IN2012DN00602A - - Google Patents

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Publication number
IN2012DN00602A
IN2012DN00602A IN602DEN2012A IN2012DN00602A IN 2012DN00602 A IN2012DN00602 A IN 2012DN00602A IN 602DEN2012 A IN602DEN2012 A IN 602DEN2012A IN 2012DN00602 A IN2012DN00602 A IN 2012DN00602A
Authority
IN
India
Prior art keywords
phenylpiperidin
exploration
pharmacologically
biologically
oxo
Prior art date
Application number
Inventor
Castells Boliart Josep
Enrique Miguel Centeno David
Pascual Gilabert Marta
Original Assignee
Inst Univ De Ciencia I Technologia S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Inst Univ De Ciencia I Technologia S A filed Critical Inst Univ De Ciencia I Technologia S A
Publication of IN2012DN00602A publication Critical patent/IN2012DN00602A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms
    • C07D211/76—Oxygen atoms attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Novel compounds are continually sought after to treat and prevent diseases and disorders. The invention relates to N-(2-oxo-I-phenylpiperidin-3-yl)sulfonamides useful for being biologically and pharmacologically screened, and to contribute to the exploration and identification of new lead molecules that are capable of modulating the functional activity of a biological target.
IN602DEN2012 2009-06-25 2010-06-23 IN2012DN00602A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200901515 2009-06-25
PCT/IB2010/052856 WO2010150204A1 (en) 2009-06-25 2010-06-23 N-(2-oxo-1-phenylpiperidin-3-yl) sulfonamides for the identification of biological and pharmacological activity

Publications (1)

Publication Number Publication Date
IN2012DN00602A true IN2012DN00602A (en) 2015-06-12

Family

ID=42797604

Family Applications (1)

Application Number Title Priority Date Filing Date
IN602DEN2012 IN2012DN00602A (en) 2009-06-25 2010-06-23

Country Status (4)

Country Link
US (1) US8569507B2 (en)
EP (1) EP2445879A1 (en)
IN (1) IN2012DN00602A (en)
WO (1) WO2010150204A1 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2352398B1 (en) 2009-06-25 2011-09-29 Institut Univ. De Ciencia I Tecnologia S.A. N-FENETILSULFONAMIDAS-N-SUBSTITUTED FOR THE IDENTIFICATION OF BIOLOGICAL AND PHARMACOLOGICAL ACTIVITY.
EP2445879A1 (en) 2009-06-25 2012-05-02 Institut Univ. de Ciència i Tecnologia, S.A. N-(2-oxo-1-phenylpiperidin-3-yl) sulfonamides for the identification of biological and pharmacological activity
ES2350548B1 (en) 2009-06-25 2011-09-29 Institut Univ. De Ciència I Tecnologia, S.A. N-FENIL-1-SULFONIL-2-PIRROLIDINACARBOXAMIDS FOR THE IDENTIFICATION OF BIOLOGICAL AND PHARMACOLOGICAL ACTIVITY.
ES2354550B1 (en) * 2009-06-26 2011-11-15 Institut Univ. De Ciència I Tecnologia, S.A. LIBRARY OF N- (1-PHENYL-2-OXO-3-PIPERIDIL) SULFONAMIDS FOR THE DISCOVERY OF DRUGS.
BR112020018094A2 (en) 2018-03-08 2020-12-22 Incyte Corporation AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-¿INHIBITORS
EP3587416A1 (en) * 2018-06-29 2020-01-01 Institut Univ. de Ciència i Tecnologia, S.A. 2-oxopiperidin-3-yl derivatives and use thereof
US11046658B2 (en) 2018-07-02 2021-06-29 Incyte Corporation Aminopyrazine derivatives as PI3K-γ inhibitors

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6939973B1 (en) 1999-02-09 2005-09-06 The Scripps Research Institute Glycoluril core molecules for combinatorial libraries
US6710058B2 (en) * 2000-11-06 2004-03-23 Bristol-Myers Squibb Pharma Company Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors
TW200307667A (en) 2002-05-06 2003-12-16 Bristol Myers Squibb Co Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors
DE102004059219A1 (en) * 2004-12-09 2006-06-14 Bayer Healthcare Ag Pyrazine dicarboxylic acid amides and their use
US7979558B2 (en) 2008-08-06 2011-07-12 Futurewei Technologies, Inc. Remote session control
EP2445879A1 (en) 2009-06-25 2012-05-02 Institut Univ. de Ciència i Tecnologia, S.A. N-(2-oxo-1-phenylpiperidin-3-yl) sulfonamides for the identification of biological and pharmacological activity
ES2350548B1 (en) 2009-06-25 2011-09-29 Institut Univ. De Ciència I Tecnologia, S.A. N-FENIL-1-SULFONIL-2-PIRROLIDINACARBOXAMIDS FOR THE IDENTIFICATION OF BIOLOGICAL AND PHARMACOLOGICAL ACTIVITY.
ES2352398B1 (en) 2009-06-25 2011-09-29 Institut Univ. De Ciencia I Tecnologia S.A. N-FENETILSULFONAMIDAS-N-SUBSTITUTED FOR THE IDENTIFICATION OF BIOLOGICAL AND PHARMACOLOGICAL ACTIVITY.
ES2351323B1 (en) 2009-06-26 2011-10-05 Institut Univ. De Ciència I Tecnologia, S.A. LIBRARIES OF N-PHENYL-1-SULFONIL-2-PIRROLIDINACARBOXAMIDS FOR THE DISCOVERY OF PHARMACOS.
ES2354550B1 (en) 2009-06-26 2011-11-15 Institut Univ. De Ciència I Tecnologia, S.A. LIBRARY OF N- (1-PHENYL-2-OXO-3-PIPERIDIL) SULFONAMIDS FOR THE DISCOVERY OF DRUGS.
US20120122920A1 (en) 2009-06-26 2012-05-17 Josep Castells Boliart Libraries of n-substituted-n-phenylethylsulfonamides for drug discovery
US20120122710A1 (en) 2009-07-01 2012-05-17 Josep Castells Boliart Libraries of n-substituted-n-phenylethylsulfonamides for the identification of biological and pharmacological activity
ES2351452B1 (en) 2009-07-01 2011-10-05 Institut Univ. De Ciència I Tecnologia, S.A. LIBRARIES OF N-PHENYL-1-SULFONIL-2-PIRROLIDINACARBOXAMIDS FOR THE IDENTIFICATION OF BIOLOGICAL AND PHARMACOLOGICAL ACTIVITY.
ES2354551B1 (en) 2009-07-01 2011-11-15 Institut Univ. De Ciencia I Tecnologia S.A. LIBRARIES OF N- (1-PHENYL-2-OXO-3-PIPERIDIL) SULFONAMIDS FOR THE IDENTIFICATION OF BIOLOGICAL AND PHARMACOLOGICAL ACTIVITY.

Also Published As

Publication number Publication date
EP2445879A1 (en) 2012-05-02
US20120142930A1 (en) 2012-06-07
US8569507B2 (en) 2013-10-29
WO2010150204A1 (en) 2010-12-29

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