IN2013MN02414A - - Google Patents
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- Publication number
- IN2013MN02414A IN2013MN02414A IN2414MUN2013A IN2013MN02414A IN 2013MN02414 A IN2013MN02414 A IN 2013MN02414A IN 2414MUN2013 A IN2414MUN2013 A IN 2414MUN2013A IN 2013MN02414 A IN2013MN02414 A IN 2013MN02414A
- Authority
- IN
- India
- Prior art keywords
- benzothiazinethione
- derivatives
- formula
- significant effect
- mycobacterium tuberculosis
- Prior art date
Links
- YWLASNQCODQVHJ-UHFFFAOYSA-N 1-sulfanylidene-2h-1$l^{4},2-benzothiazine Chemical class C1=CC=C2S(=S)NC=CC2=C1 YWLASNQCODQVHJ-UHFFFAOYSA-N 0.000 abstract 2
- 241000187479 Mycobacterium tuberculosis Species 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
- C07D279/08—1,3-Thiazines; Hydrogenated 1,3-thiazines condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
- C07D491/113—Spiro-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pulmonology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201110139840.2A CN102276598B (zh) | 2011-05-27 | 2011-05-27 | 苯并噻嗪硫酮衍生物及其制备方法和用途 |
| PCT/CN2011/075750 WO2012162912A1 (fr) | 2011-05-27 | 2011-06-15 | Dérivés de la benzothiazine thione et leurs procédés de préparation et leurs utilisations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2013MN02414A true IN2013MN02414A (fr) | 2015-06-12 |
Family
ID=45102383
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN2414MUN2013 IN2013MN02414A (fr) | 2011-05-27 | 2011-06-15 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20140303152A1 (fr) |
| EP (1) | EP2719691A1 (fr) |
| CN (1) | CN102276598B (fr) |
| IN (1) | IN2013MN02414A (fr) |
| RU (1) | RU2013157860A (fr) |
| WO (1) | WO2012162912A1 (fr) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103508980B (zh) * | 2012-06-14 | 2016-07-06 | 四川大学 | 苯并噻嗪-4-酮衍生物及其制备方法和用途 |
| WO2014014845A1 (fr) | 2012-07-18 | 2014-01-23 | Vertex Pharmaceuticals Incorporated | Thérapie combinée comprenant de la 1-éthyl-3[5-[-2-{1-hydroxy-1-méthyl-éthyl}pyrimidin-5-yl]-7-(tétrahydrofuran-2-yl}-1h-benzimidazol-2-yl]urée et ses dérivés pour traiter des maladies mycobactériennes |
| CN104211708B (zh) * | 2013-05-29 | 2018-08-24 | 中国医学科学院药物研究所 | 苯并噁嗪酮衍生物及其作为抗菌剂的应用 |
| US9481683B2 (en) * | 2014-06-09 | 2016-11-01 | University Of Notre Dame Du Lac | 1,3-benzothiazinone sulfoxide and sulfone compounds |
| CN105294597B (zh) * | 2015-11-03 | 2017-11-24 | 华东师范大学 | 苯并噻嗪类衍生物及其合成方法和应用 |
| CN110312725B (zh) * | 2016-09-22 | 2022-03-11 | 莱比尼兹自然研究和感染生物学研究所协会汉斯诺尔研究所(Hki) | 新型抗菌化合物，其在哺乳动物感染治疗中的应用及新的代谢机制 |
| CN108456204B (zh) * | 2017-02-17 | 2023-05-26 | 四川大学 | 苯并噻嗪衍生物及其制备方法和用途 |
| CN108947952B (zh) * | 2017-05-24 | 2021-09-21 | 中国医学科学院药物研究所 | 2-取代氨基-5-三氟甲基-8-硝基苯并（硫代）吡喃-4-酮类化合物及其制备方法和用途 |
| CN114957232B (zh) * | 2021-05-28 | 2023-06-30 | 四川大学 | 一种苯并二氢恶嗪类化合物及其制备方法和抗结核的用途 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2006343832B2 (en) * | 2006-05-24 | 2011-07-21 | Leibniz Institute For Natural Product Research And Infection Biology E.V. Hans-Knoll-Institut (Hki) | New benzothiazinone derivatives and their use as antibacterial agents |
| EP2020406A1 (fr) * | 2007-07-16 | 2009-02-04 | Leibniz-Institut für Naturstoff-Forschung und Infektionsbiologie e.V. Hans-Knöll-Institut | Nouveaux composés antimicrobiens, leur synthèse et utilisation pour le traitement des infections liées aux mammifères |
-
2011
- 2011-05-27 CN CN201110139840.2A patent/CN102276598B/zh not_active Expired - Fee Related
- 2011-06-15 WO PCT/CN2011/075750 patent/WO2012162912A1/fr not_active Ceased
- 2011-06-15 US US14/234,501 patent/US20140303152A1/en not_active Abandoned
- 2011-06-15 RU RU2013157860/04A patent/RU2013157860A/ru unknown
- 2011-06-15 IN IN2414MUN2013 patent/IN2013MN02414A/en unknown
- 2011-06-15 EP EP11866737.7A patent/EP2719691A1/fr not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2012162912A1 (fr) | 2012-12-06 |
| EP2719691A1 (fr) | 2014-04-16 |
| CN102276598A (zh) | 2011-12-14 |
| US20140303152A1 (en) | 2014-10-09 |
| RU2013157860A (ru) | 2015-07-10 |
| CN102276598B (zh) | 2014-11-05 |
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