IN2013MU01782A - - Google Patents

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Publication number
IN2013MU01782A
IN2013MU01782A IN1782MU2013A IN2013MU01782A IN 2013MU01782 A IN2013MU01782 A IN 2013MU01782A IN 1782MU2013 A IN1782MU2013 A IN 1782MU2013A IN 2013MU01782 A IN2013MU01782 A IN 2013MU01782A
Authority
IN
India
Prior art keywords
rasagiline
enantiomer
disease
salts
pharmaceutical compositions
Prior art date
Application number
Other languages
English (en)
Inventor
Sushrut Krishnaji Kulkarni
Pavak Rajnikanth Mehta
Ritesh Kapoor
Original Assignee
Cadila Healthcare Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cadila Healthcare Ltd filed Critical Cadila Healthcare Ltd
Priority to IN1782MU2013 priority Critical patent/IN2013MU01782A/en
Priority to PCT/IN2014/000336 priority patent/WO2014192022A1/fr
Publication of IN2013MU01782A publication Critical patent/IN2013MU01782A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IN1782MU2013 2013-05-20 2014-05-20 IN2013MU01782A (fr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
IN1782MU2013 IN2013MU01782A (fr) 2013-05-20 2014-05-20
PCT/IN2014/000336 WO2014192022A1 (fr) 2013-05-20 2014-05-20 Compositions pharmaceutiques de rasagiline

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN1782MU2013 IN2013MU01782A (fr) 2013-05-20 2014-05-20

Publications (1)

Publication Number Publication Date
IN2013MU01782A true IN2013MU01782A (fr) 2015-06-26

Family

ID=51300794

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1782MU2013 IN2013MU01782A (fr) 2013-05-20 2014-05-20

Country Status (2)

Country Link
IN (1) IN2013MU01782A (fr)
WO (1) WO2014192022A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202430137A (zh) * 2023-01-19 2024-08-01 大陸商上海雲晟研新生物科技有限公司 甲磺酸雷沙吉蘭口溶膜組合物、其製備方法及用途

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL111240A (en) * 1993-10-18 2001-10-31 Teva Pharma Salts of r(+) - enantiomers of n- propargyl-1-aminoindan and pharmaceutical compositions comprising them
EP1778196A4 (fr) * 2004-07-26 2008-12-17 Teva Pharma Dosages pharmaceutiques contenant de la rasagiline
EP1892233A1 (fr) * 2006-08-18 2008-02-27 Ratiopharm GmbH De nouveaux sels de la substance active rasagiline
CN1911211B (zh) * 2006-08-25 2010-04-14 重庆医药工业研究院有限责任公司 雷沙吉兰口服固体制剂
EP1987816A1 (fr) * 2007-04-30 2008-11-05 Ratiopharm GmbH Adsorbate d'un sel de rasagiline en combinaison avec un agent inactive soluble dans l'eau
WO2009122301A2 (fr) * 2008-03-31 2009-10-08 Actavis Group Ptc Ehf Particules de mésylate de rasagiline et leur procédé de préparation
AR074637A1 (es) * 2008-07-18 2011-02-02 Medichem Sa Formas de sal de adicion acida de r-(+)-n-propargil-1-aminoindano (es decir , base de rasagilina), un compuesto de formula (1), procesos para prepararlos y aislarlos y usos de los mismos
WO2010111264A2 (fr) * 2009-03-24 2010-09-30 Dr. Reddy's Laboratories Ltd. Préparations de rasagiline
DK2451771T3 (da) * 2009-07-09 2014-09-08 Ratiopharm Gmbh Salte af rasagilin og farmaceutiske fremstillingsmåder heraf
WO2011010324A1 (fr) * 2009-07-23 2011-01-27 Alkem Laboratories Ltd. Compositions pharmaceutiques orales stables comprenant de la rasagiline et procédé
US20120269871A1 (en) * 2009-12-30 2012-10-25 Actavis Group Ptc Ehf Solid state forms of rasagiline salts
CN102791258B (zh) * 2010-02-03 2018-05-08 图必制药公司 雷沙吉兰的延长释放制剂及其用途
WO2011121607A2 (fr) * 2010-03-29 2011-10-06 Cadila Healthcare Limited Composé de rasagiline et sels pharmaceutiquement acceptables de celui-ci
EP2389927A1 (fr) * 2010-05-30 2011-11-30 Abdi Ibrahim Ilac Sanayi ve Ticaret Anonim Sirketi Formulations pharmaceutiques de rasagiline
EP2705021A2 (fr) * 2011-05-04 2014-03-12 Cadila Healthcare Limited Rasagiline et ses sels pharmaceutiquement acceptables
ES2502140T1 (es) * 2013-02-06 2014-10-02 Galenicum Health S.L. Comprimidos de liberación inmediata de rasagilina hemitartrato

Also Published As

Publication number Publication date
WO2014192022A1 (fr) 2014-12-04

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