IS2677B - A pharmaceutical composition comprising a pyrimidine-A-derived derivative coated with an acid polymer. - Google Patents

A pharmaceutical composition comprising a pyrimidine-A-derived derivative coated with an acid polymer.

Info

Publication number: IS2677B
Authority: IS; Iceland
Prior art keywords: pyrimidine; pharmaceutical composition; acid polymer; derived derivative; derivative coated
Prior art date: 2003-09-02

Application number

IS8366A

Other languages

Icelandic (is)

Other versions

IS8366A (en

Inventor

Dirk Marinus Johannes Van Schie

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-09-02

Filing date

2006-03-20

Publication date

2010-09-15

2006-03-20 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

2006-03-20 Publication of IS8366A publication Critical patent/IS8366A/en

2010-09-15 Publication of IS2677B publication Critical patent/IS2677B/en

Links

239000002253 acid Substances 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1
229920000642 polymer Polymers 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer

Landscapes

Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

IS8366A 2003-09-02 2006-03-20 A pharmaceutical composition comprising a pyrimidine-A-derived derivative coated with an acid polymer. IS2677B (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0320522.6A GB0320522D0 (en)	2003-09-02	2003-09-02	Formulation
PCT/EP2004/009726 WO2005021002A1 (en)	2003-09-02	2004-08-31	Pharmaceutical formulation comprising a pyrimidine-a-one derivative coated with an enteric polymer

Publications (2)

Publication Number	Publication Date
IS8366A IS8366A (en)	2006-03-20
IS2677B true IS2677B (en)	2010-09-15

Family

ID=28686767

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS8366A IS2677B (en)	2003-09-02	2006-03-20	A pharmaceutical composition comprising a pyrimidine-A-derived derivative coated with an acid polymer.

Country Status (30)

Country	Link
US (2)	US20060287346A1 (en)
EP (1)	EP1663243B1 (en)
JP (1)	JP4892346B2 (en)
KR (1)	KR101115984B1 (en)
CN (2)	CN1874778B (en)
AR (1)	AR045547A1 (en)
AT (1)	ATE422889T1 (en)
AU (1)	AU2004268376B2 (en)
BR (1)	BRPI0414038A (en)
CA (1)	CA2537178C (en)
CY (1)	CY1108953T1 (en)
DE (1)	DE602004019547D1 (en)
DK (1)	DK1663243T3 (en)
ES (1)	ES2319124T3 (en)
GB (1)	GB0320522D0 (en)
HR (1)	HRP20090147T3 (en)
IL (1)	IL173910A (en)
IS (1)	IS2677B (en)
MA (1)	MA28033A1 (en)
MX (1)	MXPA06002436A (en)
MY (1)	MY139165A (en)
NO (1)	NO333744B1 (en)
NZ (1)	NZ545453A (en)
PL (1)	PL1663243T3 (en)
PT (1)	PT1663243E (en)
RU (1)	RU2359660C2 (en)
SI (1)	SI1663243T1 (en)
TW (1)	TWI343257B (en)
WO (1)	WO2005021002A1 (en)
ZA (1)	ZA200601599B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0320522D0 (en) *	2003-09-02	2003-10-01	Glaxo Group Ltd	Formulation
BRPI0721697A2 (en)	2007-05-11	2014-08-05	Univ Jefferson	"METHODS FOR TREATING AND / OR PREVENTING NEURODEGENERATIVE DISEASE OR DISORDER IN AN INDIVIDUAL, TO TREAT AND / OR PREVENTING AN INDIVIDUAL WITH OR AT RISK OF VASCULAR DEMENTIA, TO TREAT AND / OR PREVENTING A BARRIERAL DISORDER OR DISORDER AN INDIVIDUAL, TO REDUCE BETA AMILOID ACCUMULATION IN THE BRAIN OF AN INDIVIDUAL, TO TREAT AND / OR PREVENT ALZHEIMER IN AN INDIVIDUAL AND TO PREVENT OR REDUCE THE RISK OF DEVELOPING ALZHHEIMER MISUSE, AND IN USE OF AND / OR LP-PLA2 PROTEIN ACTIVITY. "
US9029383B2 (en)	2007-05-11	2015-05-12	The Trustees Of The University Of Pennsylvania	Methods of treatment of skin ulcers
CA2759123C (en)	2009-04-24	2019-01-15	Iceutica Pty Ltd	Compositions of diclofenac acid with improved dissolution
EP2651403B1 (en)	2010-12-17	2020-12-02	Glaxo Group Limited	Use of lp-pla2 inhibitors in the treatment and prevention of eye diseases
WO2013082275A1 (en)	2011-11-30	2013-06-06	Trustees Of Boston College	Inhibitors of phosphodiesterases 11 (pde11) and methods of use to elevate cortisol production
US9526734B2 (en)	2014-06-09	2016-12-27	Iceutica Pty Ltd.	Formulation of meloxicam
EP3172211B1 (en)	2014-07-22	2019-07-03	GlaxoSmithKline Intellectual Property Development Limited	Tricyclic imidazo-pyrimidinone derivatives for the treatment of diseases mediated by lp-pla2
JP2026516205A (en)	2023-04-18	2026-05-20	サイニューロセラピューティクスインコーポレイテッド	Combination therapy with an LP-PLA2 inhibitor and a second drug

Family Cites Families (21)

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DE3619570C1 (en)	1986-06-11	1987-10-29	Kneipp Werke Kneipp Mittel Zen	Coated garlic tablet
US4971805A (en)	1987-12-23	1990-11-20	Teysan Pharmaceuticals Co., Ltd.	Slow-releasing granules and long acting mixed granules comprising the same
IT1227899B (en) *	1988-12-23	1991-05-14	Poli Ind Chimica Spa	TOTAL OR PARTIAL COATING OF PHARMACEUTICAL ACTIVE SUBSTANCES AND RELATED COMPOSITIONS
TW209174B (en)	1991-04-19	1993-07-11	Takeda Pharm Industry Co Ltd
JPH07223970A (en)	1994-02-10	1995-08-22	Tanabe Seiyaku Co Ltd	Release product in place in digestive tract
JP2917799B2 (en)	1994-03-11	1999-07-12	田辺製薬株式会社	Gastrointestinal tract release formulation
JP3185206B2 (en) *	1995-07-20	2001-07-09	田辺製薬株式会社	Lower digestive tract release coated capsule formulation
SG80553A1 (en)	1995-07-20	2001-05-22	Tanabe Seiyaku Co	Pharmaceutical preparation in form of coated capsule releasable at lower part of digestive tract
NZ333182A (en) *	1996-06-06	2000-03-27	Bifodan As	Enteric coating comprising alginic acid and a water soluble binding agent for an oral preparation
JP2000516222A (en) *	1996-08-15	2000-12-05	ロザンファルマゲゼルシャフトミットベシュレンクテルハフツング	Oral pharmaceutical composition that is easy to swallow
US6296876B1 (en) *	1997-10-06	2001-10-02	Isa Odidi	Pharmaceutical formulations for acid labile substances
PT1121103E (en) *	1998-05-18	2007-02-28	Takeda Pharmaceutical	Orally disintegrable tablets comprising a benzimidazole
WO2000028989A1 (en)	1998-11-12	2000-05-25	Smithkline Beecham P.L.C.	Pharmaceutical composition for modified release of an insulin sensitiser and another antidiabetic agent
US6268385B1 (en)	1999-08-26	2001-07-31	Robert R. Whittle	Dry blend pharmaceutical formulations
DE60139429D1 (en) *	2000-02-16	2009-09-10	Smithkline Beecham Plc	Pyrimidine-5-onderivatives as LDL-PLA2 inhibitors
AUPQ672800A0 (en) *	2000-04-06	2000-05-04	Natraherbal Pty Ltd	Garlic supplement for deodoriser
EP1294358B1 (en) *	2000-06-28	2004-08-18	Smithkline Beecham Plc	Wet milling process
JP5138856B2 (en) *	2001-06-20	2013-02-06	武田薬品工業株式会社	Tablet manufacturing method
ATE508725T1 (en)	2001-06-20	2011-05-15	Takeda Pharmaceutical	METHOD FOR PRODUCING TABLETS
RU2203671C1 (en) *	2002-03-25	2003-05-10	Общество С Ограниченной Ответственностью "Научно-Технологическая Фармацевтическая Фирма "Полисан"	Antiviral medicinal preparation for oral usage
GB0320522D0 (en) *	2003-09-02	2003-10-01	Glaxo Group Ltd	Formulation

2003
- 2003-09-02 GB GBGB0320522.6A patent/GB0320522D0/en not_active Ceased
2004
- 2004-08-31 AU AU2004268376A patent/AU2004268376B2/en not_active Ceased
- 2004-08-31 ES ES04764689T patent/ES2319124T3/en not_active Expired - Lifetime
- 2004-08-31 HR HR20090147T patent/HRP20090147T3/en unknown
- 2004-08-31 CN CN2004800325934A patent/CN1874778B/en not_active Expired - Fee Related
- 2004-08-31 NZ NZ545453A patent/NZ545453A/en not_active IP Right Cessation
- 2004-08-31 RU RU2006110546/15A patent/RU2359660C2/en not_active IP Right Cessation
- 2004-08-31 SI SI200431087T patent/SI1663243T1/en unknown
- 2004-08-31 CA CA2537178A patent/CA2537178C/en not_active Expired - Fee Related
- 2004-08-31 AT AT04764689T patent/ATE422889T1/en active
- 2004-08-31 WO PCT/EP2004/009726 patent/WO2005021002A1/en not_active Ceased
- 2004-08-31 PT PT04764689T patent/PT1663243E/en unknown
- 2004-08-31 CN CN201110102640XA patent/CN102204891B/en not_active Expired - Fee Related
- 2004-08-31 EP EP04764689A patent/EP1663243B1/en not_active Expired - Lifetime
- 2004-08-31 DE DE602004019547T patent/DE602004019547D1/en not_active Expired - Lifetime
- 2004-08-31 BR BRPI0414038-9A patent/BRPI0414038A/en not_active Application Discontinuation
- 2004-08-31 AR ARP040103126A patent/AR045547A1/en unknown
- 2004-08-31 DK DK04764689T patent/DK1663243T3/en active
- 2004-08-31 US US10/570,335 patent/US20060287346A1/en not_active Abandoned
- 2004-08-31 PL PL04764689T patent/PL1663243T3/en unknown
- 2004-08-31 JP JP2006525098A patent/JP4892346B2/en not_active Expired - Fee Related
- 2004-08-31 TW TW093126106A patent/TWI343257B/en not_active IP Right Cessation
- 2004-08-31 MX MXPA06002436A patent/MXPA06002436A/en active IP Right Grant
- 2004-08-31 KR KR1020067004235A patent/KR101115984B1/en not_active Expired - Fee Related
- 2004-09-01 MY MYPI20043561A patent/MY139165A/en unknown
2006
- 2006-02-23 IL IL173910A patent/IL173910A/en not_active IP Right Cessation
- 2006-02-23 ZA ZA200601599A patent/ZA200601599B/en unknown
- 2006-03-10 MA MA28866A patent/MA28033A1/en unknown
- 2006-03-20 IS IS8366A patent/IS2677B/en unknown
- 2006-04-03 NO NO20061514A patent/NO333744B1/en not_active IP Right Cessation
2009
- 2009-04-08 CY CY20091100412T patent/CY1108953T1/en unknown
- 2009-06-05 US US12/478,934 patent/US8772303B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
MY139165A (en)	2009-08-28
AU2004268376B2 (en)	2010-04-22
BRPI0414038A (en)	2006-10-24
RU2359660C2 (en)	2009-06-27
EP1663243B1 (en)	2009-02-18
IL173910A (en)	2010-11-30
IS8366A (en)	2006-03-20
CN1874778B (en)	2011-06-22
TWI343257B (en)	2011-06-11
IL173910A0 (en)	2006-07-05
ATE422889T1 (en)	2009-03-15
PL1663243T3 (en)	2009-07-31
KR20060118422A (en)	2006-11-23
US20090306113A1 (en)	2009-12-10
NZ545453A (en)	2009-12-24
CN102204891B (en)	2013-08-21
NO333744B1 (en)	2013-09-09
AU2004268376A1 (en)	2005-03-10
CN1874778A (en)	2006-12-06
EP1663243A1 (en)	2006-06-07
JP4892346B2 (en)	2012-03-07
CY1108953T1 (en)	2014-07-02
DK1663243T3 (en)	2009-05-04
MA28033A1 (en)	2006-07-03
KR101115984B1 (en)	2012-03-13
RU2006110546A (en)	2006-08-10
NO20061514L (en)	2006-04-03
HK1091734A1 (en)	2007-01-26
HRP20090147T3 (en)	2009-04-30
JP2007504195A (en)	2007-03-01
US8772303B2 (en)	2014-07-08
CA2537178A1 (en)	2005-03-10
GB0320522D0 (en)	2003-10-01
DE602004019547D1 (en)	2009-04-02
TW200517113A (en)	2005-06-01
ZA200601599B (en)	2007-05-30
SI1663243T1 (en)	2009-06-30
PT1663243E (en)	2009-04-27
MXPA06002436A (en)	2006-06-20
AR045547A1 (en)	2005-11-02
CA2537178C (en)	2013-03-19
US20060287346A1 (en)	2006-12-21
ES2319124T3 (en)	2009-05-04
CN102204891A (en)	2011-10-05
WO2005021002A1 (en)	2005-03-10

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