IN2014MN00976A - - Google Patents
Info
- Publication number
- IN2014MN00976A IN2014MN00976A IN976MUN2014A IN2014MN00976A IN 2014MN00976 A IN2014MN00976 A IN 2014MN00976A IN 976MUN2014 A IN976MUN2014 A IN 976MUN2014A IN 2014MN00976 A IN2014MN00976 A IN 2014MN00976A
- Authority
- IN
- India
- Prior art keywords
- amine
- alcohol
- solvent
- reaction
- preparation
- Prior art date
Links
- 239000004593 Epoxy Substances 0.000 abstract 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 229930182558 Sterol Natural products 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
- 150000003432 sterols Chemical class 0.000 abstract 1
- 235000003702 sterols Nutrition 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
The present invention relates to a process for the preparation of sterol derivatives comprising the reaction of an a epoxy compound with an amine in an alcohol comprising 3 to 5 carbon atoms as a solvent.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11306548 | 2011-11-24 | ||
| PCT/EP2012/073489 WO2013076257A1 (en) | 2011-11-24 | 2012-11-23 | Process for the preparation of sterol derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2014MN00976A true IN2014MN00976A (en) | 2015-04-24 |
Family
ID=47216329
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN976MUN2014 IN2014MN00976A (en) | 2011-11-24 | 2012-11-23 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US9447141B2 (en) |
| EP (1) | EP2782923B1 (en) |
| JP (1) | JP6157492B2 (en) |
| KR (1) | KR20140098131A (en) |
| CN (1) | CN104039807B (en) |
| AU (1) | AU2012342460B2 (en) |
| BR (1) | BR112014012458A2 (en) |
| CA (1) | CA2856609C (en) |
| ES (1) | ES2613753T3 (en) |
| IN (1) | IN2014MN00976A (en) |
| MX (1) | MX343787B (en) |
| RU (1) | RU2014125435A (en) |
| WO (1) | WO2013076257A1 (en) |
| ZA (1) | ZA201403736B (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3091970B1 (en) | 2014-01-10 | 2020-10-28 | Rgenix, Inc. | Lxr agonists and uses thereof |
| US11648220B2 (en) | 2016-01-11 | 2023-05-16 | The Rockefeller University | Methods for the treatment of myeloid derived suppressor cells related disorders |
| FR3064470A1 (en) * | 2017-03-31 | 2018-10-05 | Lessonia | MASK OR PATCH PREPARED FROM ALGINATE COMPOSITION |
| AU2018373028A1 (en) | 2017-11-21 | 2020-04-30 | Inspirna, Inc. | Polymorphs and uses thereof |
| WO2020061317A1 (en) * | 2018-09-19 | 2020-03-26 | Modernatx, Inc. | Sterol purification |
| BE1027157B9 (en) * | 2019-08-01 | 2020-11-03 | Dendrogenix | Composition of sterol derivatives for its use in the treatment of neuronal pathology linked to hypoxia and / or hypoglycemia and corresponding composition |
| EP4073025B1 (en) | 2019-12-13 | 2024-03-27 | Inspirna, Inc. | Metal salts and uses thereof |
| BE1028852B1 (en) * | 2020-12-03 | 2022-07-05 | Dendrogenix | 5α-Hydroxy-6β-[2-(1H-imidazol-4-yl)ethylamino]cholestan-3β-ol PRODRUG AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR USE IN THE TREATMENT OF CANCER |
| JP7849051B2 (en) * | 2020-10-29 | 2026-04-21 | デンドロゲニックス | 5α-hydroxy-6β-[2-(1H-imidazole-4-yl)ethylamino]-cholestane-3β-ol analogs and pharmaceutical compositions containing the same for use in the treatment of cancer |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2838741B1 (en) * | 2002-04-19 | 2006-01-27 | Inst Nat Sante Rech Med | STEROL DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS COMPRISING THE SAME |
-
2012
- 2012-11-23 IN IN976MUN2014 patent/IN2014MN00976A/en unknown
- 2012-11-23 MX MX2014006303A patent/MX343787B/en active IP Right Grant
- 2012-11-23 AU AU2012342460A patent/AU2012342460B2/en active Active
- 2012-11-23 RU RU2014125435/04A patent/RU2014125435A/en not_active Application Discontinuation
- 2012-11-23 WO PCT/EP2012/073489 patent/WO2013076257A1/en not_active Ceased
- 2012-11-23 EP EP12788589.5A patent/EP2782923B1/en active Active
- 2012-11-23 US US14/359,658 patent/US9447141B2/en active Active
- 2012-11-23 CA CA2856609A patent/CA2856609C/en active Active
- 2012-11-23 CN CN201280065737.0A patent/CN104039807B/en active Active
- 2012-11-23 JP JP2014542857A patent/JP6157492B2/en active Active
- 2012-11-23 BR BR112014012458A patent/BR112014012458A2/en not_active IP Right Cessation
- 2012-11-23 ES ES12788589.5T patent/ES2613753T3/en active Active
- 2012-11-23 KR KR1020147016187A patent/KR20140098131A/en not_active Withdrawn
-
2014
- 2014-05-22 ZA ZA2014/03736A patent/ZA201403736B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX2014006303A (en) | 2014-09-08 |
| CN104039807A (en) | 2014-09-10 |
| CA2856609A1 (en) | 2013-05-30 |
| MX343787B (en) | 2016-10-31 |
| EP2782923B1 (en) | 2016-11-23 |
| US20140309417A1 (en) | 2014-10-16 |
| CA2856609C (en) | 2021-01-12 |
| ZA201403736B (en) | 2015-11-25 |
| JP6157492B2 (en) | 2017-07-05 |
| KR20140098131A (en) | 2014-08-07 |
| WO2013076257A1 (en) | 2013-05-30 |
| JP2015502934A (en) | 2015-01-29 |
| ES2613753T3 (en) | 2017-05-25 |
| AU2012342460B2 (en) | 2017-06-29 |
| EP2782923A1 (en) | 2014-10-01 |
| AU2012342460A1 (en) | 2014-06-12 |
| CN104039807B (en) | 2018-02-13 |
| RU2014125435A (en) | 2015-12-27 |
| US9447141B2 (en) | 2016-09-20 |
| BR112014012458A2 (en) | 2017-06-06 |
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