) 2015-04-27
EA201270253A1 (en) 2012-07-30
HRP20190919T1 (en) 2019-09-20
CN102548981B (en) 2015-05-13
JP5748754B2 (en) 2015-07-15
SI2519512T1 (en) 2019-09-30
MX2012001620A (en) 2012-04-11
PL2519512T3 (en) 2019-09-30
US20110034490A1 (en) 2011-02-10
WO2011017538A1 (en) 2011-02-10
DK2519512T3 (en) 2019-05-27
NZ597570A (en) 2014-04-30
KR20120041786A (en) 2012-05-02
ES2728966T3 (en) 2019-10-29
IL217952A0 (en) 2012-03-29
HK1172894A1 (en) 2013-05-03
EP2519512A4 (en) 2013-01-16
ECSP12011653A (en) 2012-03-30
HUE045290T2 (en) 2019-12-30
US8470839B2 (en) 2013-06-25
EP2519512B1 (en) 2019-03-20
PE20120688A1 (en) 2012-06-06
BR112012002810B1 (en) 2018-12-11
CA2768510A1 (en) 2011-02-10
KR101792285B1 (en) 2017-10-31
PT2519512T (en) 2019-06-04

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