IN2014DN08417A - - Google Patents

Info

Publication number
IN2014DN08417A
IN2014DN08417A IN8417DEN2014A IN2014DN08417A IN 2014DN08417 A IN2014DN08417 A IN 2014DN08417A IN 8417DEN2014 A IN8417DEN2014 A IN 8417DEN2014A IN 2014DN08417 A IN2014DN08417 A IN 2014DN08417A
Authority
IN
India
Prior art keywords
formulations
insulin
rapid acting
absorption
mixing
Prior art date
Application number
Inventor
Roderike Pohl
Robert Hauser
Ming Li
Bryan R Wilson
Original Assignee
Biodel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biodel Inc filed Critical Biodel Inc
Publication of IN2014DN08417A publication Critical patent/IN2014DN08417A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/28Insulins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)

Abstract

Compositions and methods for modulating injection site pain associated with rapid acting injectable insulin formulations have been developed for subcutaneous injection. The formulations contain insulin in combination with a zinc chelator such as ethylenediaminetetraacetic acid ('EDTA') a dissolution/stabilization agent such as citric acid a magnesium salt and optionally additional excipients. New presentations include rapid acting concentrated insulin formulations and a way to enhance the absorption of commercially available rapid acting analog formulations by mixing them with a vial containing dry powder excipients that accelerate their absorption. Devices for mixing excipient and insulin together at the time of administration while minimizing residence time of the mixture are also described.
IN8417DEN2014 2012-04-16 2013-04-16 IN2014DN08417A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201261624844P 2012-04-16 2012-04-16
US201261704066P 2012-09-21 2012-09-21
US13/826,806 US9381247B2 (en) 2012-04-16 2013-03-14 Magnesium compositions for modulating the pharmacokinetics and pharmacodynamics of insulin and insulin analogs, and injection site pain
PCT/US2013/036742 WO2013158618A1 (en) 2012-04-16 2013-04-16 Magnesium compositions for modulating the pharmacokinetics and pharmacodynamics of insulin and insulin analogs, and injection site pain

Publications (1)

Publication Number Publication Date
IN2014DN08417A true IN2014DN08417A (en) 2015-05-08

Family

ID=48326401

Family Applications (1)

Application Number Title Priority Date Filing Date
IN8417DEN2014 IN2014DN08417A (en) 2012-04-16 2013-04-16

Country Status (25)

Country Link
US (1) US9381247B2 (en)
EP (2) EP2838506B1 (en)
JP (2) JP6422855B2 (en)
KR (1) KR101966484B1 (en)
CN (1) CN104394847A (en)
AU (1) AU2013249495B2 (en)
CA (1) CA2869883A1 (en)
CY (1) CY1123825T1 (en)
DK (1) DK2838506T3 (en)
ES (1) ES2854874T3 (en)
HK (2) HK1207577A1 (en)
HR (1) HRP20210417T1 (en)
HU (1) HUE053303T2 (en)
IL (1) IL234987A0 (en)
IN (1) IN2014DN08417A (en)
LT (1) LT2838506T (en)
MX (1) MX2014012245A (en)
PL (1) PL2838506T3 (en)
PT (1) PT2838506T (en)
RS (1) RS61533B1 (en)
RU (1) RU2014145846A (en)
SG (1) SG11201406491PA (en)
SI (1) SI2838506T1 (en)
WO (1) WO2013158618A1 (en)
ZA (1) ZA201407410B (en)

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Publication number Priority date Publication date Assignee Title
CN104902922B (en) 2012-11-13 2017-12-12 阿道恰公司 Rapid-acting insulin preparations comprising substituted anionic compounds
KR102351111B1 (en) * 2014-01-13 2022-01-14 써멀린 다이어비티즈, 엘엘씨 Rapid action insulin formulations and pharmaceutical delivery systems
WO2015120457A1 (en) * 2014-02-10 2015-08-13 Biodel Inc. Stabilized ultra-rapid-acting insulin formulations
TWI685348B (en) * 2014-05-08 2020-02-21 美國禮來大藥廠 Rapid-acting insulin compositions
WO2016007935A2 (en) 2014-07-10 2016-01-14 Companion Medical, Inc. Medicine administering system including injection pen and companion device
TW201630622A (en) 2014-12-16 2016-09-01 美國禮來大藥廠 Fast-acting insulin composition
KR20170106373A (en) * 2015-01-20 2017-09-20 케이스 웨스턴 리저브 유니버시티 Insulin analogs with selective signaling properties and reduced mitogenesis promotion
JO3749B1 (en) * 2015-08-27 2021-01-31 Lilly Co Eli Fast acting insulin formulations
US10864327B2 (en) 2016-01-29 2020-12-15 Companion Medical, Inc. Automatic medication delivery tracking
GB201607918D0 (en) 2016-05-06 2016-06-22 Arecor Ltd Novel formulations
JP2019529506A (en) 2016-09-29 2019-10-17 アレコル リミテッド New formulation
GB201707189D0 (en) * 2017-05-05 2017-06-21 Arecor Ltd Novel formulations
CN110662551B (en) 2017-06-01 2023-07-18 伊莱利利公司 Rapid-acting insulin composition
US11484657B2 (en) 2017-06-09 2022-11-01 Medtronic Minimed, Inc. Intelligent medication delivery systems and methods
US11568975B2 (en) 2017-10-12 2023-01-31 Medtronic Minimed, Inc. Intelligent medication delivery systems and methods for dose recommendation and management
JP7512203B2 (en) 2017-12-12 2024-07-08 ビッグフット バイオメディカル インコーポレイテッド TREATMENT SUPPORT INFORMATION AND/OR TRACKING DEVICE AND ASSOCIATED METHODS AND SYSTEMS - Patent application
US11083852B2 (en) 2017-12-12 2021-08-10 Bigfoot Biomedical, Inc. Insulin injection assistance systems, methods, and devices
US11197964B2 (en) 2017-12-12 2021-12-14 Bigfoot Biomedical, Inc. Pen cap for medication injection pen having temperature sensor
US11116899B2 (en) 2017-12-12 2021-09-14 Bigfoot Biomedical, Inc. User interface for diabetes management systems and devices
US10987464B2 (en) 2017-12-12 2021-04-27 Bigfoot Biomedical, Inc. Pen cap for insulin injection pens and associated methods and systems
US11464459B2 (en) 2017-12-12 2022-10-11 Bigfoot Biomedical, Inc. User interface for diabetes management systems including flash glucose monitor
US11077243B2 (en) 2017-12-12 2021-08-03 Bigfoot Biomedical, Inc. Devices, systems, and methods for estimating active medication from injections
US12357562B2 (en) 2018-04-04 2025-07-15 Arecor Limited Injection pen system for the delivery of an insulin compound
US11664107B2 (en) 2018-05-08 2023-05-30 Medtronic Minimed, Inc. Intelligent medication delivery systems and methods using a prescription-regulated software application
US10898653B2 (en) 2018-05-08 2021-01-26 Companion Medical, Inc. Intelligent medication delivery systems and methods for dose setting and dispensing monitoring
USD893020S1 (en) 2018-05-11 2020-08-11 Companion Medical, Inc. Injection pen
USD892819S1 (en) 2018-06-20 2020-08-11 Companion Medical, Inc. Display screen with graphical user interface
US11587663B2 (en) 2018-06-20 2023-02-21 Medtronic Minimed, Inc. Intelligent medication delivery systems and methods for medicine dose calculation and reporting
WO2019243627A1 (en) 2018-06-23 2019-12-26 Adocia Device for injecting an insulin solution
FR3083985A1 (en) 2018-07-23 2020-01-24 Adocia DEVICE FOR INJECTING AN INSULIN SOLUTION (S)
FR3083984A1 (en) 2018-07-23 2020-01-24 Adocia DEVICE FOR INJECTING AN INSULIN SOLUTION (S)
US12205699B1 (en) 2018-10-30 2025-01-21 Bigfoot Biomedical, Inc. Method of pairing therapy devices using shared secrets, and related systems, methods and devices
US11948671B2 (en) 2019-04-11 2024-04-02 Medtronic Minimed, Inc. Intelligent accessories for medicine dispensing device
CN116847869A (en) * 2020-10-08 2023-10-03 美商玛丽莫里斯博士联合有限责任公司 Methods and compositions for treating and preventing type 1 diabetes
US11701473B2 (en) 2021-06-23 2023-07-18 Medtronic Minimed, Inc. Reusable injection pens

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US20080096800A1 (en) 2004-03-12 2008-04-24 Biodel, Inc. Rapid mucosal gel or film insulin compositions
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US20080090753A1 (en) 2004-03-12 2008-04-17 Biodel, Inc. Rapid Acting Injectable Insulin Compositions
EP2543249B1 (en) 2007-02-17 2018-05-23 President and Fellows of Harvard College Compositions and method for tissue preservation
TWI394580B (en) 2008-04-28 2013-05-01 Halozyme Inc Super fast-acting insulin compositions
US9060927B2 (en) * 2009-03-03 2015-06-23 Biodel Inc. Insulin formulations for rapid uptake
FR2943538B1 (en) * 2009-03-27 2011-05-20 Adocia QUICK ACTION FORMULATION OF RECOMBINANT HUMAN INSULIN
CA2805031A1 (en) 2010-07-07 2012-01-12 Biodel, Inc. Compositions and methods for modulating the pharmacokinetics and pharmacodynamics of insulin

Also Published As

Publication number Publication date
ES2854874T3 (en) 2021-09-23
US9381247B2 (en) 2016-07-05
SG11201406491PA (en) 2014-11-27
EP2838506A1 (en) 2015-02-25
CY1123825T1 (en) 2022-05-27
EP3827813A1 (en) 2021-06-02
LT2838506T (en) 2021-03-25
HUE053303T2 (en) 2021-06-28
EP2838506B1 (en) 2021-01-06
KR101966484B1 (en) 2019-04-05
ZA201407410B (en) 2015-06-24
JP2015512952A (en) 2015-04-30
HRP20210417T1 (en) 2021-04-30
CA2869883A1 (en) 2013-10-24
SI2838506T1 (en) 2021-02-26
WO2013158618A1 (en) 2013-10-24
CN104394847A (en) 2015-03-04
HK1203371A1 (en) 2015-10-30
MX2014012245A (en) 2015-06-05
RS61533B1 (en) 2021-04-29
DK2838506T3 (en) 2021-01-18
KR20140146209A (en) 2014-12-24
PT2838506T (en) 2021-02-23
JP2019023223A (en) 2019-02-14
HK1207577A1 (en) 2016-02-05
US20140113856A1 (en) 2014-04-24
IL234987A0 (en) 2014-12-31
RU2014145846A (en) 2016-06-10
AU2013249495B2 (en) 2016-05-12
PL2838506T3 (en) 2021-06-28
JP6422855B2 (en) 2018-11-14

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