IN2012DN01661A - - Google Patents

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Publication number
IN2012DN01661A
IN2012DN01661A IN1661DEN2012A IN2012DN01661A IN 2012DN01661 A IN2012DN01661 A IN 2012DN01661A IN 1661DEN2012 A IN1661DEN2012 A IN 1661DEN2012A IN 2012DN01661 A IN2012DN01661 A IN 2012DN01661A
Authority
IN
India
Prior art keywords
disclosed
compounds
intended
kits
abstract
Prior art date
Application number
Other languages
English (en)
Inventor
H Alex Brown
Craig W Lindsley
Alex G Waterson
Sarah A Scott
Original Assignee
Univ Vanderbilt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Vanderbilt filed Critical Univ Vanderbilt
Publication of IN2012DN01661A publication Critical patent/IN2012DN01661A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/438The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
IN1661DEN2012 2009-07-24 2010-07-23 IN2012DN01661A (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22849209P 2009-07-24 2009-07-24
PCT/US2010/043045 WO2011011680A1 (en) 2009-07-24 2010-07-23 Isoform selective phospholipase d inhibitors

Publications (1)

Publication Number Publication Date
IN2012DN01661A true IN2012DN01661A (pl) 2015-06-05

Family

ID=43499428

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1661DEN2012 IN2012DN01661A (pl) 2009-07-24 2010-07-23

Country Status (14)

Country Link
US (1) US9127005B2 (pl)
EP (1) EP2456307B1 (pl)
JP (1) JP2013500260A (pl)
KR (1) KR20120090034A (pl)
CN (1) CN102573474A (pl)
AU (1) AU2010275526A1 (pl)
BR (1) BR112012001586A2 (pl)
CA (1) CA2768940C (pl)
IL (1) IL217720A0 (pl)
IN (1) IN2012DN01661A (pl)
MX (1) MX2012001064A (pl)
RU (1) RU2012106657A (pl)
SG (1) SG178102A1 (pl)
WO (1) WO2011011680A1 (pl)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9453017B2 (en) 2011-09-30 2016-09-27 Vanderbilt University Antiviral therapies with phospholipase D inhibitors

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG178102A1 (en) 2009-07-24 2012-03-29 Univ Vanderbilt Isoform selective phospholipase d inhibitors
AU2013359315B2 (en) * 2012-12-11 2016-12-08 Vanderbilt University Methods and compositions comprising Akt inhibitors and/or phospholipase D inhibitors
CA2894843A1 (en) * 2012-12-11 2014-06-19 Vanderbilt University Methods and compositions of treating hiv infection
CN114778844A (zh) * 2022-03-07 2022-07-22 天津市肿瘤医院(天津医科大学肿瘤医院) Pld1作为评估肿瘤患者对于化疗药物敏感性的分子标志物的用途
TW202413374A (zh) * 2022-06-16 2024-04-01 日商日本煙草產業股份有限公司 二氫二𠯤酮化合物及其醫藥用途

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1281502B1 (it) 1995-06-13 1998-02-18 Sardinian Antiviral Research C Impiego di un inibitore non nucleosidico della trascrittasi inversa in associazione con inibitori nucleosidici per il trattamento della
US6187559B1 (en) 1997-08-28 2001-02-13 Novartis Ag Phospholipase D gene
EP1313498A4 (en) 2000-05-25 2004-04-21 Ben-Tsion Williger PHOSPHOLIPASE D EFFECTORS FOR THERAPY AND SCREENING
US6482829B2 (en) * 2000-06-08 2002-11-19 Hoffmann-La Roche Inc. Substituted heterocyclic siprodecane compound active as an antagonist of neurokinin 1 receptor
KR101144889B1 (ko) 2002-09-18 2012-05-14 학교법인 포항공과대학교 포스포리파제 d를 포함하는 펩티드 복합체
CN101128435A (zh) * 2004-12-27 2008-02-20 阿斯利康(瑞典)有限公司 作为代谢型谷氨酸受体激动剂用于治疗神经病学及精神病学病症的吡唑酮化合物
JP2008542192A (ja) 2005-02-23 2008-11-27 アービサー ジャック エル. 増殖の障害の治療用のホノキオール誘導体
MX2008014690A (es) * 2006-05-18 2008-11-27 Hoffmann La Roche Derivados de tiazolo-pirimidina/piridina-urea.
US20100009970A1 (en) 2008-03-19 2010-01-14 Combinatorx (Singapore) Pte. Ltd. Compositions and methods for treatment of viral diseases
WO2010037081A1 (en) 2008-09-29 2010-04-01 Palatin Technologies, Inc. Melanocortin receptor-specific spiro-piperidine compounds
JP6029467B2 (ja) 2009-03-31 2016-11-24 サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング 薬物送達デバイスの本体
CN102459584A (zh) 2009-05-29 2012-05-16 纽约市哥伦比亚大学理事会 用于治疗神经退行性病症的磷脂酶d的调节
SG178102A1 (en) 2009-07-24 2012-03-29 Univ Vanderbilt Isoform selective phospholipase d inhibitors
WO2011019498A1 (en) 2009-07-27 2011-02-17 The Trustees Of Princeton University Inhibition of glycerol-3-phosphate acyltransferase (gpat) and associated enzymes for treatment of viral infections
EP2760447A4 (en) 2011-09-30 2015-10-21 Univ Vanderbilt ANTIVIRAL THERAPIES WITH D PHOSPHOLIPASE INHIBITORS
CA2894843A1 (en) 2012-12-11 2014-06-19 Vanderbilt University Methods and compositions of treating hiv infection
AU2013359315B2 (en) 2012-12-11 2016-12-08 Vanderbilt University Methods and compositions comprising Akt inhibitors and/or phospholipase D inhibitors

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9453017B2 (en) 2011-09-30 2016-09-27 Vanderbilt University Antiviral therapies with phospholipase D inhibitors

Also Published As

Publication number Publication date
KR20120090034A (ko) 2012-08-16
US9127005B2 (en) 2015-09-08
RU2012106657A (ru) 2013-08-27
EP2456307A1 (en) 2012-05-30
EP2456307A4 (en) 2013-01-16
US20120214832A1 (en) 2012-08-23
CN102573474A (zh) 2012-07-11
JP2013500260A (ja) 2013-01-07
WO2011011680A1 (en) 2011-01-27
CA2768940C (en) 2018-03-13
SG178102A1 (en) 2012-03-29
CA2768940A1 (en) 2011-01-27
IL217720A0 (en) 2012-03-29
MX2012001064A (es) 2012-07-17
AU2010275526A1 (en) 2012-03-15
EP2456307B1 (en) 2016-11-02
BR112012001586A2 (pt) 2015-09-01

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