IN2014DN07129A - - Google Patents

Info

Publication number
IN2014DN07129A
IN2014DN07129A IN7129DEN2014A IN2014DN07129A IN 2014DN07129 A IN2014DN07129 A IN 2014DN07129A IN 7129DEN2014 A IN7129DEN2014 A IN 7129DEN2014A IN 2014DN07129 A IN2014DN07129 A IN 2014DN07129A
Authority
IN
India
Prior art keywords
fluoroalkyl
bis
pyrazol
carboxylic acid
acid derivatives
Prior art date
Application number
Inventor
Sergii Pazenok
Norbert Lui
Jean Pierre Vors
Frédéric Leroux
Florence Giornal
Original Assignee
Bayer Cropscience Ag
Centre Nat Rech Scient
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag, Centre Nat Rech Scient filed Critical Bayer Cropscience Ag
Publication of IN2014DN07129A publication Critical patent/IN2014DN07129A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/30Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

The invention relates to novel 3 5 bis(fluoroalkyl) pyrazol 4 carboxylic acid derivatives and to a method for producing 3 5 bis(fluoroalkyl) pyrazol 4 carboxylic acid derivatives and 3 5 bis(fluoroalkyl) pyrazoles.
IN7129DEN2014 2012-02-01 2013-01-31 IN2014DN07129A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12356001.3A EP2623496A1 (en) 2012-02-01 2012-02-01 Method for producing 3,5-bis(fluoralkyl)-pyrazol-4-carboxylic acid derivatives and 3,5-bis(fluoralkyl)-pyrazoles
PCT/EP2013/051930 WO2013113829A1 (en) 2012-02-01 2013-01-31 Method for producing 3,5-bis(fluoroalkyl)-pyrazol-4-carboxylic acid derivatives and 3,5-bis(fluoroalkyl)-pyrazoles

Publications (1)

Publication Number Publication Date
IN2014DN07129A true IN2014DN07129A (en) 2015-04-24

Family

ID=47624109

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7129DEN2014 IN2014DN07129A (en) 2012-02-01 2013-01-31

Country Status (13)

Country Link
US (2) US9309202B2 (en)
EP (2) EP2623496A1 (en)
JP (1) JP6155283B2 (en)
KR (1) KR101861116B1 (en)
CN (1) CN104245676B (en)
BR (1) BR112014019036B1 (en)
DK (1) DK2809653T3 (en)
ES (1) ES2647348T3 (en)
IL (1) IL233926B (en)
IN (1) IN2014DN07129A (en)
MX (1) MX362689B (en)
TW (1) TWI609006B (en)
WO (1) WO2013113829A1 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102233203B1 (en) * 2013-05-22 2021-03-26 바이엘 크롭사이언스 악티엔게젤샤프트 Method for the production of 3,5-bis(fluoroalkyl)pyrazole derivatives
TWI647215B (en) * 2013-11-11 2019-01-11 德商拜耳作物科學股份有限公司 Method for preparing 3,5-dihaloalkylpyrazole derivatives from α,α-dihalamine
EP3015458A1 (en) * 2014-11-03 2016-05-04 Bayer CropScience AG Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines
EP3122727B1 (en) * 2014-03-24 2018-01-31 Bayer CropScience Aktiengesellschaft Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from alpha , alpha-dihaloamines and ketimines
CN106458918B (en) * 2014-06-11 2019-07-09 拜耳作物科学股份公司 Process for the preparation of 3,5-bis(haloalkyl)pyrazoles via acylation of ketimines
BR112016028702B1 (en) * 2014-06-11 2021-05-04 Bayer Cropscience Aktiengesellschaft process for preparing 3,5-bis(haloalkyl)pyrazole derivatives via acylation of hydrazones
BR112017015061B1 (en) 2015-02-11 2022-09-27 Basf Se PESTICIDE MIXTURE COMPRISING AN ACTIVE COMPOUND OF FORMULA IA AND BROFLANILIDE
KR20180021798A (en) * 2015-06-26 2018-03-05 바이엘 크롭사이언스 악티엔게젤샤프트 Process for preparing substituted pyrazoles having haloalkoxy- and haloalkylthio groups from?,? -haloalkylamines and ketimines
US20210253533A1 (en) 2018-06-18 2021-08-19 Bayer Aktiengesellschaft Disubstituted 5(3)-pyrazole carboxylates and a process for their preparation from enolates and fluoroalkylaminoreagents (far) reagents
EP3953336A4 (en) * 2019-04-06 2023-05-03 Trinapco, Inc SULFONYLDIAZOLES AND N-(FLUOROSULFONYL)AZOLES AND PROCESS FOR THEIR PRODUCTION

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2004460A6 (en) * 1987-07-29 1989-01-01 Consejo Superior Investigacion 3,5-Di:halomethyl pyrazole deriv. prepn.
JP3533134B2 (en) * 1999-02-15 2004-05-31 三井化学株式会社 Fluorinating agents and their production and use
JP2001192369A (en) * 2000-01-12 2001-07-17 Mitsui Chemicals Inc Method of producing fluorine-containing heterocyclic aromatic compound and novel pyrazole ping compound
DE10215292A1 (en) 2002-02-19 2003-08-28 Bayer Cropscience Ag New N-biphenylyl-1-methyl-3-(di- or trifluoromethyl)-1H-pyrazole-4-carboxamides, useful as microbicides, especially fungicides and bactericides for protection of plants or materials such as wood
US7842693B2 (en) * 2002-06-12 2010-11-30 Chemocentryx, Inc. Substituted piperazines
DE10349500A1 (en) 2003-10-23 2005-06-02 Bayer Cropscience Ag A process for producing 2-dihaloacyl-3-amino-acrylic acid esters and 3-dihalomethyl-pyrazole-4-carboxylic acid esters
TW200738701A (en) * 2005-07-26 2007-10-16 Du Pont Fungicidal carboxamides
GB0526044D0 (en) * 2005-12-21 2006-02-01 Syngenta Ltd Novel herbicides
WO2008013622A2 (en) 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
DE102006039909A1 (en) 2006-08-25 2008-03-13 Bayer Cropscience Ag Process for the preparation of 3-dihalomethyl-pyrazole-4-carboxylic acid derivatives
WO2008091594A2 (en) * 2007-01-24 2008-07-31 E. I. Du Pont De Nemours And Company Fungicidal mixtures
EP2133341A1 (en) 2008-02-25 2009-12-16 Bayer CropScience AG Method for regioselective synthesis of 1-alkyl-3-haloalkyl-1-pyrazol-4-carbonic acid derivatives
EP2100883A1 (en) 2008-03-10 2009-09-16 Bayer CropScience AG Method for regioselective synthesis of 1-alkyl-3-haloalkyl-1-pyrazol-4-carbonic acid derivatives
JP2010083763A (en) * 2008-09-29 2010-04-15 Mitsui Chemicals Inc Pyrazole derivative, method of producing the same, and bactericide

Also Published As

Publication number Publication date
US9309202B2 (en) 2016-04-12
IL233926A0 (en) 2014-09-30
JP2015511227A (en) 2015-04-16
US20160185731A1 (en) 2016-06-30
KR20140128344A (en) 2014-11-05
MX2014009203A (en) 2014-11-12
TWI609006B (en) 2017-12-21
US20150011779A1 (en) 2015-01-08
DK2809653T3 (en) 2017-11-27
ES2647348T3 (en) 2017-12-21
JP6155283B2 (en) 2017-06-28
IL233926B (en) 2018-08-30
MX362689B (en) 2019-02-01
CN104245676A (en) 2014-12-24
EP2809653B1 (en) 2017-08-16
EP2809653A1 (en) 2014-12-10
CN104245676B (en) 2016-09-21
WO2013113829A1 (en) 2013-08-08
US10035773B2 (en) 2018-07-31
BR112014019036A2 (en) 2017-08-22
BR112014019036B1 (en) 2019-10-08
TW201336826A (en) 2013-09-16
KR101861116B1 (en) 2018-05-25
EP2623496A1 (en) 2013-08-07

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