IN2012DN02474A - - Google Patents
Download PDFInfo
- Publication number
- IN2012DN02474A IN2012DN02474A IN2474DEN2012A IN2012DN02474A IN 2012DN02474 A IN2012DN02474 A IN 2012DN02474A IN 2474DEN2012 A IN2474DEN2012 A IN 2474DEN2012A IN 2012DN02474 A IN2012DN02474 A IN 2012DN02474A
- Authority
- IN
- India
- Prior art keywords
- pain
- receptor
- pharmaceutical compositions
- hyperalgesia
- present
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Immunology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pyrane Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27550609P | 2009-08-28 | 2009-08-28 | |
| US39658810P | 2010-05-28 | 2010-05-28 | |
| US40014610P | 2010-07-22 | 2010-07-22 | |
| PCT/US2010/002360 WO2011025541A1 (fr) | 2009-08-28 | 2010-08-27 | Modulateurs des récepteurs de cannabinoïdes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2012DN02474A true IN2012DN02474A (fr) | 2015-08-21 |
Family
ID=43127457
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN2474DEN2012 IN2012DN02474A (fr) | 2009-08-28 | 2010-08-27 |
Country Status (19)
| Country | Link |
|---|---|
| US (6) | US8778950B2 (fr) |
| EP (4) | EP3363788A1 (fr) |
| JP (5) | JP5746698B2 (fr) |
| KR (6) | KR102682216B1 (fr) |
| CN (2) | CN103539785B (fr) |
| AR (1) | AR077991A1 (fr) |
| AU (1) | AU2010286988B2 (fr) |
| BR (1) | BR112012008159A2 (fr) |
| CA (1) | CA2770866C (fr) |
| EA (1) | EA023586B1 (fr) |
| HK (1) | HK1259082A1 (fr) |
| IL (1) | IL218130A (fr) |
| IN (1) | IN2012DN02474A (fr) |
| MX (1) | MX2012002499A (fr) |
| NZ (1) | NZ598288A (fr) |
| SG (3) | SG178907A1 (fr) |
| TW (1) | TWI503316B (fr) |
| WO (1) | WO2011025541A1 (fr) |
| ZA (1) | ZA202205142B (fr) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IN2012DN02474A (fr) * | 2009-08-28 | 2015-08-21 | Arena Pharm Inc | |
| AU2012222149B2 (en) | 2011-02-25 | 2017-06-29 | Arena Pharmaceuticals, Inc. | Cannabinoid receptor modulators |
| US9597340B2 (en) * | 2011-02-25 | 2017-03-21 | Arena Pharmaceuticals, Inc. | Cannabinoid receptor modulators |
| EP2678330A1 (fr) | 2011-02-25 | 2014-01-01 | Arena Pharmaceuticals, Inc. | Formes cristallines et procédés de préparation d'azacycles condensés (modulateurs des récepteurs des cannabinoïdes) |
| ITMI20122221A1 (it) | 2012-12-21 | 2014-06-22 | C4T S C A R L | Nuovi composti del 2,3-diidro-4h-1,3-benzossazin-4-one, metodo per prepararli e forma farmaceutica che li comprende |
| EP2803668A1 (fr) | 2013-05-17 | 2014-11-19 | Boehringer Ingelheim International Gmbh | Nouveau (cyano-dimethyl-methyl)-isoxazoles et - [1,3,4] thiadiazoles |
| JP5983714B2 (ja) * | 2013-11-29 | 2016-09-06 | 大正製薬株式会社 | 含フッ素アミノ酸プロドラッグの結晶形とその製造方法 |
| WO2015095953A1 (fr) | 2013-12-27 | 2015-07-02 | The Centre For Drug Research And Development | Systèmes de liaison contenant un sulfonamide pour conjugués de médicaments |
| ES2905569T3 (es) | 2014-09-17 | 2022-04-11 | Zymeworks Inc | Compuestos citotóxicos y antimitóticos y métodos para utilizarlos |
| WO2016085941A1 (fr) * | 2014-11-25 | 2016-06-02 | Arena Pharmaceuticals, Inc. | Procédés de préparation de modulateurs des récepteurs de cannabinoïdes |
| US10172786B2 (en) | 2014-12-16 | 2019-01-08 | Axim Biotechnologies, Inc. | Oral care composition comprising cannabinoids |
| AU2017249211A1 (en) * | 2016-04-10 | 2018-11-22 | Arena Pharmaceuticals, Inc. | Methods of treatment with selective CB2 receptor agonists |
| CN109689045A (zh) | 2016-05-04 | 2019-04-26 | 因美制药公司 | 大麻素的局部制剂在治疗大疱性表皮松解症和相关结缔组织病症中的用途 |
| WO2018208847A1 (fr) | 2017-05-08 | 2018-11-15 | Arena Pharmaceuticals, Inc. | Compositions et méthodes pour le traitement de la douleur résultant de la maladie inflammatoire chronique de l'intestin |
| US20200078358A1 (en) | 2017-05-08 | 2020-03-12 | Arena Pharmaceuticals, Inc. | Compounds and Methods for Treatment of Visceral Pain |
| WO2019043635A1 (fr) | 2017-09-01 | 2019-03-07 | Richter Gedeon Nyrt. | Composés inhibiteurs de l'activité de d-amino acide oxydase |
| US12357604B2 (en) | 2017-09-22 | 2025-07-15 | Inmed Pharmaceuticals Inc. | Topical formulations of cannabinoids and use thereof in the treatment of pain |
| EP3886845B1 (fr) | 2018-11-28 | 2024-09-04 | Merck Sharp & Dohme LLC | Nouveaux composés de piperazine amide substitués utilisés en tant qu'inhibiteurs de l'indoléamine 2,3-dioxygénase (ido) |
| WO2021047583A1 (fr) * | 2019-09-12 | 2021-03-18 | 四川海思科制药有限公司 | Dérivé de pyrazole tricyclique et sa préparation |
| WO2021047581A1 (fr) * | 2019-09-12 | 2021-03-18 | 四川海思科制药有限公司 | Dérivé d'hexahydrobenzopyrazole et sa préparation |
| JP7620024B2 (ja) | 2020-09-24 | 2025-01-22 | 富士フイルム株式会社 | 複合パターンの製造方法、樹脂組成物、積層体の製造方法、及び、半導体デバイスの製造方法 |
| CN115536648B (zh) * | 2021-06-29 | 2024-09-17 | 深圳开悦生命科技有限公司 | 一类抑制rna解旋酶dhx33的多环化合物及其应用 |
| CN114736173B (zh) * | 2022-05-24 | 2024-06-11 | 无锡捷化医药科技有限公司 | 一种3-（二氟甲基）氧杂环丁烷-3-胺盐酸盐的制备方法 |
| WO2025090133A1 (fr) | 2023-10-23 | 2025-05-01 | Inmed Pharmaceuticals Inc. | Compositions et procédés d'utilisation de composés de cannabinol dans la neuroprotection |
| WO2025090587A1 (fr) | 2023-10-23 | 2025-05-01 | Inmed Pharmaceuticals Inc. | Composés cannabinoïdes et leur utilisation dans le traitement de troubles neuronaux |
Family Cites Families (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3964478B2 (ja) | 1995-06-30 | 2007-08-22 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ヘテロ環含有カルボン酸誘導体及びそれを含有する医薬 |
| YU72201A (sh) | 1999-04-28 | 2005-07-19 | Aventis Pharma Deutschland Gmbh. | Derivati di-aril kiseline kao ppar receptorski ligandi |
| EP1461027A4 (fr) | 2001-12-07 | 2005-09-07 | Univ Virginia Commonwealth | Traitement de la neoplasie |
| SE0300010D0 (sv) | 2003-01-07 | 2003-01-07 | Astrazeneca Ab | Novel Compounds |
| ITMI20041033A1 (it) * | 2004-05-24 | 2004-08-24 | Neuroscienze S C A R L | Composti farmaceutici |
| EP2343302A1 (fr) | 2004-07-12 | 2011-07-13 | Cadila Healthcare Limited | Derives tricycliques de pyrazole comme modulateurs des recepteurs cannabinoides |
| WO2006010379A1 (fr) * | 2004-07-29 | 2006-02-02 | Actelion Pharmaceuticals Ltd. | Nouveaux derives du thiophene utilises comme agents immunosupresseurs |
| FR2875230A1 (fr) * | 2004-09-13 | 2006-03-17 | Sanofi Aventis Sa | Derives de pyrazole condense, leur preparation et leur application en therapeutique |
| DE102004054666A1 (de) | 2004-11-12 | 2006-05-18 | Bayer Cropscience Gmbh | Substituierte Pyrazol-3-carboxamide, Verfahren zur Herstellung und Verwendung als Herbizide und Pflanzenwachstumsregulatoren |
| PE20060949A1 (es) * | 2004-12-23 | 2006-10-11 | Arena Pharm Inc | Derivados fusionados de pirazol como agonistas del receptor de niacina |
| CA2613678A1 (fr) * | 2005-06-02 | 2006-12-07 | Glenmark Pharmaceuticals S.A. | Nouveaux ligands des recepteurs des cannabinoides, compositions pharmaceutiques contenant ces ligands, et procede servant a leur preparation |
| ATE459352T1 (de) | 2006-07-04 | 2010-03-15 | Janssen Pharmaceutica Nv | Benzimidazol-cannabinoid-agonisten mit einer substituierten heterocyclischen gruppe |
| US7928123B2 (en) | 2006-09-25 | 2011-04-19 | Boehringer Ingelheim International Gmbh | Compounds which modulate the CB2 receptor |
| US8481574B2 (en) | 2006-10-12 | 2013-07-09 | Abbott Laboratories | Compounds as cannabinoid receptor ligands |
| WO2008048914A1 (fr) | 2006-10-17 | 2008-04-24 | Boehringer Ingelheim International Gmbh | Composés qui modulent le récepteur cb2 |
| EP2091921A2 (fr) | 2006-11-03 | 2009-08-26 | Glenmark Pharmaceuticals S.A. | Indazoles bicycliques pontes comme ligands de récepteurs cannabinoïdes |
| US8173638B2 (en) | 2006-11-21 | 2012-05-08 | Boehringer Ingelheim International Gmbh | Compounds which modulate the CB2 receptor |
| US20080161340A1 (en) | 2006-12-20 | 2008-07-03 | Cara Therapeutics, Inc. | Tetrahydroquinilinones, tetrahydronaphthyridones and derivatives thereof |
| WO2008085302A1 (fr) | 2006-12-20 | 2008-07-17 | Merck & Co., Inc. | Analogues de l'imidazopyridine en tant que modulateurs du récepteur de cb2, utilisables pour le traitement de la douleur et des maladies respiratoires et non respiratoires |
| US20080214537A1 (en) | 2007-03-02 | 2008-09-04 | Cara Therapeutics, Inc. | Bridged phenanthridines |
| US8193369B2 (en) | 2007-03-30 | 2012-06-05 | Janssen Pharmaceutica Nv | Benzimidazole cannabinoid agonists |
| WO2008157500A1 (fr) | 2007-06-17 | 2008-12-24 | Kalypsys, Inc. | Modulateurs du récepteur cannabinoïde à base d'aminoquinazoline pour le traitement de maladies |
| CN101686989B (zh) | 2007-06-21 | 2016-10-19 | 卡拉治疗学股份有限公司 | 取代的咪唑并杂环 |
| US8338623B2 (en) | 2007-07-09 | 2012-12-25 | Abbvie Inc. | Compounds as cannabinoid receptor ligands |
| US7943658B2 (en) | 2007-07-23 | 2011-05-17 | Bristol-Myers Squibb Company | Indole indane amide compounds useful as CB2 agonists and method |
| EP2203171A2 (fr) | 2007-08-21 | 2010-07-07 | Merck Sharp & Dohme Corp. | Ligands de récepteur cb2 pour le traitement de la douleur |
| UA104010C2 (en) | 2008-12-18 | 2013-12-25 | Эли Лилли Энд Компани | Purine compounds |
| US7741350B1 (en) | 2009-01-28 | 2010-06-22 | Cara Therapeutics, Inc. | Bicyclic pyrazolo-heterocycles |
| WO2010088050A2 (fr) | 2009-01-28 | 2010-08-05 | Cara Therapeutics, Inc. | Hétérocycles pyrazolo bicycliques |
| IN2012DN02474A (fr) | 2009-08-28 | 2015-08-21 | Arena Pharm Inc | |
| AU2012222149B2 (en) * | 2011-02-25 | 2017-06-29 | Arena Pharmaceuticals, Inc. | Cannabinoid receptor modulators |
| US9597340B2 (en) * | 2011-02-25 | 2017-03-21 | Arena Pharmaceuticals, Inc. | Cannabinoid receptor modulators |
| EP2678330A1 (fr) * | 2011-02-25 | 2014-01-01 | Arena Pharmaceuticals, Inc. | Formes cristallines et procédés de préparation d'azacycles condensés (modulateurs des récepteurs des cannabinoïdes) |
-
2010
- 2010-08-27 IN IN2474DEN2012 patent/IN2012DN02474A/en unknown
- 2010-08-27 TW TW099128986A patent/TWI503316B/zh active
- 2010-08-27 KR KR1020227032376A patent/KR102682216B1/ko active Active
- 2010-08-27 AU AU2010286988A patent/AU2010286988B2/en not_active Ceased
- 2010-08-27 EP EP18150186.7A patent/EP3363788A1/fr not_active Withdrawn
- 2010-08-27 KR KR1020207001281A patent/KR20200008045A/ko not_active Ceased
- 2010-08-27 EP EP22159802.2A patent/EP4036082A1/fr active Pending
- 2010-08-27 CA CA2770866A patent/CA2770866C/fr active Active
- 2010-08-27 SG SG2012013967A patent/SG178907A1/en unknown
- 2010-08-27 SG SG10201901293RA patent/SG10201901293RA/en unknown
- 2010-08-27 CN CN201310463585.6A patent/CN103539785B/zh active Active
- 2010-08-27 EP EP22160034.9A patent/EP4036089A1/fr not_active Withdrawn
- 2010-08-27 US US13/392,074 patent/US8778950B2/en active Active
- 2010-08-27 EP EP10757325A patent/EP2470508A1/fr not_active Withdrawn
- 2010-08-27 AR ARP100103145A patent/AR077991A1/es active IP Right Grant
- 2010-08-27 KR KR1020187029637A patent/KR20180115807A/ko not_active Ceased
- 2010-08-27 EA EA201270336A patent/EA023586B1/ru unknown
- 2010-08-27 JP JP2012526732A patent/JP5746698B2/ja not_active Expired - Fee Related
- 2010-08-27 KR KR1020217014027A patent/KR20210057213A/ko not_active Ceased
- 2010-08-27 KR KR1020177016103A patent/KR20170072358A/ko not_active Ceased
- 2010-08-27 WO PCT/US2010/002360 patent/WO2011025541A1/fr not_active Ceased
- 2010-08-27 KR KR1020127007857A patent/KR101749778B1/ko not_active Expired - Fee Related
- 2010-08-27 SG SG10201404925TA patent/SG10201404925TA/en unknown
- 2010-08-27 BR BR112012008159A patent/BR112012008159A2/pt not_active Application Discontinuation
- 2010-08-27 NZ NZ598288A patent/NZ598288A/en not_active IP Right Cessation
- 2010-08-27 MX MX2012002499A patent/MX2012002499A/es active IP Right Grant
- 2010-08-27 CN CN201080049159.2A patent/CN102596913B/zh active Active
-
2012
- 2012-02-15 IL IL218130A patent/IL218130A/en active IP Right Grant
- 2012-09-14 US US13/616,918 patent/US9944606B2/en active Active
-
2015
- 2015-05-08 JP JP2015095753A patent/JP2015145423A/ja not_active Withdrawn
-
2017
- 2017-10-26 JP JP2017207036A patent/JP2018021074A/ja not_active Withdrawn
-
2018
- 2018-03-06 US US15/912,700 patent/US20180354907A1/en not_active Abandoned
-
2019
- 2019-01-29 HK HK19101582.1A patent/HK1259082A1/en unknown
- 2019-09-24 US US16/580,697 patent/US11214548B2/en active Active
- 2019-12-06 JP JP2019221000A patent/JP2020033387A/ja not_active Withdrawn
-
2020
- 2020-09-18 US US17/024,752 patent/US11746091B2/en active Active
-
2021
- 2021-10-22 JP JP2021173078A patent/JP2022009408A/ja not_active Withdrawn
- 2021-11-08 US US17/520,952 patent/US20220306586A1/en not_active Abandoned
-
2022
- 2022-05-10 ZA ZA2022/05142A patent/ZA202205142B/en unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ZA202205142B (en) | Cannabinoid receptor modulators | |
| WO2021071788A3 (fr) | Compositions oligonucléotidiques et leurs procédés d'utilisation | |
| WO2020227691A3 (fr) | Compositions oligonucléotidiques et leurs procédés d'utilisation | |
| PH12018502028A1 (en) | Allosteric modulators of nicotinic acetylcholine receptors | |
| UA101493C2 (ru) | Производные азетидина и циклобутана как ингибиторы jak | |
| MY159575A (en) | Dihydroorotate dehydrogenase inhibitors | |
| MY165767A (en) | Crystalline forms and processes for the preparation of condensed azacycles (cannabinoid receptor modulators) | |
| MX2010001446A (es) | Derivados de 6-amino-pirimidina-4-carboxamida y compuestos relacionados que se enlazan a los receptores para esfingosina 1-fosfato (s1p) para el tratamiento de esclerosis multiple. | |
| PH12017500841B1 (en) | 2-amino-6-(difluoromethyl)- 5,5-difluoro-6-phenyl-3,4,5,6-tetrahydropyridines as bace1 inhibitors | |
| MX2011012409A (es) | Metodos y composiciones de endoxifeno en el tratamiento de enfermedades mamiferas. | |
| MX2013009226A (es) | Polipeptidos interleuquina- 2 mutantes. | |
| PH12017501043A1 (en) | 2-amino-5,5-difluoro-6-(fluoromethyl)-6-phenyl-3,4,5,6-tetrahydropyridines as bace1 inhibitors | |
| MY152282A (en) | Compositions and methods for use antibodies against sclerostin | |
| IN2013CN01340A (fr) | ||
| TN2013000362A1 (en) | Benzodioxane inhibitors of leukotriene production | |
| NZ603789A (en) | Heteroaryl compounds and methods of use thereof | |
| MY187450A (en) | Heteroaryl amides as inhibitors of protein aggregation | |
| MX2017006048A (es) | 2-amino-3,5-difluoro-3,6-dimetil-6-fenil-3,4,5,6-tetrahidropiridi nas en calidad de inhibidores de bace1 para tratar enfermedad de alzheimer. | |
| MX2012004548A (es) | Nuevas composiciones para prevenir y/o tratar transtornos degenerativos del sistema nervioso central. | |
| MX336711B (es) | Inhibidores de catecol o-metil transferasa y su uso en el tratamiento de transtornos psicoticos. | |
| MX343376B (es) | Anticuerpos humanizados que tienen como objetivo el dominio ec1 de cadherina-11 y composiciones y metodos relacionados. | |
| MX2012006206A (es) | Preparaciones combinacion comprendiendo exosomas y corticosteroide. | |
| MX2023009372A (es) | Proceso para la preparacion de compuestos enlazantes de farmaco. | |
| MX348957B (es) | Derivados de imidazol azabiciclicos sustituidos utiles como moduladores del receptor del canal 8 (subfamilia melastatina) del potencial de receptor transitorio. | |
| WO2014052179A3 (fr) | Composition de soin de la peau à rincer contenant des tensioactifs de type alkylamidopropylbétaïnes |